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1-(2H-1,3-benzodioxol-5-ylmethyl)-3-(oxolan-3-yl)-5-(1H-pyrazol-3-yl)-1H-1,2,4-triazole
5-[(isoquinolin-5-yloxy)methyl]-N-methyl-N-(pyridin-2-ylmethyl)-1,2-oxazole-3-carboxamide
N-[2-(6-hydroxypyrimidin-4-yl)ethyl]-5-methyl-3-phenyl-1,2-oxazole-4-carboxamide
2-[2-({[1-(hydroxymethyl)cyclobutyl]methyl}(methyl)amino)pyrimidin-4-yl]pyridine-4-carboxylic acid
3-(1H-1,2,3-benzotriazol-1-yl)-N-(butan-2-yl)-N-(thiophen-3-ylmethyl)propanamide
1-[(2-ethoxyphenyl)methyl]-3-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidine
N-methyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}-3-azaspiro[5.5]undecan-9-amine
N-(but-2-yn-1-yl)-N-(furan-2-ylmethyl)-1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carboxamide
1-{4-[2-amino-6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperazin-1-yl}-2,2-dimethylpropan-1-one
5-(2-{3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}phenyl)-1H-1,2,3,4-tetrazole
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-3-(4H-1,2,4-triazol-4-yl)benzamide
5-(4-methoxy-3-methylphenyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
1-{[1-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidin-3-yl]methyl}-1H-1,2,3-triazole-4-carboxylic acid
N-{[2-(2-cyclobutaneamidophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(3-hydroxy-3-methylbut-1-yn-1-yl)benzamide
N-{4-[2-(cyclopropylcarbamoyl)ethyl]phenyl}-3-(hydroxymethyl)piperidine-1-carboxamide
1-[3-(4-chloro-1H-pyrazol-1-yl)propanoyl]-3-(3-methoxypropyl)piperidine-3-carboxylic acid
N-(5-chloro-2-methoxyphenyl)-4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)piperidine-1-carboxamide
N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-(1-{1-[(6-chloroquinolin-2-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-methylbutanamide
4-[6-(2-methoxyphenyl)pyridazin-3-yl]-1-[(3-methylphenyl)methyl]piperazin-2-one
3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]piperidine
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]propanamide
1-[benzyl(methyl)amino]-3-(4-{[(3-ethoxypropyl)amino]methyl}phenoxy)propan-2-ol
N,2,2,6,6-pentamethyl-N-{[5-methyl-2-(naphthalen-1-yl)-1,3-oxazol-4-yl]methyl}piperidin-4-amine
N-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-5-phenyl-1,2-oxazole-3-carboxamide
N-methyl-5-({[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
4-(1H-imidazol-1-yl)-1-(4-methylbenzenesulfonyl)piperidine-4-carboxylic acid
2-(3-methoxypropyl)-9-(4-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
(1R,3S,5S)-8-{[4-(5-methylpyridin-2-yl)piperidin-4-yl]methyl}-8-azabicyclo[3.2.1]octan-3-ol
(4aR,7aS)-1-(2-methylpropanoyl)-4-[4-(1H-pyrazol-4-yl)butanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(1H-imidazol-4-ylmethyl)-N-[4-(1H-indol-2-yl)phenyl]pyrrolidine-2-carboxamide
2-{2-[2-(4-fluorophenyl)pyrrolidin-1-yl]ethyl}pyridine
(4aS,7aR)-1-(4-hydroxybenzoyl)-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-5-(morpholin-4-yl)-2,3-dihydropyridazin-3-one
4-{[4-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}quinoline
N'-(2-methylphenyl)-N-[1-(2-propoxyphenyl)ethyl]propanediamide
1-{2-[4-(4-methoxy-2,3-dimethylphenyl)-1H-1,2,3-triazol-1-yl]ethyl}piperidin-4-ol
5-{[6-oxo-4-(1,2,3,4-tetrahydroisoquinolin-2-yl)-1,6-dihydropyridazin-1-yl]methyl}-1,2,4-oxadiazole-3-carboxamide
2-[(3R,4R)-3-(hydroxymethyl)-4-[(4-hydroxypiperidin-1-yl)methyl]pyrrolidin-1-yl]-1,3-thiazole-4-carboxamide
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-N-[2-(1,3-thiazol-4-yl)ethyl]acetamide
4-(2,4-dioxoimidazolidin-1-yl)-N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}benzamide
4-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-[2-oxo-2-(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)ethyl]piperazin-2-one
N-[(2,6-dimethoxyphenyl)methyl]-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetamide
4-(1-methyl-1H-indole-6-carbonyl)-1λ6-thiomorpholine-1,1-dione
4-[(4-methanesulfonylphenyl)methyl]-1,9-dimethyl-1,4,9-triazaspiro[5.5]undecane
4-{1-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-1H-1,2,3-triazol-4-yl}quinoline
N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
methyl 5-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-cyclopentyl-N-[(2,4-dimethoxyphenyl)methyl]-1-ethyl-3-methyl-1H-pyrazole-4-carboxamide
3-(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)-1-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}urea