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2-ethyl-9-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-4-phenyl-2,9-diazaspiro[5.5]undecane
1-(1-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-3-yl)-3,5-dimethyl-1H-pyrazole
N-[2-(4-{[cyclohexyl(methyl)amino]methyl}phenoxy)propyl]-3-fluorobenzamide
N-cyclopropyl-3-{5-[(5-methylthiophen-2-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
4-{[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}-1,4-oxazepane
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N,N-dimethyl-1-{[1-(2-methylpropyl)-2-phenylmethanesulfonyl-1H-imidazol-5-yl]methyl}pyrrolidin-3-amine
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-3-(1H-1,2,4-triazol-1-yl)propanamide
6-methyl-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-2-(morpholin-4-yl)pyrimidin-4-amine
2-(3,4-dichlorophenyl)-4-(3,3,4,4-tetrafluorobutyl)morpholine
dimethyl[1-(4-{1-[2-(pyridin-3-yl)ethyl]-1H-1,2,3-triazol-4-yl}phenyl)ethyl]amine
3-{[(4-fluorophenyl)methyl]sulfanyl}-N-[1-(1-methyl-1H-1,2,4-triazol-5-yl)propyl]propanamide
3-{1-[(dimethyl-1,2-oxazol-4-yl)methyl]piperidin-3-yl}-1-methyl-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]-N-methylpyrrolidine-2-carboxamide
3-[(4-methoxyphenyl)methyl]-1-methyl-8-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(2-methoxyphenoxy)-N-{[1-(morpholine-4-carbonyl)piperidin-3-yl]methyl}acetamide
(4aS,7aR)-N-(3-chlorophenyl)-4-cyclopropanecarbonyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
4-[(3-{3-[cyclohexyl(methyl)amino]-2-hydroxypropoxy}phenyl)methyl]-1-methylpiperazin-2-one
2-[1-(2-methylpropyl)-3-oxopiperazin-2-yl]-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]acetamide
2-(phenylamino)-N-[2-(pyrrolidin-1-yl)ethyl]pyrimidine-5-carboxamide
2-(2-methoxyethyl)-8-{[3-(methylsulfanyl)phenyl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
N-(1-methoxybutan-2-yl)-4-[(pyridin-2-ylsulfanyl)methyl]benzamide
2-(2-hydroxyethyl)-8-[3-(1H-pyrrol-1-yl)propyl]-2,8-diazaspiro[5.5]undecan-3-one
1-[4-(4-fluorophenyl)piperazin-1-yl]-3-(pyrazin-2-yl)propan-1-one
N-[(2,3-dimethylphenyl)methyl]-4-[(2-methylpyridin-3-yl)oxy]piperidine-4-carboxamide
4-(3-methyl-1-propyl-1H-pyrazol-4-yl)-N-[(2R)-oxolan-2-ylmethyl]pyrimidin-2-amine
1'-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-2-(2-phenyl-1H-imidazol-1-yl)acetamide
(2R,6R)-4-[(3-ethyl-1,2-oxazol-5-yl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
5-{3-[(4-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}-N-methyl-N-(pyridin-3-ylmethyl)pyridin-2-amine
2-amino-N-[(5-chloro-2-methoxyphenyl)methyl]-2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-methylacetamide
6-hydroxy-N-{2-[2-(pyridin-2-yl)ethoxy]phenyl}-1,4-oxazepane-4-carboxamide
N-(1H-indazol-5-yl)-4-(3-phenylpropyl)-1,4-diazepane-1-carboxamide
2-chloro-N-(1-{1-[(4-acetamidophenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
1-methyl-6-oxo-N-(2-propoxypropyl)-1,6-dihydropyridine-3-carboxamide
N-(3-hydroxy-2,2-dimethylpropyl)-2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
2-(1H-pyrazol-4-yl)-4-[2-(1,3-thiazol-2-yl)piperidine-1-carbonyl]quinoline
N-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)-2-(pyridin-4-ylsulfanyl)acetamide
3,5,7-trimethyl-2-(3-phenylpiperazine-1-carbonyl)-1H-indole
N,5-dimethyl-2-phenyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}furan-3-carboxamide
N-(2H-1,3-benzodioxol-5-yl)-1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidin-3-amine
2-(3,3-diethylpyrrolidin-1-yl)-5-[3-(methoxymethyl)piperidine-1-carbonyl]pyridine
N-[2-(2-ethoxyphenoxy)ethyl]-4-ethyl-N,5-dimethylthiophene-3-carboxamide
4-[2-(2-methoxyphenyl)pyrrolidine-1-carbonyl]-1-phenyl-1H-1,2,3-triazole
(3R,4S)-4-propyl-1-[4-(trifluoromethyl)pyridin-2-yl]pyrrolidin-3-amine
N-[(3S,4R)-1-[3-(3-fluorophenyl)propanoyl]-4-propylpyrrolidin-3-yl]methanesulfonamide
(3R,4S)-4-{4-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]-1,4-diazepan-1-yl}oxolan-3-ol
1-(6-hydroxy-4-{[3-(morpholin-4-yl)phenyl]methyl}-1,4-diazepan-1-yl)propan-1-one
2,2-dimethyl-3-{[1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}propan-1-ol