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benzyl({[2-methanesulfonyl-1-(2-methylpropyl)-1H-imidazol-5-yl]methyl})(2-phenylethyl)amine
1-(5-ethyl-1,2-oxazole-3-carbonyl)-3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
1-({5-[1-(cyclopropylmethyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)-4-methylpiperazine
4-({[2-(5-chloro-4-methyl-1,3-thiazol-2-yl)ethyl]carbamoyl}amino)-N-ethylbenzamide
1-benzyl-N3-(1-benzylpyrrolidin-3-yl)-N5-ethyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
ethyl 3-(3-phenylpropyl)-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxylate
2-{[2-(2-carboxyethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]methyl}benzoic acid
N-(cyclopropylmethyl)-4-{[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]amino}-5-methyl-N-propylthieno[2,3-d]pyrimidine-6-carboxamide
N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-3-methoxypyridine-2-carboxamide
(1R,5R)-N,N-dimethyl-6-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
3-chloro-5-({3-[2-(pyridin-2-yl)pyrrolidine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)pyridine
1-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]-3-(1H-pyrazol-4-yl)propan-1-one
N-[(3-phenyl-1H-pyrazol-4-yl)methyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
2-methoxy-N-[1-(2-phenylethyl)-7-(2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)-1H-1,3-benzodiazol-5-yl]acetamide
2-[2-methyl-3-({[3-(1H-1,2,4-triazol-1-yl)propyl]amino}methyl)-1H-indol-1-yl]acetamide
N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
4-{[2-(4-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-methyl-2,3,4,5-tetrahydro-1H-1,4-benzodiazepine-2,5-dione
4-(pyrrolidin-1-ylmethyl)-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]benzamide
5-methyl-N-(prop-2-en-1-yl)-6-(pyrrolidine-1-carbonyl)thieno[2,3-d]pyrimidin-4-amine
2-methyl-6-{3-[(1-methylpiperidin-4-yl)oxy]propyl}-2H,6H,7H-pyrazolo[4,3-d]pyrimidin-7-one
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}-N-(2-methoxyethyl)-2-oxopropanamide
2-(2-methylpropyl)-8-[4-(pyrrolidine-1-carbonyl)pyridin-2-yl]-2,8-diazaspiro[4.5]decan-3-one
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N-methyl-3,4-dihydro-2H-1-benzopyran-3-carboxamide
4-(2,2-diphenylethyl)-3-[2-(1,2-oxazinan-2-yl)-2-oxoethyl]piperazin-2-one
N-[1-(2-hydroxyethyl)-3,5-dimethyl-1H-pyrazol-4-yl]-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl](2-methoxyethyl){[2-(propan-2-yl)pyrimidin-4-yl]methyl}amine
1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]piperazine
1-[4-(7-methoxy-4-methylquinazolin-2-yl)piperazin-1-yl]-2,2-dimethylpropan-1-one
3-chloro-5-({3-[2-(1,3-thiazol-2-yl)piperidine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)pyridine
[1-(5-{[(4-methoxy-3-methylphenyl)methyl]amino}-5,6,7,8-tetrahydroquinazolin-2-yl)piperidin-4-yl]methanol
1-(oxan-4-yl)-4-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)piperazine
5-ethyl-N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
8-[(5-cyclopentylthiophen-2-yl)methyl]-1,3-dioxa-8-azaspiro[4.5]decan-2-one
N-(3-methylbutyl)-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carboxamide
methyl 1-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine-2-carboxylate
2-[benzyl({[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl})amino]ethan-1-ol
5-acetyl-3-[(3S,4R)-4-hydroxy-4-methyl-3-(2-methylpropyl)piperidine-1-carbonyl]-6-methyl-1,2-dihydropyridin-2-one
N-(2-methyl-1-benzofuran-5-yl)-2-(pyridin-3-yl)piperidine-1-carboxamide
N-[2-(1H-imidazol-4-yl)ethyl]-4-[(1S,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]pyridine-2-carboxamide
1-{4-[2-(4-fluorophenyl)piperidine-1-carbonyl]piperidin-1-yl}-2-methoxyethan-1-one
4-{[2-(3-methoxyphenyl)ethyl]amino}-5-methyl-N-(pyridin-4-ylmethyl)thieno[2,3-d]pyrimidine-6-carboxamide
N-{1-[(3-fluorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-3-(1,2-oxazinan-2-yl)propanamide
N-[(3S,4R)-4-propyl-1-{thieno[3,2-d]pyrimidin-4-yl}pyrrolidin-3-yl]methanesulfonamide
3-{[3-(3-fluorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-1,3-oxazolidin-2-one
2-cyclopentyl-1-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}ethan-1-one
{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(methyl)[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amine
4-(2,3-dihydro-1H-inden-2-yl)-3-{2-[4-(methoxymethyl)piperidin-1-yl]-2-oxoethyl}piperazin-2-one
1-[3-(2-ethylphenoxy)azetidin-1-yl]-2-(methylsulfanyl)propan-1-one
3-{[4-(cyclobutylmethyl)piperazin-1-yl]methyl}-1-(cyclohexylmethyl)-3-hydroxypiperidin-2-one
1-{3-fluoro-7-methylimidazo[1,2-a]pyridine-2-carbonyl}-4-(4-fluorophenyl)piperidin-4-ol