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3-{2-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-oxoethyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(2H-1,3-benzodioxol-5-yl)-N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)propanamide
6-cyclopentyl-N,1-dimethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(1R,5R)-6-(2-methoxyethyl)-3-(1H-pyrazole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
4-methyl-6-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidine
1-methyl-6-(propan-2-yl)-N-{[4-(pyrrolidine-1-carbonyl)phenyl]methyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-3-[4-(methylsulfanyl)benzoyl]piperidine
4-[4-(1-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]piperidine
2-(2,5-dimethylfuran-3-carbonyl)-7-[(2-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
5-(2-methylpropyl)-1'-(2-methylpyrimidin-4-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-6-[2-(pyridin-2-yl)pyrrolidin-1-yl]pyridine-3-carboxamide
4-(5-{1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]pyrrolidin-2-yl}-1,2,4-oxadiazol-3-yl)pyridine
N-{1-[4-(1H-pyrazol-3-yl)benzoyl]piperidin-4-yl}methanesulfonamide
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-5-methyl-2-(methylamino)benzamide
(3aR,6aR)-2-cyclopentyl-5-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(3-fluorophenyl)-1-{7-methyl-[1,2,4]triazolo[4,3-a]pyrimidine-3-carbonyl}piperidin-3-amine
1-{3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}-2-(2-hydroxyphenyl)ethan-1-one
3-[(3R,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[(1S)-1-phenylethyl]urea
1-(1H-imidazol-2-ylmethyl)-3-(4-methoxy-3,5-dimethylbenzoyl)piperidine
5-(5-chloro-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1-cycloheptylpiperidin-2-one
(3R,4S)-4-cyclopropyl-1-(5-propyl-1,2,4-oxadiazol-3-yl)pyrrolidin-3-amine
2-{4-[1-(4-cyclopentylpyrimidin-2-yl)piperidin-4-yl]piperazin-1-yl}ethan-1-ol
9-(4-cyclobutyl-6-methylpyrimidin-2-yl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
2-(2-chlorophenyl)-3-methyl-N-[2-(pyridin-4-yl)ethyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
N1-(3-methoxy-4-methylphenyl)-N3-methylpyrrolidine-1,3-dicarboxamide
N-{[3-(pyrazin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
N-[(2R,4R,6S)-2-(propan-2-yl)-6-{pyrazolo[1,5-a]pyrimidin-3-yl}oxan-4-yl]benzamide
N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]-3-(1H-pyrazol-1-yl)benzamide
methyl (2S)-2-{[6-(3-fluorophenyl)imidazo[2,1-b][1,3]thiazol-3-yl]formamido}-2-phenylacetate
N-[(2R,3R)-2-methoxy-1'-{[2-(2-methylphenyl)pyrimidin-5-yl]methyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
1-{5-methanesulfonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-methoxybutan-1-one
2-(adamantan-1-yl)-1-[2-(morpholin-4-ylmethyl)pyrrolidin-1-yl]ethan-1-one
N4-[3-(furan-2-yl)propyl]-N2,N2-dimethyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
N-(4-fluorophenyl)-4-(thiomorpholin-4-yl)piperidine-1-carboxamide
2-methoxy-N-methyl-5-({[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]carbamoyl}amino)benzamide
4-[(4-ethoxyphenyl)methyl]-3-[2-oxo-2-(3-oxopiperazin-1-yl)ethyl]piperazin-2-one
(4aR,8aS)-1-(3,3-diphenylpropyl)-6-(pyridin-2-ylmethyl)-decahydro-1,6-naphthyridin-2-one
2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-{2-[(4-methylpyridin-2-yl)amino]ethyl}acetamide
[4-(oxan-2-ylmethyl)-1-(pyridin-3-ylmethyl)piperidin-4-yl]methanol
(1R,5R)-6-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
2-(3-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}phenoxy)acetic acid
ethyl 4-({[(4-fluorophenyl)methyl](prop-2-en-1-yl)amino}methyl)-1H-pyrazole-3-carboxylate
methyl (2S,4R)-4-hydroxy-1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)pyrrolidine-2-carboxylate
(1R,5S)-3-[3-(2-methoxyphenyl)propanoyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
8-(4-methylpentanoyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
(4-{[1-(benzenesulfonyl)-1H-pyrrol-2-yl]methyl}morpholin-2-yl)methanamine
N-{3-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]-3-oxopropyl}acetamide
N-(3,4-difluorophenyl)-1-(3-ethyl-1-methyl-1H-pyrazole-5-carbonyl)piperidin-3-amine
5-(2,6-dimethylphenoxymethyl)-N-{[1-(2-methoxyethyl)piperidin-3-yl]methyl}-1,2-oxazole-3-carboxamide
4-{[(4-hydroxy-6-methylquinolin-2-yl)methyl]amino}-N-methylbutanamide