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N-(2-chloro-6-methylphenyl)-8-cyclopropyl-9-oxo-2,8-diazaspiro[5.5]undecane-2-carboxamide
4-[4-(3-fluorophenoxy)piperidine-1-carbonyl]-1,2-dihydroquinolin-2-one
methyl 3-(4-methoxybenzamido)-1-methyl-5-{[(2E)-2-methylbut-2-en-1-yl]amino}-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-1-[4-(methylsulfanyl)phenyl]urea
4-[1-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]-1-(3-fluoropropyl)-1,2,3,6-tetrahydropyridine
5-{[4-(2-phenoxyethyl)piperazin-1-yl]methyl}-2-(pyridin-2-yl)pyrimidine
2-{1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]pyrrolidin-2-yl}ethan-1-ol
N-{1-[(3-chlorophenyl)methyl]-1H-pyrazol-5-yl}-2-(ethanesulfonyl)propanamide
3-cyclohexyl-4-(2-ethyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-1H-pyrazole
N-(1-ethynylcyclohexyl)-3-(4-methyl-1,3-thiazol-5-yl)propanamide
5-[(3S,4R)-3-(dimethylamino)-4-(4-methoxyphenyl)pyrrolidine-1-carbonyl]-4-ethyl-1,3-thiazol-2-amine
4,5-dimethyl-3-(2-{3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}ethyl)-1H-pyrazole
1-{[2-(2-methoxyethyl)pyrimidin-5-yl]methyl}-N-[3-(1H-pyrazol-1-yl)phenyl]piperidine-3-carboxamide
8-(furan-3-carbonyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-1-{4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}ethan-1-one
1-[(3-methylphenyl)methyl]-5-[3-(1H-1,2,4-triazol-1-yl)propyl]-1H-1,2,4-triazole
1-[2-(methylsulfanyl)ethyl]-4-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}piperazine
2-(pyridin-4-yl)-N-[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]pyrimidine-5-carboxamide
N-[(2,6-dimethylpyridin-4-yl)methyl]-3-(1-methylpiperidin-3-yl)propanamide
(4aS,8aR)-1-(2-methylpropyl)-6-[3-(1H-1,2,4-triazol-1-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
(3S,4S)-4-(dimethylamino)-1-{[2-(3-methylphenyl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}pyrrolidin-3-ol
2-(4-{[4-(benzyloxy)phenyl]methyl}-1-(propan-2-yl)piperazin-2-yl)ethan-1-ol
N-[3-(2-methoxyphenoxy)propyl]-N-methyl-4-(5-methylfuran-2-yl)benzamide
5-{[2-(3,4-dichlorophenyl)morpholin-4-yl]methyl}quinoline
8-(1-ethyl-1H-pyrazole-5-carbonyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[(3S,5S)-5-(diethylcarbamoyl)-1-(1H-imidazol-2-ylmethyl)pyrrolidin-3-yl]pyrazine-2-carboxamide
4-{[2-(2-hydroxyethyl)-3-oxopiperazin-1-yl]methyl}-N-(3-methylpyridin-2-yl)benzamide
1-[3-({[3-(4-fluorophenyl)oxolan-3-yl]methyl}amino)phenyl]pyrrolidin-2-one
1-(3-fluoropyridin-4-yl)-4-(4-methoxybenzoyl)piperazine
1-(3-chlorophenyl)-3-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}urea
1-ethyl-3-methyl-N-{[4-(2-phenylethyl)-4H-1,2,4-triazol-3-yl]methyl}piperidine-3-carboxamide
1-(2-methylpropyl)-5-(4-oxo-1,4-dihydroquinoline-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
N-({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-N-methylcyclohexanamine
N-{1-[(4-methoxy-2,3,6-trimethylphenyl)methyl]pyrrolidin-3-yl}acetamide
N-methyl-N-(2-phenylethyl)-1-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-amine
1-(pyridin-3-ylmethyl)-4-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-2-one
4-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-(2-methoxyethyl)-9-(1H-pyrazole-4-sulfonyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
N-butyl-3-{[(1H-indol-4-ylmethyl)amino]methyl}-N-methylimidazo[1,2-a]pyridine-2-carboxamide
3-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-triene-4-carbonyl]benzonitrile
N-(1-hydroxybutan-2-yl)-N-(pyridin-2-ylmethyl)-2,3-dihydro-1-benzofuran-5-carboxamide
({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)({[4-methoxy-3-(methoxymethyl)phenyl]methyl})methylamine
5-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-N-ethylpyrimidin-2-amine
1-[(2,2-dimethyloxan-4-yl)methyl]-4-(3-methyl-1H-1,2,4-triazol-5-yl)piperidine
3-{[2-(1,3-benzothiazol-2-yl)ethyl]amino}-N-(1,3-thiazol-2-yl)propanamide
1-[(2,3-difluoro-6-methoxyphenyl)methyl]-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methyl-1-(1,3,4-thiadiazol-2-yl)piperidine
2-(2-aminoethyl)-N-(furan-2-ylmethyl)-N-(pyridin-2-ylmethyl)quinazolin-4-amine
1-{2-[2-(1-methyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]ethyl}-4-(propan-2-yl)piperazine