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N-(cyclohexylmethyl)-5-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
({3-[(1-{3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}piperidin-4-yl)oxy]phenyl}methyl)(furan-3-ylmethyl)methylamine
[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]({[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl})methylamine
4-[(dimethylamino)methyl]-1-(5-propyl-1,3,4-oxadiazol-2-yl)azepan-4-ol
3-[4-(1-methyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]-1-(pyrrolidin-1-yl)propan-1-one
methyl 2-chloro-5-{[(2-methoxyethyl)(1,3-thiazol-2-ylmethyl)carbamoyl]amino}benzoate
4-[(4-cyclopentyl-1H-1,2,3-triazol-1-yl)methyl]-1-(1,3-thiazole-4-carbonyl)piperidine
(3,3-diphenylpropyl)({[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
N-(oxan-4-ylmethyl)-6-(piperidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
ethyl 4-benzyl-1-[(2,4,5-trimethoxyphenyl)methyl]piperidine-4-carboxylate
3-[2-(2,6-difluorophenyl)ethyl]-N-(propan-2-yl)piperidine-1-carboxamide
1-methanesulfonyl-4-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]-1,4-diazepane
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-4-{[(3-phenoxyphenyl)methyl]amino}-1-(propan-2-yl)pyrrolidine-2-carboxamide
4-({4-[3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl]furan-2-yl}methyl)morpholine
4-(4-fluorophenyl)-1-[3-(3-hydroxy-3-methylbutyl)benzoyl]piperidin-4-ol
2-ethyl-9-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]-2,9-diazaspiro[5.5]undecan-3-one
N,2,3,5-tetramethyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
4-methyl-1-{[1-(oxolan-2-ylmethyl)-2-(propane-1-sulfonyl)-1H-imidazol-5-yl]methyl}piperidine
N-{[4-(2,3-dihydro-1H-inden-2-yloxy)-3-methoxyphenyl]methyl}-2,4-difluoro-N-(oxolan-2-ylmethyl)benzene-1-sulfonamide
ethyl 4-[(3-methoxyphenyl)methyl]-1-(1H-pyrazol-3-ylmethyl)piperidine-4-carboxylate
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-4-(2-oxopyrrolidin-1-yl)butanamide
{[(1-cycloheptylpyrrolidin-3-yl)methyl]sulfamoyl}(ethyl)methylamine
N,N-diethyl-3-methyl-4-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)benzamide
4-(2-phenylpropyl)-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
methyl[(1-methyl-1H-indol-2-yl)methyl][(3-methylpyridin-4-yl)methyl]amine
N-(2-hydroxyethyl)-5-(3-methylbut-2-en-1-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
1-[1-(4-methoxypyrimidin-2-yl)piperidin-4-yl]-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide
N-{[7-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,3,4,9-tetrahydro-1H-carbazole-1-carboxamide
N3-cycloheptyl-1-cyclopropyl-4-oxo-N5-[(4-phenyl-1,3-thiazol-2-yl)methyl]-1,4-dihydropyridine-3,5-dicarboxamide
4-{[(2-methoxyphenyl)methyl]amino}-5-methyl-N-(prop-2-en-1-yl)thieno[2,3-d]pyrimidine-6-carboxamide
1-{[5-(1-methanesulfonylpiperidin-4-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}azepane
N-cyclohexyl-1-(2-methoxyphenyl)-N-(pyridin-2-ylmethyl)-1H-pyrazole-4-carboxamide
N-[2-(N-methylmethanesulfonamido)ethyl]-2-(2-phenyl-1,3-thiazol-4-yl)acetamide
N-[(8-methoxyquinolin-5-yl)methyl]-N,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
2-(2-cyclopropyl-1H-1,3-benzodiazol-1-yl)-N-methyl-N-[(3-methylpyridin-4-yl)methyl]acetamide
2-[(4aR,7aS)-4-[2-(dimethylamino)benzoyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]acetic acid
4-{[2-(2,3-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-ethylpiperazin-2-one
2-{5-[1-(2H-1,3-benzodioxol-5-yl)propan-2-yl]-4-phenyl-1H-imidazol-1-yl}ethan-1-ol
2-{3-[(3,4-dimethoxyphenyl)methyl]-5-(2,5-dimethylfuran-3-yl)-1H-1,2,4-triazol-1-yl}ethan-1-ol
4-{3-fluoro-5-methylimidazo[1,2-a]pyridine-2-carbonyl}-1-(2-methylphenyl)piperazin-2-one
[(1-cyclopentylpiperidin-4-yl)methyl][(4-ethoxyphenyl)methyl](oxolan-2-ylmethyl)amine
4-[(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)amino]-1λ4-thian-1-one
N-[(5-ethylpyridin-2-yl)methyl]-N-methyl-1,3-dioxo-2-propyl-2,3-dihydro-1H-isoindole-5-carboxamide
2-(3,4-dimethylphenoxy)-1-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
N-(4-hydroxybutyl)-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
3-[(3S,4R)-1-[(4-chlorophenyl)methyl]-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]propanamide
N-[(4-{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethoxy}-3-methoxyphenyl)methyl]-5,6-dimethyl-2-oxo-N-[(3S)-2-oxoazepan-3-yl]-1,2-dihydropyridine-3-carboxamide
5-[1-cyclohexyl-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]-3,4-dihydropyrimidin-4-one
3-(3-tert-butyl-1-methyl-1H-pyrazol-5-yl)-1-cyclopropyl-1-{[4-(methylsulfanyl)phenyl]methyl}urea
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide