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N-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-1-methyl-1H-1,3-benzodiazole-5-carboxamide
N-ethyl-2-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-oxopiperazin-2-yl}-N-(2-methylprop-2-en-1-yl)acetamide
1-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
1-[(1R,5S,6R)-6-{[methyl(1,2-oxazol-5-ylmethyl)amino]methyl}-3-azabicyclo[3.1.0]hexan-3-yl]-2-phenoxyethan-1-one
4-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-2,6-dimethoxypyrimidine
N-(1-{1-[(4-methoxy-2,5-dimethylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopropanecarboxamide
N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-1-(2-phenylethyl)piperidin-3-amine
2-(4-methoxyphenyl)-N-[(1-{5-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidin-3-yl)methyl]acetamide
N-(1-{[4-(butan-2-yloxy)-3-chlorophenyl]methyl}piperidin-4-yl)methanesulfonamide
2-({2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}amino)-N-(pyrazin-2-yl)acetamide
1-{[(3R,4R)-4-(hydroxymethyl)-1-[6-methyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]pyrrolidin-3-yl]methyl}piperidin-4-ol
5-methyl-N2-[(1-phenyl-1H-pyrazol-4-yl)methyl]pyrimidine-2,4-diamine
ethyl 1-[(5-chlorothiophen-2-yl)sulfonyl]-4-(oxan-2-ylmethyl)piperidine-4-carboxylate
N-[(3R,4S)-1-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]-2-methoxy-2-methylpropanamide
3-[2-(dimethylamino)ethyl]-5-[1-(2,5-dimethylbenzoyl)piperidin-4-yl]-5-(2-phenylethyl)imidazolidine-2,4-dione
9-[(2,2-dimethyloxan-4-yl)methyl]-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-({3-methoxy-4-[2-(pyridin-2-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]benzamide
6-methyl-2-{2-[2-(6-methylpyridin-2-yl)-1H-imidazol-1-yl]ethyl}-3,4-dihydropyrimidin-4-one
(4aS,8aR)-6-[(5-ethylfuran-2-yl)methyl]-1-[2-(1H-imidazol-4-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
N-benzyl-N-[2-(dimethylamino)ethyl]-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propanamide
1-(3-methylpyridin-2-yl)-4-[1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperazine
2-({4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}methyl)quinolin-8-ol
2-(6-chloro-2H-1,3-benzodioxol-5-yl)-1-[3-(1H-imidazol-1-yl)propyl]-1H-imidazole
4-(5-chloro-2-methoxyphenyl)-3-(pyridin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
ethyl 5-{[(2-hydroxyethyl)(methyl)amino]methyl}-1-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]-1H-pyrazole-4-carboxylate
1-ethyl-N-[(3S,5S)-5-(ethylcarbamoyl)-1-(prop-2-en-1-yl)pyrrolidin-3-yl]-1H-pyrazole-4-carboxamide
N-(2-methoxy-2-methylpropyl)-6-(4-methylphenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
2-[2-methoxy-5-(pyrrolidin-1-ylmethyl)phenoxy]-6-methyl-4-(trifluoromethyl)pyridine
2-[1-({1-[4-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}methyl)-1H-1,2,3-triazol-4-yl]ethan-1-ol
4-{[5-fluoro-2-(trifluoromethyl)phenyl]methyl}-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
(4aS,7aR)-1-[5-(methoxymethyl)furan-2-carbonyl]-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-[1-(2,5-difluorobenzoyl)pyrrolidin-2-yl]-3-phenyl-1,2,4-oxadiazole
1-methyl-2-[1-(oxolane-2-carbonyl)piperidin-4-yl]-1H-1,3-benzodiazole
N-cyclopentyl-5-[4-(2-methoxyphenyl)piperazine-1-carbonyl]-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
1-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}-4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidine
3-[1-(5-ethyl-1,2-oxazole-3-carbonyl)piperidin-3-yl]-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
6-{4-[(2-methoxyphenyl)methyl]piperazine-1-carbonyl}-N-(3-methoxypropyl)-5-methylthieno[2,3-d]pyrimidin-4-amine
5-{4-[4-(propan-2-yl)piperazin-1-yl]phenyl}pyrazin-2-amine
2-[2-methyl-4-oxo-1-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indol-3-yl]-N-(prop-2-en-1-yl)acetamide
N-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)-1-[2-(morpholin-4-yl)ethyl]-6-oxopiperidine-3-carboxamide
(3aR,5S,6S,7aS)-2-[(2-methyl-1,3-benzothiazol-6-yl)sulfonyl]-octahydro-1H-isoindole-5,6-diol
3-{2-[4-(1,3-benzoxazol-2-yl)piperazin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
2-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-2,7-diazaspiro[4.5]decane
N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}quinoxalin-2-amine
7-{imidazo[1,2-b]pyridazine-3-carbonyl}-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
3-{[1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}-N-(1,3-thiazol-2-yl)propanamide
2-[3-(3-methoxyphenyl)-1H-pyrazol-1-yl]-N-[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]acetamide
4-[2-(1,4-oxazepan-4-yl)-2-oxoethyl]-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
2-(1-{[5-chloro-1-methyl-3-(5-methyl-1,2-oxazol-3-yl)-1H-pyrazol-4-yl]methyl}pyrrolidin-2-yl)pyridine
N-{1-[1-(1,3-benzothiazol-2-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-phenylacetamide