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5-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}-2-methylpyridine
(3R,4R)-1-(furan-3-carbonyl)-4-[4-(2-phenylethyl)piperazin-1-yl]piperidin-3-ol
(4aS,8aR)-6-[(4-methyl-1H-imidazol-5-yl)methyl]-1-(2-phenylethyl)-decahydro-1,6-naphthyridin-2-one
1-methyl-2-(morpholin-4-yl)-5-{1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-1H-1,3-benzodiazole
4-(2-{5H,6H,7H,8H-imidazo[1,5-a]pyrazine-7-carbonyl}phenyl)morpholine
(3aS,6aR)-5-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-1-methyl-N-(pyridin-4-ylmethyl)piperidin-4-amine
2-chloro-4-{[3-(3-methoxypropyl)piperidin-1-yl]methyl}phenol
1-[(4aR,8aR)-6-(3-methylbutyl)-decahydro-1,6-naphthyridin-1-yl]-3-(1H-indol-3-yl)propan-1-one
N-[3-(4-fluorophenyl)-3-(furan-2-yl)propyl]-3-(8-methoxy-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propanamide
2-(4-chlorophenyl)-5-(2,6-difluorobenzoyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
(2R,3R,6R)-3-(4-fluorophenyl)-5-(2-methyl-1,3-thiazole-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
methyl 2-[2-(5-methylfuran-2-yl)-1H-imidazol-1-yl]-2-(3-methylphenyl)acetate
2-{[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl](thiophen-3-ylmethyl)amino}butan-1-ol
9-(cyclopropylmethyl)-1-methyl-4-(pyrimidin-2-ylmethyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
6-[(3-methoxyphenyl)methoxy]-4-(5-methyl-1,2-oxazole-3-carbonyl)-1-(2-phenylethyl)-1,4-diazepan-2-one
1-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(1H-imidazol-1-yl)ethan-1-one
5-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidine-1-carbonyl]-4,6-dimethyl-1,2-dihydropyridin-2-one
4-ethyl-5-methyl-6-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]pyrimidin-2-amine
3-{[1-(5-oxopyrrolidine-2-carbonyl)piperidin-4-yl]methyl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{4-[(2-methylphenyl)sulfanyl]piperidin-1-yl}-2-(1H-1,2,3,4-tetrazol-5-yl)ethan-1-one
N-methyl-N-(2-phenoxyethyl)-1,8-naphthyridine-2-carboxamide
2-[4-(oxan-4-yl)piperazin-1-yl]-5-propylpyrimidine
1-(2-methoxyethyl)-3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidine
1-(3-chlorophenyl)-4-({4-[(1-{imidazo[1,2-a]pyridine-2-carbonyl}piperidin-4-yl)oxy]phenyl}methyl)piperazine
3-({[(4-fluorophenyl)methyl]amino}methyl)-5,6,7-trimethoxy-N,N-dimethylquinolin-2-amine
(2S,4R)-4-(cycloheptylamino)-N,N-diethyl-1-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
ethyl 2-[1-(2,1,3-benzoxadiazol-4-ylmethyl)piperidin-2-yl]acetate
2,4-dimethyl-N-[(1R,2S)-2-phenylcyclohexyl]pyrimidine-5-carboxamide
2-amino-6-[1-(3-chlorophenyl)-1H-pyrazol-4-yl]-4-(oxolan-3-yl)pyridine-3-carbonitrile
N,1,3-trimethyl-N-(quinolin-5-ylmethyl)-1H-pyrazole-4-carboxamide
N'-cycloheptyl-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}butanediamide
1-[1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carbonyl]-4-[3-(trifluoromethyl)phenyl]piperazine
(benzylsulfamoyl)[(8-methoxyquinolin-5-yl)methyl]methylamine
(2S,4R)-4-amino-N-methyl-1-{[5-(pyridin-2-yl)thiophen-2-yl]sulfonyl}pyrrolidine-2-carboxamide
N-(2,4-dimethoxyphenyl)-3-[3-(trifluoromethyl)benzoyl]piperidine-1-carboxamide
1-(1-cyclopentanecarbonylpiperidin-4-yl)-N-(2-phenylethyl)piperidine-4-carboxamide
(3S,4R)-4-(hydroxymethyl)-1-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}piperidin-3-ol
N-[2-(cyclohexylsulfanyl)ethyl]-3-(3-methoxyphenyl)-1H-pyrazole-4-carboxamide
3-[5-(furan-2-yl)-1,3,4-thiadiazol-2-yl]-1-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)urea
(3E)-2-({[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}(methyl)amino)-4-phenylbut-3-enoic acid
2-{[4-(pyrazin-2-yl)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino}ethan-1-ol
N-[2-(2,3-dimethoxyphenyl)ethyl]-6-ethyl-2-oxo-1,2-dihydropyridine-4-carboxamide
2-(5-{1-[2-(2-amino-4,6-dimethylpyrimidin-5-yl)acetyl]piperidin-4-yl}-1H-pyrazol-3-yl)acetic acid
5-fluoro-N-methyl-2-(pyrimidin-5-yl)pyrimidin-4-amine
N-(1-benzothiophen-2-ylmethyl)-3-(2-methyl-5-oxopyrrolidin-2-yl)propanamide
4-({2,4-dimethyl-5H,6H-furo[2,3-d]pyrimidin-6-yl}methyl)benzamide
N-({1-[(3-methyl-1H-indol-2-yl)methyl]pyrrolidin-3-yl}methyl)-1H-1,2,4-triazole-5-carboxamide
2-(1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}piperidin-4-yl)-1,2,3,4-tetrahydroisoquinoline
[(2S)-1-{[1-(3-fluorophenyl)-3-(5-methylfuran-2-yl)-1H-pyrazol-4-yl]methyl}pyrrolidin-2-yl]methanol