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3-(3-fluorophenyl)-N-[2-(4-methyl-5-{[2-(morpholin-4-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl)ethyl]benzamide
1,3-dimethyl-5-[1-(1-phenylethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-1H-pyrazole
2-[3-(2-methylpiperidin-1-yl)azetidine-1-carbonyl]thiophene-3-sulfonamide
N-[2-(1H-imidazol-4-yl)ethyl]-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
4-{2-[cyclohexyl(methyl)amino]propanoyl}-1-phenylpiperazin-2-one
2-({[(3-chlorophenyl)methyl]amino}methyl)-4-phenylphenol
N-(2-oxo-2,3-dihydro-1H-indol-5-yl)-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carboxamide
3-[(3S,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidine-1-carbonyl]-1-methyl-1,2-dihydropyridin-2-one
N-ethyl-2-[4-(2-methoxy-2-phenylacetyl)piperazin-1-yl]acetamide
5-[(4-ethylpiperazin-1-yl)methyl]-N-({5-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1,2-oxazole-3-carboxamide
{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[1-(1,3-thiazol-2-yl)ethyl]amine
9-(2-hydroxy-4-methylbenzoyl)-2-(2-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
(2R,3R,6R)-5-(3-fluoropyridine-4-carbonyl)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[2-(5-ethyl-1,2,4-oxadiazol-3-yl)ethyl]-2-(furan-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N4-[(1,4-dimethylpiperazin-2-yl)methyl]-2-{[(4-methylphenyl)methyl]sulfanyl}pyrimidine-4,6-diamine
ethyl 1-(6-methylpyridine-2-carbonyl)-4-(2-phenylethyl)piperidine-4-carboxylate
(3S,5R,9R)-11-{[1-(2-chlorophenyl)-1H-pyrazol-4-yl]methyl}-5-hydroxy-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
1-methyl-8-[(5-methylfuran-2-yl)methyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
(3aR,6aR)-2-(cyclobutylmethyl)-5-(4,4,4-trifluorobutanoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[5-fluoro-4-(morpholin-4-yl)pyrimidin-2-yl]-N-methylpyrrolidine-3-carboxamide
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-1-(difluoromethyl)-1H-pyrazole-5-carboxamide
1-(2,3-dihydro-1-benzofuran-5-carbonyl)-4-(2-methyl-1H-imidazol-1-yl)piperidine-4-carboxylic acid
2-[(2-amino-6-{4-[1-(morpholin-4-yl)ethyl]phenyl}pyrimidin-4-yl)amino]ethan-1-ol
4-methoxy-3-(oxan-2-ylmethyl)benzamide
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]benzamide
3-(5-{spiro[azepane-4,2'-chromene]-1-ylmethyl}thiophen-3-yl)prop-2-yn-1-ol
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-5-propyl-1,2-oxazole-3-carboxamide
N-[3-(2-ethylphenoxy)propyl]-N-methyl-3-(4H-1,2,4-triazol-4-yl)benzamide
(1S,5R)-6-{3-fluoro-5-methylimidazo[1,2-a]pyridine-2-carbonyl}-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane
2,6,6-trimethyl-3-[2-(1,2-oxazinan-2-yl)-2-oxoethyl]-1-(propan-2-yl)-4,5,6,7-tetrahydro-1H-indol-4-one
3-[(3S,4R)-1-[(4-chlorophenyl)methyl]-4-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-3-yl]-1-(piperidin-1-yl)propan-1-one
N-[3-hydroxy-2-(thiophen-2-ylmethyl)propyl]pyridine-3-carboxamide
2-(3-methylphenyl)-1-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
2-({3-[(3,4-difluorophenyl)amino]piperidin-1-yl}methyl)-3-methoxyphenol
1-cyclohexyl-N-[2-(4-fluorophenyl)-2-hydroxyethyl]piperidine-4-carboxamide
N-{[5-(4-fluorophenyl)furan-2-yl]methyl}-1-propanoylpiperidine-3-carboxamide
3-[(2-methyl-1,3-oxazol-4-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(1-butyl-1H-imidazol-2-yl)-1-(3-phenyl-1H-pyrazole-4-carbonyl)piperidine
3-[5-(3-fluoro-2,4-dimethylphenyl)-4-phenyl-1H-imidazol-1-yl]propan-1-ol
2-{[5-(2-chloro-4-methoxyphenoxymethyl)-1H-pyrazol-3-yl]formamido}-N-methylpropanamide
N-ethyl-7-[(thiophen-2-ylmethyl)sulfamoyl]-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
{[1-benzyl-2-(2-methoxyethanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)(1,2-oxazol-5-ylmethyl)amine
2-[(3-methoxyphenyl)amino]-N-[2-(pyridin-2-ylsulfanyl)ethyl]butanamide
1-[2-(cyclohexylmethyl)morpholin-4-yl]-2-phenylethane-1,2-dione
{[3-(methylsulfanyl)phenyl]methyl}({[2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
(1S,2R)-2-{[(8-chloroquinolin-2-yl)methyl](methyl)amino}cyclohexan-1-ol
4-(4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}phenyl)but-3-yn-1-ol
(1R,5R)-6-(1-benzofuran-2-ylmethyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
4-{4-[(4-fluorophenyl)methyl]-5-oxo-3-(propan-2-yl)-1,4-diazepan-1-yl}-N-methyl-4-oxobutanamide
(1S,3R)-N-(2-chlorophenyl)-3-[2-(2,5-dimethylphenyl)acetamido]cyclopentane-1-carboxamide