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7-(2-amino-5,6,7,8-tetrahydroquinazoline-4-carbonyl)-1-oxa-3,7-diazaspiro[4.5]decan-2-one
3-{[1-(2-methylpropyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}pyridine
3-benzyl-1-methyl-8-{[3-(2-methylphenyl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-methyl-2-[4-oxo-8-(trifluoromethyl)-3,4-dihydroquinazolin-3-yl]acetamide
2-{4-[(4-chloro-3-fluorophenyl)methyl]-2-oxopiperazin-1-yl}benzonitrile
3-(1-methyl-1H-pyrrol-2-yl)-N-[(5-methylpyrazin-2-yl)methyl]-1H-pyrazole-5-carboxamide
N-(9H-fluoren-9-yl)-2-[1-(3-methoxypropyl)-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]acetamide
6-[(3-aminopyrrolidin-1-yl)methyl]-N-({2-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-5-methyl-1-propyl-1H-pyrazole-4-carboxamide
(1R,3S,5S)-8-[5-(propan-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl]-8-azabicyclo[3.2.1]octan-3-ol
2-(dimethylamino)-N-[2-(ethylsulfanyl)ethyl]-2-(2-fluorophenyl)acetamide
2-methoxy-5-{3-[2-(pyridin-4-yl)pyridin-4-yl]pyrrolidine-1-carbonyl}pyrimidine
N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetamide
2-(3-methoxypropyl)-8-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2,8-diazaspiro[4.5]decan-3-one
1-ethyl-3-{[3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}piperidine
1-cyclohexyl-3-[2-(methylsulfanyl)ethyl]-5-{[1,2,3,4]tetrazolo[1,5-a]pyridin-7-yl}-1H-1,2,4-triazole
4-({[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]carbamoyl}amino)-N-(oxolan-2-ylmethyl)benzamide
[(3R,4R)-1-(3-methoxy-2-methylbenzoyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-4-({[4-(methylsulfanyl)phenyl]methyl}amino)-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
1-[3-(2-oxopyrrolidin-1-yl)propyl]-5-[4-(thiophene-2-carbonyl)piperazine-1-carbonyl]piperidin-2-one
2-[4-(1H-indol-3-ylmethyl)-1-(propan-2-yl)piperazin-2-yl]ethan-1-ol
N-(3,4-difluorophenyl)-1-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)piperidin-3-amine
2-(2-{[(3R,4R)-3-hydroxy-4-(pyridine-2-amido)piperidin-1-yl]methyl}phenoxy)acetic acid
6-[(2-butyl-1H-imidazol-4-yl)methyl]-1-[(2E)-3-phenylprop-2-en-1-yl]-3-(pyridin-4-yl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N-(cyclobutylmethyl)-5-methyl-N-(oxolan-2-ylmethyl)-2-phenyl-1H-imidazole-4-carboxamide
(3aR,6aR)-2-(prop-2-en-1-yl)-5-[(propan-2-yl)carbamoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(5-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepane-1-carbonyl}-1H-pyrazol-3-yl)ethan-1-one
4-({5-[1-(3-cyclopentylpropyl)piperidin-3-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)morpholine
2-[(2-{1-[5-(methoxymethyl)furan-2-carbonyl]piperidin-3-yl}-1H-imidazol-1-yl)methyl]pyridine
N-methyl-2-[(propan-2-yl)amino]-N-[2-(2,3,6-trimethylphenoxy)ethyl]pyrimidine-5-carboxamide
1-(4-{[4-(1-phenylcyclopropanecarbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperazin-1-yl)ethan-1-one
1-ethyl-4-{3-[2-(3-methoxyphenyl)ethyl]piperidine-1-carbonyl}piperidine
[(3R,4R)-4-(azepan-1-ylmethyl)-1-(2,3-dimethoxybenzoyl)pyrrolidin-3-yl]methanol
(1S,5R)-6-[(1,4-dimethyl-1H-pyrazol-5-yl)methyl]-1,3,3-trimethyl-6-azabicyclo[3.2.1]octane
1-[2-(2,2-diphenylethyl)morpholin-4-yl]propan-1-one
2-(dimethylamino)-2-(4-methylphenyl)-N-[2-(1H-pyrrol-1-yl)ethyl]acetamide
N-benzyl-5-(pyrrolidin-2-yl)-N-(1,3-thiazol-2-ylmethyl)thiophene-2-carboxamide
6-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
3-(4-ethyl-1H-pyrazol-5-yl)-1-{3-methyl-3H-[1,2,3]triazolo[4,5-b]pyridine-6-carbonyl}piperidine
4-[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl]piperidine
2-amino-2-methyl-1-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)propan-1-one
{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}[(5-methylpyrazin-2-yl)methyl]amine
1-(1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carbonyl)piperidin-3-ol
methyl 3-[2-oxo-6-(pyridin-4-ylmethoxy)-4-(pyridine-2-carbonyl)-1,4-diazepan-1-yl]propanoate
N-methyl-2-oxo-N-[2-(pyridin-2-yl)ethyl]-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
2-{4-[2-amino-6-(cyclopropylamino)pyrimidin-4-yl]-1-(thiophen-2-ylmethyl)piperazin-2-yl}ethan-1-ol
(3S,4R)-3-benzyl-4-methyl-1-(1-methyl-1H-indazole-3-carbonyl)piperidin-4-ol
1-[4-(4-fluorophenyl)-4-hydroxypiperidin-1-yl]-4-(1H-pyrazol-4-yl)butan-1-one
2-(2,5-dimethoxyphenyl)-1-[9-methoxy-7-(6-methoxypyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)quinoline-3-carboxamide