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N-(furan-2-ylmethyl)-3-[4-(pyridin-3-yloxy)piperidin-1-yl]propanamide
N-benzyl-N-methyl-3-[(2-methylpyrrolidin-1-yl)methyl]imidazo[1,2-a]pyridine-2-carboxamide
3-{2-[2-(thiophen-2-yl)ethyl]piperidine-1-carbonyl}phenol
(1S,6R)-3-{2-[4-(2-methylphenyl)-1,4-diazepan-1-yl]-2-oxoethyl}-3,9-diazabicyclo[4.2.1]nonan-4-one
5-methoxy-4-(1-methyl-1H-pyrazol-5-yl)-N-[1-(thiophen-3-yl)propan-2-yl]pyrimidin-2-amine
1-{5H,6H-benzo[h]quinazolin-2-yl}-5-cyclopropyl-N-[3-(pyridin-3-yloxy)propyl]-1H-pyrazole-4-carboxamide
4-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]-2-methylphenol
{[1-(2-methoxyethyl)piperidin-4-yl]methyl}[(3-methyl-1H-pyrazol-5-yl)methyl](pyridin-4-ylmethyl)amine
7-(methylsulfanyl)-3-{[4-(pyrrolidin-1-yl)piperidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
ethyl 5-{2-oxo-1,2-dihydrospiro[indole-3,4'-piperidine]-1'-ylmethyl}furan-2-carboxylate
2-[3-methyl-5-oxo-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N-[(1r,4r)-4-hydroxycyclohexyl]acetamide
(5S,9aS,9bS)-2-[(4-methoxyphenyl)methyl]-5-(3-methyl-1-propyl-1H-pyrazol-4-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-(pent-2-yn-1-yl)-2,8-diazaspiro[4.5]decan-3-one
2-amino-4-[2-(dimethylamino)pyrimidin-5-yl]-6-(2,5-dimethylthiophen-3-yl)pyridine-3-carbonitrile
3-{[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}pyridine
1-{4-[(dimethylamino)methyl]-2-methoxyphenoxy}-3-(thiomorpholin-4-yl)propan-2-ol
N-butyl-5-(4-cyclopentylpiperazine-1-carbonyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
4-[(4-methyl-5-{1-[(2-methyl-1,3-oxazol-4-yl)methyl]piperidin-3-yl}-4H-1,2,4-triazol-3-yl)methyl]morpholine
2-(6-chloro-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}imidazo[1,2-a]pyridine-2-carbonyl)-1,2,3,4-tetrahydroisoquinoline
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-{1-[3-(1,2-oxazolidin-2-yl)propanoyl]piperidin-4-yl}propanamide
N-(4-{4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl}phenyl)ethane-1-sulfonamide
6-[2-(aminomethyl)-2,3-dihydro-1-benzofuran-7-yl]pyrimidin-4-amine
1-(cyclopropylmethyl)-N-ethyl-5-[(5-methylfuran-2-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2,2-dimethyl-N-(1-{1-[2-(pyridin-2-yl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)propanamide
3-[4-(propan-2-yl)phenyl]-3-[(pyrimidin-4-yl)amino]propan-1-ol
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-({[(6-hydroxypyrimidin-4-yl)methyl]amino}methyl)piperidin-2-one
(5S,9aS,9bS)-2-(3-methoxyphenyl)-5-(1-methyl-1H-pyrazol-4-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-4-(4-methoxyphenyl)butan-1-one
({5-[3-cyclopropyl-1-(2-methoxyphenyl)-1H-1,2,4-triazol-5-yl]furan-2-yl}methyl)dimethylamine
(4aS,7aR)-1-(4-hydroxybenzoyl)-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[2-(naphthalen-1-yl)ethyl]-5-oxopyrrolidine-3-carboxylic acid
1-benzyl-3-({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)-3-methylurea
N-(piperidin-4-yl)-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
8-[2-(3,4-dimethylphenoxy)acetyl]-2-(3-methoxypropyl)-2,8-diazaspiro[4.5]decan-3-one
7-(3-methoxypropyl)-2-(2-methylquinolin-4-yl)-2,7-diazaspiro[4.5]decan-6-one
1-{4-[(cyclohexylamino)methyl]-2-methoxyphenoxy}-3-(thiomorpholin-4-yl)propan-2-ol
6-(2,3,4-trimethoxyphenyl)quinoline
1-(1,3-benzothiazol-2-yl)-N-{[2-(2-methylphenyl)pyrimidin-5-yl]methyl}piperidin-3-amine
4-[3-(2,5-dimethyl-1H-pyrrol-1-yl)-4,5-dimethylthiophene-2-carbonyl]piperazin-2-one
2-[(1S,5R)-6-[2-(2,4-dimethoxyphenyl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
(3aS,6aR)-5-(3,6-dimethylpyrazin-2-yl)-3-(pyridin-2-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
3-[2-(azocan-1-yl)-2-oxoethyl]-4-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-2-one
N-(3-cyano-4-methoxyphenyl)-4-[2-(pyrrolidin-1-yl)ethyl]piperazine-1-carboxamide
(3aR,6aR)-2-(prop-2-en-1-yl)-5-(pyridine-3-sulfonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(2,3-difluoro-4-methylphenyl)methyl]-2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-methyl-2-[3-(2-methylphenyl)-2,5-dioxo-1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]-N-(1-methylpiperidin-4-yl)acetamide
2-methyl-2-(methylamino)-N-({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)propanamide
2-(3,4-difluorophenyl)-8-methoxy-5-[(6-methylpyridin-2-yl)methyl]-2,3,4,5-tetrahydro-1,5-benzothiazepine
2-{[4-(1H-indol-2-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-4-methylphenol
N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide