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1-(4-fluorophenyl)-N-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}cyclopropane-1-carboxamide
1-{1-[2-(2-hydroxyphenyl)acetyl]piperidin-3-yl}-3-phenylpropan-1-one
N-[2-(benzylsulfanyl)ethyl]-3-(pyridin-2-yl)-1H-pyrazole-5-carboxamide
2-(1H-1,3-benzodiazol-1-yl)-1-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]propan-1-one
butyl(furan-2-ylmethyl){[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}amine
3-{[4-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]methyl}pyridine
N-methyl-N-(2-methylpropyl)-5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]pyridin-2-amine
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-6-methoxypyrimidin-4-amine
N-(1-{7-[(4-chlorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)furan-2-carboxamide
2,4-dimethoxy-N-[(1-methylpiperidin-3-yl)methyl]-N-(2-phenylethyl)benzamide
N-[(5-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]acetamide
1-methyl-2-phenyl-4-[1-(pyrrolidin-1-yl)cyclopentanecarbonyl]piperazine
[(5-{[(3-fluorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl](methyl)[(3-methylthiophen-2-yl)methyl]amine
N-[2-(4-methoxyphenyl)ethyl]-N-[(1-methylpiperidin-4-yl)methyl]-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
N-[5-(pentan-2-yl)-1,3,4-thiadiazol-2-yl]-4-phenyl-1,2,3,6-tetrahydropyridine-1-carboxamide
1-tert-butyl-3-[2-(methylsulfanyl)ethyl]-5-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-1H-1,2,4-triazole
N-[(3R,4S)-1-(1-acetylpiperidin-4-yl)-4-(propan-2-yl)pyrrolidin-3-yl]furan-2-carboxamide
1-(5-methyl-1,3-oxazole-4-carbonyl)-4-[2-(methylsulfanyl)ethyl]piperazine
1-({3-methoxy-4-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)azetidin-3-ol
4-[5-chloro-2-(piperidine-1-carbonyl)phenoxy]-1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidine
1-(4-methoxyphenyl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}cyclopentane-1-carboxamide
2-benzyl-8-(1,4-dithiepan-6-yl)-2,8-diazaspiro[4.5]decan-3-one
3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)propanamide
[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]({[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl})methylamine
N-[2-(dimethylamino)-2-(4-methylphenyl)ethyl]-3-propyl-1H-pyrazole-5-carboxamide
2-(dimethylamino)-N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2-(3-methylphenyl)acetamide
N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(3,4-dimethoxyphenyl)acetamide
methyl 2-(5-methyl-2-{[2-(2-methyl-1,3-thiazol-4-yl)acetamido]methyl}-2,3-dihydro-1-benzofuran-7-yl)benzoate
3-(hydroxymethyl)-1-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]piperidin-3-ol
2-[(1-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperidin-3-yl)methyl]-1H-1,3-benzodiazole
(1S,5R)-6-(5-ethylthiophene-3-carbonyl)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
4-[(2,3-dihydro-1H-inden-2-yl)amino]-1-[(3-fluorophenyl)methyl]pyrrolidin-2-one
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-6-(2-methoxyphenyl)pyridazin-3-amine
4-(5-{imidazo[1,2-a]pyridine-2-carbonyl}-1-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl)morpholine
8-(1-hydroxypropan-2-yl)-1-(2-phenylethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-cyclopentyl-2-oxo-N-(3-phenylprop-2-yn-1-yl)-2,3-dihydro-1H-imidazole-4-carboxamide
5-(3-benzyl-1,2,4-oxadiazol-5-yl)-2-[(3-methylpiperidin-3-yl)methoxy]pyridine
N-(3-fluorophenyl)-1-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)piperidin-3-amine
2-[3-benzyl-1-(4-chlorophenyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-(propan-2-yl)acetamide
1-{1-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}-2-phenylethan-1-one
3-(3-fluorophenyl)-N-{[4-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-1H-pyrazole-4-carboxamide
(3aR,7aS)-2-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-2,3,3a,4,7,7a-hexahydro-1H-isoindole
2-{4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine-4-carbonitrile
(4aR,7aS)-N,N-diethyl-4-[(2-methylpyrimidin-5-yl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
N-[(1R,3R)-3-aminocyclopentyl]-1-phenyl-1H-1,2,3-triazole-5-carboxamide
3-[2-(7-fluoro-1-methyl-1,2,3,4-tetrahydroisoquinolin-2-yl)-2-oxoethyl]-1,3-diazinane-2,4-dione
2-(4-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}piperazin-1-yl)-4-methyl-6-(trifluoromethyl)pyrimidine
N-[2-(2-hydroxyethoxy)ethyl]-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
7-(cyclopropylmethyl)-2-[1-(3,4-difluorophenyl)piperidin-4-yl]-2,7-diazaspiro[4.5]decane
1-(4-methylpiperazin-1-yl)-3-[1-(pyridine-3-carbonyl)piperidin-3-yl]propan-1-one