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1-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-3-phenylpropan-1-one
2-methyl-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)imidazo[1,2-a]pyrimidine-3-carboxamide
2-(dimethoxy-1,3,5-triazin-2-yl)aniline
N-[2-(4-sulfamoylphenyl)ethyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
N-methyl-6-(2-methylfuran-3-carbonyl)-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
2-[3-(hydroxymethyl)-8-methylquinolin-2-yl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-1-(furan-2-ylmethyl)piperidine-4-carboxamide
2-methyl-4-phenyl-3-[3-(thiophene-2-carbonyl)piperidine-1-carbonyl]pyridine
(furan-2-ylmethyl)({[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl})(prop-2-yn-1-yl)amine
N-[2-(5-methylthiophen-2-yl)ethyl]-3-(1H-1,2,4-triazol-1-yl)propanamide
3-{[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]methyl}-8-methyl-1,2-dihydroquinolin-2-one
3-(3,4-difluorophenyl)-1-[4-(1H-imidazol-2-yl)piperidin-1-yl]propan-1-one
8-(5,6-dimethylpyrimidin-4-yl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-({1-[6-(propylamino)pyridine-3-carbonyl]piperidin-4-yl}methyl)pyrrolidin-2-one
1-[4-(ethylsulfanyl)phenyl]-3-[3-(1H-imidazol-2-yl)propyl]urea
1-[(3R,4S)-3-amino-4-(3-methoxyphenyl)pyrrolidin-1-yl]-2-(2-methyl-1H-1,3-benzodiazol-1-yl)ethan-1-one
3-[5-(3,3,3-trifluoropropyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl]phenol
N6-cyclopentyl-N5-[(1-methyl-1H-imidazol-2-yl)methyl]-N5-(propan-2-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
5-[4-(2-chlorophenyl)piperazine-1-carbonyl]-1-[2-(morpholin-4-yl)ethyl]piperidin-2-one
2-amino-6-{4-[(6-methoxypyrimidin-4-yl)amino]piperidin-1-yl}-3,4-dihydropyrimidin-4-one
N-ethyl-5-(methoxymethyl)-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)furan-2-carboxamide
2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-5-(piperidin-1-yl)-2,3-dihydropyridazin-3-one
3-[(3R,4S)-1-(3-chloro-4-methylbenzoyl)-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
2-amino-8-(3-chloro-4-propoxyphenyl)-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-1-propyl-1H-pyrazole-5-carboxamide
4-{3-[5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-2-oxopiperidin-1-yl]propyl}piperazin-2-one
5-(3-fluorophenoxymethyl)-N-[(6-hydroxypyrimidin-4-yl)methyl]-1H-pyrazole-3-carboxamide
2-[4-(dimethylamino)phenyl]-1-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]ethan-1-one
1-(2-methoxyacetyl)-N-{1-[(3-methylphenyl)methyl]cyclopropyl}piperidine-4-carboxamide
1-(4-methoxyphenyl)-3-methyl-4-[2-(pyridin-2-yl)ethyl]piperazin-2-one
N-[(3S,4R)-4-(propan-2-yl)-1-[1-(pyridine-4-carbonyl)piperidin-4-yl]pyrrolidin-3-yl]acetamide
N-(2-methoxyethyl)-1-[1-(pyridine-3-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
4-[(3S)-3-ethylmorpholine-4-carbonyl]-6-(propan-2-yl)pyrimidin-2-amine
3-[4-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]-1,2,3,4-tetrahydroisoquinolin-1-one
methyl 3-[7-chloro-2-(acetamidomethyl)-2,3-dihydro-1-benzofuran-5-yl]benzoate
1-[(4-methoxyphenyl)methyl]-4-[3-(pyridin-2-yl)propanoyl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
6-[(4-methoxyphenyl)methyl]-1-[2-(piperidin-1-yl)ethyl]-3-(pyridin-4-yl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N-(2-methyl-2H-1,2,3-triazol-4-yl)-2-{1H-pyrrolo[2,3-b]pyridin-1-yl}acetamide
1-{4-[7-(cyclohexylmethyl)-2,7-diazaspiro[4.5]decan-2-yl]piperidin-1-yl}ethan-1-one
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methyloxane-2-carboxamide
2-(3-hydroxypropyl)-9-(2,4,6-trimethylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
8-(3-methoxy-5-methylthiophene-2-carbonyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
N-(2,1,3-benzoxadiazol-4-ylmethyl)-1-(3,5-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
5-[4-(4-methylphenoxy)piperidine-1-carbonyl]-1-[2-(morpholin-4-yl)ethyl]piperidin-2-one
N-{[(3S,4S)-3-hydroxypiperidin-4-yl]methyl}-3-(1H-indol-3-yl)propanamide
2-{imidazo[1,2-a]pyridin-2-yl}-7-(2-methoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
4-{4-[methyl(quinolin-5-ylmethyl)amino]piperidin-1-yl}-N-[2-(morpholin-4-yl)ethyl]benzamide
2-(2-methyl-1,3-thiazol-4-yl)-1-[2-(trifluoromethyl)pyrrolidin-1-yl]ethan-1-one
2-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-7-[(3,4-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decane
3-[3-methyl-1-(propan-2-yl)-1H-pyrazol-5-yl]-1-[1-(morpholine-4-carbonyl)piperidin-4-yl]urea