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methyl 4-{[(2-{1-[(4-methylphenyl)methyl]-5-oxopyrrolidin-2-yl}ethyl)amino]methyl}benzoate
2-methyl-6-(piperidin-4-yl)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]pyrimidin-4-amine
2-[1-(2-methoxyethyl)-1H-1,2,3,4-tetrazol-5-yl]-4-{2-methylthieno[2,3-d]pyrimidin-4-yl}morpholine
(4aS,7aR)-4-(1-benzofuran-5-ylmethyl)-N-ethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
3-[1-(1-benzofuran-2-ylmethyl)piperidin-3-yl]-N-methyl-N-(1-methylpiperidin-4-yl)propanamide
N-tert-butyl-2-[4-methyl-6-(morpholine-4-carbonyl)-3,4-dihydro-2H-1,4-benzoxazin-3-yl]acetamide
N,8-dimethyl-N-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
(2E)-N-({7-[2-(1H-indol-3-yl)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-3-(thiophen-2-yl)prop-2-enamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2-ethyl-6-methyl-4-oxo-1-[2-(piperidin-1-yl)ethyl]-1,4-dihydropyridine-3-carboxamide
(2E)-3-(2-chlorophenyl)-1-[3-(4-{[4-(pyridin-3-ylmethyl)piperazin-1-yl]methyl}phenoxymethyl)piperidin-1-yl]prop-2-en-1-one
3-[(3R,4S)-1-[(1-ethenyl-1H-pyrazol-4-yl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
2-[1-(2,3-dihydro-1H-inden-5-yl)-5-[(3-methyl-6-oxo-1,6-dihydropyridazin-1-yl)methyl]-1H-1,2,4-triazol-3-yl]acetamide
1-methyl-3-(2-methylpropyl)-N-[2-(morpholin-4-yl)butyl]-1H-pyrazole-5-carboxamide
2-({[(3R,4R)-1-(2,4-difluorobenzoyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(ethyl)amino)ethan-1-ol
1-{[1-({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidin-3-yl]methyl}pyrrolidin-2-one
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}quinolin-2-amine
N-methyl-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}-1H-pyrrolo[2,3-b]pyridin-6-amine
3-{1-[2-(3-methylpyridin-2-yl)ethyl]-4-phenyl-1H-imidazol-5-yl}pyridine
N-[2-(5-cyclobutyl-1,2,4-oxadiazol-3-yl)ethyl]-3-(trifluoromethyl)benzamide
1-{5-methyl-6-[(2-methylpyridin-3-yl)oxy]pyrimidin-4-yl}-N-(1,2-oxazol-3-ylmethyl)piperidin-4-amine
N-[(3S,4R)-4-(propan-2-yl)-1-[1-(pyrazine-2-carbonyl)piperidin-4-yl]pyrrolidin-3-yl]acetamide
4-[3-(1-methoxypropan-2-yl)-3H-imidazo[4,5-b]pyridin-2-yl]-1-{1-oxa-7-azaspiro[3.5]nonan-7-yl}butan-1-one
methyl({[3-(naphthalen-1-yl)-1H-pyrazol-4-yl]methyl})[1-(pyrimidin-4-yl)ethyl]amine
3-[(3aR,5R,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindole-2-carbonyl]-6-methyl-1,2-dihydropyridin-2-one
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetamide
methyl 2-{[(3S)-2-oxoazepan-3-yl]({[4-(pyridin-2-ylmethoxy)phenyl]methyl})sulfamoyl}benzoate
2-{5-[2-(2-fluorophenyl)benzoyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl}ethan-1-ol
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-1-(methoxymethyl)cyclobutane-1-carboxamide
(2S,4S,5R)-2-ethyl-5-(4-methoxyphenyl)-1-methyl-4-(4-methylpiperazine-1-carbonyl)pyrrolidine-2-carboxylic acid
N-[1-(1-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]-2-methoxybenzamide
(1S,5R)-3-[(4-fluorophenyl)methyl]-6-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-3,6-diazabicyclo[3.2.2]nonane
2-(4-fluorophenyl)-1-(pyrrolidine-1-sulfonyl)piperidine
2-{[2-(2-ethyl-4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]methyl}-4-methyl-6-(trifluoromethyl)pyrimidine
ethyl 4-{1-[2-(2-methoxyphenyl)acetyl]piperidin-3-yl}piperazine-1-carboxylate
3-cyclopropyl-5-{2,7-dimethylpyrazolo[1,5-a]pyrimidin-5-yl}-1H-1,2,4-triazole
(1S,5R)-3-cyclobutanecarbonyl-6-(3,5-dimethyl-1-benzofuran-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-N-[(4-methylphenyl)methyl]piperidine-4-carboxamide
4-{[2-(3-chlorophenyl)-6,7-dimethoxyquinolin-3-yl]methyl}piperazin-2-one
5-ethyl-3-(2-{2-[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]-1H-imidazol-1-yl}ethyl)-1,2,4-oxadiazole
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidin-6-yl}pyrrolidine-1-carboxamide
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}-3-(pyridin-3-yl)propanamide
1-[(2R,3R,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(morpholin-4-yl)propan-1-one
4-(1H-imidazol-1-yl)-1-{thieno[2,3-d]pyrimidin-4-yl}piperidine-4-carboxylic acid
(4aS,8aR)-6-[3-(5-amino-1H-1,2,4-triazol-3-yl)propanoyl]-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)(methyl){[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}amine
N-[(dimethyl-1,3-thiazol-2-yl)methyl]-1-[2-(dimethylamino)ethyl]-5-oxopyrrolidine-3-carboxamide
8-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
5-{3-[4-(4-chlorophenoxy)piperidin-1-yl]-3-oxopropyl}-5-{[4-(methylsulfanyl)phenyl]methyl}pyrrolidin-2-one
8-(2-ethylpyrimidine-5-carbonyl)-2-(3-methylphenyl)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
5,6-dimethyl-N-[2-(3-phenylpyrrolidin-1-yl)ethyl]pyrimidin-4-amine