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(3R,4R)-4-amino-1-(5,6,7,8-tetrahydroquinolin-2-yl)piperidin-3-ol
{1-[(2,3-dimethoxyphenyl)methyl]-3-[(3-methoxyphenyl)methyl]piperidin-3-yl}methanol
N-[(1-ethylpyrrolidin-2-yl)methyl]-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-1,3-dimethyl-1H-pyrazole-5-carboxamide
8-(2-fluorobenzoyl)-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-2-[(2-fluorophenyl)methyl]-1,3-benzoxazole-6-carboxamide
4-amino-2-(6-methoxypyridin-3-yl)pyrimidine-5-carbonitrile
{1-[(1-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}piperidin-4-yl)methyl]-1H-1,2,3-triazol-4-yl}methanamine
1-methyl-3-[3-(pyrazin-2-yl)-1,2,4-oxadiazol-5-yl]-1H-indole
2-amino-6-(2,4-dichlorophenyl)-4-(1,5-dimethyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
(1R,7S)-3-[(3,4-dimethylphenyl)methyl]-N-methyl-N-(1,2-oxazol-3-ylmethyl)-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl][(2-ethoxypyridin-3-yl)methyl]amine
1-(isoquinolin-5-yl)-3-(2-methoxyethyl)-3-[(trimethyl-1H-pyrazol-4-yl)methyl]urea
4,6-dimethoxy-2-{1H-pyrrolo[2,3-b]pyridin-4-yl}pyrimidine
9-(3-methoxypyrazin-2-yl)-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
2-(4-methyl-1,4-diazepan-1-yl)-N-[2-(morpholin-4-yl)ethyl]acetamide
N-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)sulfanyl]acetamide
5-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)pyridin-2-amine
5-cyclopropanecarbonyl-1'-(3-propyl-1H-pyrazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[(2-{4-[5-(methoxymethyl)furan-2-amido]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]imidazo[1,2-a]pyridine-2-carboxamide
1-[3-(dimethylsulfamoyl)-5-{[(3-hydroxy-4-methoxyphenyl)methyl]amino}benzoyl]piperidine-3-carboxamide
methyl({[4-(piperidin-1-ylmethyl)thiophen-2-yl]methyl})(pyrazin-2-ylmethyl)amine
N3-(adamantan-1-ylmethyl)-N3,N5-dimethyl-4-oxo-1-(3-phenylpropyl)-1,4-dihydropyridine-3,5-dicarboxamide
1'-(5-methyl-1,2-oxazole-3-carbonyl)-5-(3-methylbut-2-en-1-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-{1-[(2-ethoxyphenyl)methyl]-4-[(3-phenyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
2,3,6-trimethyl-4-[2-(pyridin-2-yl)piperidine-1-carbonyl]quinoline
4-(2-ethylpyrimidine-5-carbonyl)-2-(3-phenylpropyl)morpholine
5-[4-(dimethylamino)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]pyridin-2-amine
(1S,5R)-3-[(4-fluorophenyl)methyl]-6-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
2,5-dimethyl-3-(3-{1-[2-(1H-pyrazol-1-yl)ethyl]-1H-pyrazol-3-yl}phenyl)pyrazine
2-(4,6-dimethyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]acetamide
4-[(4-methoxyphenyl)methyl]-3-(1-methyl-5-oxopyrrolidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
{4-methyl-5-[1-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methanol
(3S,4R)-4-(2-methylphenyl)-1-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}pyrrolidine-3-carboxylic acid
2-methyl-N-{1-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]ethyl}-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
N-{3-[2-(dimethylamino)acetamido]-4-methylphenyl}-4-methyl-1,4-diazepane-1-carboxamide
3-[1-methyl-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-amido]pyrrolidine-3-carboxylic acid
N-(oxan-4-ylmethyl)-3-[(2-oxopyrrolidin-3-yl)sulfamoyl]benzamide
N-[2-(methylsulfanyl)phenyl]-3-(4-phenylpiperazin-1-yl)piperidine-1-carboxamide
9-[2-(4-chlorophenyl)acetyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
6-methyl-1-{3-[4-(piperidin-3-yl)-1H-1,2,3-triazol-1-yl]propyl}-1,2-dihydropyridin-2-one
2-[(6-{3,9-diazaspiro[5.5]undecan-3-yl}pyrimidin-4-yl)amino]ethan-1-ol
2-[3-(oxolan-3-yl)-5-(1H-pyrrol-2-yl)-1H-1,2,4-triazol-1-yl]-1H-1,3-benzodiazole
1-[(4-ethyl-1,3-thiazol-2-yl)methyl]-3-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)urea
2-(2-methoxyethyl)-9-(2,4,6-trimethylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[1-(2-phenylethyl)-1H-1,2,3-triazole-4-carbonyl]-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
3-[2-(3,4-difluorophenyl)ethyl]-1-(5-methyl-1,2-oxazole-3-carbonyl)piperidine
N-[2-(4-chlorophenyl)ethyl]-1-methyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-[methyl(phenyl)amino]-1-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
ethyl({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)(1H-imidazol-4-ylmethyl)amine
6-[1-(3-fluorophenyl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]-2-methyl-2,3-dihydropyridazin-3-one