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[(3R,4R)-4-(azepan-1-ylmethyl)-1-(2,6-dimethylpyridine-4-carbonyl)pyrrolidin-3-yl]methanol
2-ethoxy-5-{2-[(oxan-4-ylmethyl)amino]pyrimidin-4-yl}benzoic acid
2-(2,5-dioxo-1-propylimidazolidin-4-yl)-N-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)acetamide
3-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}propan-1-one
(4aS,7aR)-1-[2-(1H-1,3-benzodiazol-1-yl)acetyl]-4-(2-hydroxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(1-{[5-(2-cyanophenyl)furan-2-yl]methyl}piperidin-4-yl)-N-methylacetamide
1-cyclopentanecarbonyl-4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]piperidine
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-N5-[2-(2-oxoimidazolidin-1-yl)ethyl]-1-(2-phenylethyl)piperidine-3,5-dicarboxamide
3-{1-[1-(2,1,3-benzoxadiazol-5-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(2-methylphenyl)urea
5-methanesulfonyl-1'-(pyridin-3-ylmethyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-(2-fluorophenyl)-N-[2-(N-methylmethanesulfonamido)ethyl]cyclopropane-1-carboxamide
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(naphthalen-2-ylmethyl)pyrrolidin-3-yl]methanol
(3S,5R)-N3-(6-methylpyridin-3-yl)-N5-[3-(1H-pyrazol-1-yl)propyl]piperidine-3,5-dicarboxamide
N4,6-dimethyl-N4-[3-(1H-pyrazol-1-yl)propyl]pyrimidine-2,4-diamine
N-{[(3S,4S)-3-hydroxypiperidin-4-yl]methyl}-3-(5-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)propanamide
1,5-dimethyl-2-phenyl-4-({3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}methyl)-2,3-dihydro-1H-pyrazol-3-one
1-methyl-1'-[2-(methylsulfanyl)pyrimidin-4-yl]-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
1-(isoquinoline-1-carbonyl)-N-methyl-N-(2-phenylethyl)piperidin-3-amine
2-benzyl-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-1,3-thiazole-4-carboxamide
2-[(4aS,8aR)-1-(4-hydroxybutyl)-2-oxo-decahydro-1,6-naphthyridin-6-yl]-4,6-dimethylpyridine-3-carbonitrile
N-(1-propyl-1H-1,3-benzodiazol-5-yl)-4-(pyridin-2-yl)piperazine-1-carboxamide
2-methoxy-5-({3-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)phenol
2-{4-[(2-fluoro-4-methylphenyl)methyl]morpholin-2-yl}ethan-1-ol
6-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-N,N-dimethylpyridazin-3-amine
N-cyclohexyl-4-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidine-1-carboxamide
4-[3-(1-methoxyethyl)phenyl]thieno[3,2-d]pyrimidine
3-[(2-methoxyethyl)sulfamoyl]-5-(2-methyl-1H-1,3-benzodiazol-1-yl)benzoic acid
N-{2-[5-(1-ethyl-1H-1,2,4-triazol-5-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}pyridin-3-amine
N-cyclopropyl-5-(1-{pyrazolo[1,5-a]pyridine-3-carbonyl}pyrrolidin-2-yl)thiophene-2-carboxamide
2-(4-fluorophenyl)-1-(2-methyl-1,3-thiazole-5-carbonyl)piperidine
2-{[2-(2-methoxypyrimidin-5-yl)-1H-imidazol-1-yl]methyl}-5,6-dimethyl-1H-1,3-benzodiazole
N5-[(2-fluoro-5-methoxyphenyl)methyl]-N2,N2-dimethyl-5,6,7,8-tetrahydroquinazoline-2,5-diamine
3-(3-hydroxyquinoxalin-2-yl)-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}propanamide
4-[2-(oxolan-3-yl)-1H-imidazol-1-yl]benzene-1-sulfonamide
4-(2,3-dimethoxyphenyl)-1-[1-(3-ethyl-1,2-oxazol-5-yl)ethyl]-1H-1,2,3-triazole
N-(pyridin-2-ylmethyl)-2-[3-(1H-1,2,3,4-tetrazol-1-yl)propanamido]benzamide
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]acetamide
3-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1H-indazole
3-[(2R,3R,6R)-5-(2,6-dimethylbenzoyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
methyl 3-[2-(2-methylphenyl)acetyl]-7-oxo-9-[2-(2-oxopyrrolidin-1-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]-1-[2-methyl-4-(pyrrolidin-1-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
N-(1-{1-[(2-fluoro-5-methoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopentanecarboxamide
6-(4-fluorophenyl)-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
3-[2-(5-amino-1,3,4-thiadiazol-2-yl)acetamido]-N-tert-butyl-2-methylbenzamide
2-[(5-methylpyrazin-2-yl)methyl]-8-[2-(2-oxopyrrolidin-1-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
5-[4-(5-chloropyridin-2-yl)piperazine-1-carbonyl]-1-[2-(pyridin-2-yl)ethyl]piperidin-2-one
5-[5-(4-methoxyphenyl)furan-2-carbonyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
2-[(1-benzylpyrrolidin-3-yl)methyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}[(3-methoxyphenyl)methyl]amine
2-amino-N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carboxamide