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5-[3-cyclopropyl-1-(3-methylpyridin-4-yl)-1H-1,2,4-triazol-5-yl]pyridine-2-thiol
2-chloro-N,N-dimethyl-4-[({2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}carbamoyl)amino]benzamide
1-{4-[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]phenyl}-3-[1-(3-methylpyridin-2-yl)propan-2-yl]urea
2,2,3,3-tetramethyl-N-(2-methyl-1H-1,3-benzodiazol-6-yl)cyclopropane-1-carboxamide
2-{3-[(1-methylpiperidin-4-yl)methyl]-5-(1,3-thiazol-4-ylmethyl)-1H-1,2,4-triazol-1-yl}acetic acid
1-[(2-fluorophenyl)methyl]-3-hydroxy-3-({[(5-methylfuran-2-yl)methyl]amino}methyl)piperidin-2-one
3-({3-[3-(1,3-thiazol-2-yl)phenyl]-1H-pyrazol-1-yl}methyl)pyridine
4-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-(oxolan-2-yl)-1-[1-(thiophen-3-ylmethyl)piperidin-4-yl]-5-(trifluoromethyl)-1H-1,3-benzodiazole
N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-N-methyl-5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
1-{3-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-1-yl}butan-1-one
3-(propan-2-yl)-5-{1-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]pyrrolidin-2-yl}-1,2,4-oxadiazole
N-(2-methoxyethyl)-5-methyl-N-(1-methylpiperidin-4-yl)-1-propyl-1H-pyrazole-4-carboxamide
8-{3-methyl-5-[2-(morpholin-4-yl)pyridin-3-yl]-1H-1,2,4-triazol-1-yl}quinoline
1-methyl-9-(piperidin-3-ylmethyl)-1,4,9-triazaspiro[5.5]undecan-5-one
(3R,5S)-N-(2,3-dihydro-1H-inden-5-yl)-1-(2-phenylethyl)-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxamide
(3S,4S)-1-[(4-methyl-1H-imidazol-5-yl)methyl]-4-(naphthalen-2-yl)piperidin-3-ol
2-methoxy-N-[(1S,3S)-3-{[4-(pyridin-2-yl)pyrimidin-2-yl]amino}cyclopentyl]acetamide
methyl (2S,4R)-4-(5-chloro-3-phenyl-1H-indole-2-amido)-1-[(2,5-dimethoxyphenyl)methyl]pyrrolidine-2-carboxylate
N-(1-cyclohexyl-1H-pyrazol-5-yl)-2-[3-(dimethyl-1,3-thiazol-5-yl)-1H-pyrazol-1-yl]acetamide
1-{[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(2-methoxyethyl)piperazine
5-oxo-N-[(1-propyl-1H-imidazol-2-yl)methyl]-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
3-[6-amino-5-cyano-4-(piperidin-4-yl)pyridin-2-yl]benzoic acid
1-methoxy-8-[2-(4-phenylpiperidin-1-yl)acetyl]-1,8-diazaspiro[4.5]decan-2-one
9-(dimethyl-1,2-oxazole-4-carbonyl)-2-(1-methylpyrrolidin-3-yl)-2,9-diazaspiro[5.5]undecan-3-one
(4aS,7aR)-1-(4-chloro-2-fluorobenzoyl)-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3S,4R)-1-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}-3-ethyl-4-methylpiperidin-4-ol
methyl 3-({2-[4-(4-fluorophenyl)-5-{[(2-methylphenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl]ethyl}sulfamoyl)thiophene-2-carboxylate
(3S,4R)-1-{5-[(diethylamino)methyl]-2-methylfuran-3-carbonyl}-4-(hydroxymethyl)piperidin-3-ol
6-(propan-2-yl)-N4-{3-[(pyridin-3-yl)amino]propyl}pyrimidine-2,4-diamine
2-(4-chloro-1H-pyrazol-1-yl)-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}propanamide
2-(1H-1,3-benzodiazol-2-yl)-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)acetamide
3-ethyl-5-{3-[2-(1-methyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]phenyl}-4H-1,2,4-triazole
3-cyano-N-[2-(dimethylamino)-2-(3-methylphenyl)ethyl]benzamide
1-(4-fluorophenyl)-4-[1-(1,3-thiazole-4-carbonyl)piperidin-3-yl]piperazine
(3R,4R)-1-(6,7-diethoxy-3-methyl-1-benzofuran-2-carbonyl)-3,4-dimethylpyrrolidin-3-ol
(2E)-N-{[5-(pyridin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(thiophen-2-yl)prop-2-enamide
3-methyl-N-{1-oxaspiro[4.5]decan-3-yl}-1-propyl-1H-pyrazole-4-carboxamide
3-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-6-ethyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
7-[2-(3,4-dichlorophenyl)acetyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
2-amino-4-[(3S,4S)-3-hydroxy-4-(4-methylpiperazin-1-yl)pyrrolidin-1-yl]quinazoline-6-carboxylic acid
N-{[7-(5-acetylthiophen-2-yl)-1H,2H-naphtho[2,1-b]furan-2-yl]methyl}-1-methylpiperidine-3-carboxamide
N-methyl-3-(1H-pyrazol-1-ylmethyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)benzamide
{[5-(4-methoxyphenyl)furan-2-yl]methyl}(methyl)[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amine
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-4,5,6,7-tetrahydro-2-benzothiophene-1-carboxamide
2-({4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}methyl)pyridine
1-(4-benzylpiperidin-1-yl)-3-[1-(1-methylpiperidine-3-carbonyl)piperidin-4-yl]propan-1-one
2-ethyl-9-(3-methoxypropyl)-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
2-(2-methyl-1H-1,3-benzodiazol-5-yl)-N-[(4-sulfamoylphenyl)methyl]acetamide
4-[5-(methoxymethyl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-3-yl]pyridine