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1-ethyl-N-{[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-1H-pyrazole-4-carboxamide
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-6-methoxy-2,3-dihydro-1H-indene-5-carboxamide
4-[2-(2-hydroxyethoxy)ethyl]-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-[(3-fluorophenyl)methyl]-4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
2-[(4-{5-[(cyclohexylmethyl)sulfanyl]-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]pyridine
1-[2-(1-methyl-1H-pyrazol-3-yl)piperidin-1-yl]-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propan-1-one
7-methoxy-3-[5-(pyrrolidin-2-yl)thiophene-2-carbonyl]-2,3,4,5-tetrahydro-1H-3-benzazepine
1-(5-{[benzyl(2-hydroxyethyl)amino]methyl}-2-methoxyphenoxy)-3-[methyl(propan-2-yl)amino]propan-2-ol
1-{1-[4-(3-methoxyphenyl)phenyl]piperidin-4-yl}-1,4-diazepan-5-one
N-[(3R,4S)-1-acetyl-4-(propan-2-yl)pyrrolidin-3-yl]-3-fluoro-4-methoxybenzene-1-sulfonamide
3-[7-(2,2-dimethylpropyl)-2,7-diazaspiro[4.5]decane-2-carbonyl]pyridin-1-ium-1-olate
1-[(3,4-difluorophenyl)methyl]-3-(2-methoxyethyl)piperidine
1-{2-[8-(trifluoromethyl)-[1,2,4]triazolo[4,3-a]pyridin-3-yl]ethyl}-1H-pyrazole
7-(phenoxathiin-4-yl)-4-(pyridin-4-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
[(3-cyclopropyl-1H-pyrazol-5-yl)methyl][(4-fluorophenyl)methyl]methylamine
4-chloro-N,N-dimethyl-5-{[(2-methylpropyl)(pyridin-2-ylmethyl)amino]methyl}-1,3-thiazol-2-amine
4-{4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-5-propylpyrimidine
methyl 4-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}carbamoyl)butanoate
4-(2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-1,3-oxazole-4-carbonyl)-3-methylpiperazin-2-one
1-[(3-cyclopropyl-1H-pyrazol-5-yl)methyl]-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[2-(pyridin-3-yl)ethyl]acetamide
N-(2,3-dihydro-1H-inden-2-yl)-2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
6-[2-(1-benzylpyrrolidin-3-yl)ethyl]-2-methyl-2H,6H,7H-pyrazolo[4,3-d]pyrimidin-7-one
1-[(1S,5R)-3-acetyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-4-(4-methoxyphenyl)butan-1-one
{4-[({6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}(methyl)amino)methyl]oxan-4-yl}methanol
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-N1,5-bis[(3,4-dimethoxyphenyl)methyl]piperidine-3,5-dicarboxamide
3-[5-(1-ethyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazol-1-yl]-1λ6-thiolane-1,1-dione
N-[2-methoxy-2-(thiophen-2-yl)ethyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
4,6-dimethyl-N-[1-(pyridin-3-ylmethyl)piperidin-4-yl]pyrimidin-2-amine
{[2-(ethanesulfonyl)-1-(2-phenylethyl)-1H-imidazol-5-yl]methyl}(methyl)(2-methylprop-2-en-1-yl)amine
4-{[4-(2-methylphenyl)phenyl]methyl}-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-[3-(2-chlorophenyl)propanoyl]-N-cyclopropyl-1-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[6-(1H-pyrazol-3-yl)pyridine-3-carbonyl]-4-(pyrimidin-2-yl)-1,4-diazepane
5-[3,5-dimethyl-4-(2-oxopropyl)-1H-pyrazol-1-yl]pyridine-3-carboxamide
1-(2-fluorobenzoyl)-4-(2-methylpropyl)-1,4-diazepan-5-one
dimethyl({4-[1-(3,3,3-trifluoropropyl)piperidin-2-yl]phenyl}methyl)amine
(4aS,8aS)-2-(8-chloroquinolin-2-yl)-decahydro-2,7-naphthyridin-4a-ol
2-(3-methoxypropyl)-8-[2-(phenylsulfanyl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
1-[4-(4-tert-butyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-2-propylpentan-1-one
N-methyl-5-(5-methyl-1H-imidazol-2-yl)-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
(2S,4S)-4-{[(3,4-difluorophenyl)methyl]amino}-N-(propan-2-yl)-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
N-[1-(pyrimidin-2-yl)piperidin-3-yl]cyclohex-1-ene-1-carboxamide
2-[cyclopentyl(methyl)amino]-1-[(3R,4R)-3-hydroxy-4-methyl-3-(propan-2-yl)pyrrolidin-1-yl]ethan-1-one
N-[(1S)-1-[3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]-3-(methylsulfanyl)propyl]acetamide
methyl 1-[(2-methyl-1,3-oxazol-4-yl)methyl]-3-(3-methylbutyl)-2-oxo-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylate
3-(1-hydroxy-3-methylbutan-2-yl)-5,6-dimethyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
3-(4-hydroxyphenyl)-N-(1H-imidazol-2-ylmethyl)benzamide
3-(5-methyl-1,2,4-oxadiazol-3-yl)-1-[(2-phenyl-1,3-oxazol-4-yl)methyl]piperidine
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]-2-phenylethan-1-one
2-(2-ethyl-1H-imidazol-1-yl)-N-[1-phenyl-3-(propan-2-yl)-1H-pyrazol-5-yl]acetamide