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3-[2-(2,6-difluorophenyl)ethyl]-1-(1-methyl-1H-pyrazole-4-carbonyl)piperidine
(3aS,6aR)-5-(1,3-benzoxazol-2-yl)-3-[2-(4-fluorophenyl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
4-{1-[(3-chlorophenyl)methyl]-5-[1-(methoxymethyl)cyclopropyl]-1H-1,2,4-triazol-3-yl}pyridine
{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}[(3-methoxyphenyl)methyl]amine
5-(3-chloropyridine-4-carbonyl)-N-(2-hydroxyethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-methyl-4-{4-[(4-{4-[3-(trifluoromethyl)phenyl]-1H-pyrazol-5-yl}piperidin-1-yl)methyl]phenyl}but-3-yn-2-ol
2-(4-{[4-(benzenesulfonyl)piperazin-1-yl]methyl}-3-methyl-1H-pyrazol-1-yl)ethan-1-ol
2-[2-(dimethylamino)ethyl]-9-{[2-(methylsulfanyl)phenyl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
5-(propan-2-yl)-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)pyrimidin-4-amine
2-{2-[5-(1-benzofuran-2-yl)-4-phenyl-1H-imidazol-1-yl]ethoxy}ethan-1-ol
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-6-(3-hydroxypiperidin-1-yl)pyridine-3-carboxamide
8-cyclopropanecarbonyl-2-[2-(pyridin-3-yl)acetyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-(3-methylthiophene-2-carbonyl)-3-(naphthalene-1-carbonyl)piperidine
N-(2-methoxyethyl)-6-methyl-4-oxo-2-(2-phenylethyl)-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
5-methyl-6-(piperidine-1-carbonyl)-N-(thiophen-2-ylmethyl)thieno[2,3-d]pyrimidin-4-amine
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1,4-dioxane-2-carboxamide
N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]pyrazolo[1,5-a]pyridine-7-carboxamide
3-(furan-2-yl)-3-[(2,3,6-trimethylquinolin-4-yl)formamido]propanoic acid
N,N-dimethyl-1-[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]pyrrolidin-3-amine
2-[({[4-(3-chlorophenyl)-5-[(3-hydroxypropyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}(methyl)amino)methyl]phenol
N-{3-[({3-hydroxy-1-[4-(propan-2-yl)phenyl]propyl}carbamoyl)amino]phenyl}-N-methylacetamide
2-[(2,6-dichloro-3,4-dimethoxyphenyl)methyl]-octahydropyrrolo[1,2-a]piperazine
1-(2-{[4-(pyridin-4-yl)pyrimidin-2-yl]amino}ethyl)imidazolidin-2-one
3-ethyl-8-[2-hydroxy-5-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(3R,4R)-4-ethyl-1-(3-hydroxybenzoyl)piperidine-3,4-diol
3-hexyl-8-(2-hydroxybenzoyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(3-chloro-4-methoxyphenyl)-6-[2-(1,3-dioxo-2,3-dihydro-1H-isoindol-2-yl)acetyl]-6-azaspiro[2.5]octane-1-carboxamide
2-(5-{1-[3-(1H-pyrazol-4-yl)benzoyl]piperidin-4-yl}-1H-pyrazol-3-yl)acetic acid
N-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
1-{3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecan-11-yl}-2-(2-ethylpiperidin-1-yl)ethan-1-one
1-{6-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-5-methylthieno[2,3-d]pyrimidin-4-yl}azocane
6-hydroxy-1-[3-(2-oxopyrrolidin-1-yl)propyl]-4-{[1-(propan-2-yl)-1,2,3,4-tetrahydroquinolin-6-yl]methyl}-1,4-diazepan-2-one
1-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
6-[2-(1,3-thiazol-2-yl)piperidine-1-carbonyl]-1,2,3,4-tetrahydroquinoxaline-2,3-dione
1-{4-[3-(2-chlorophenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}cyclobutan-1-amine
N-{[1-(morpholin-4-yl)cyclopentyl]methyl}-5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carboxamide
N-[(3S,4R)-4-(4-methoxyphenyl)-1-(quinolin-4-ylmethyl)pyrrolidin-3-yl]acetamide
({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amine
(3aR,6aR)-2-(2-ethyl-6-methylpyrimidin-4-yl)-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-({[(3R,4R)-4-(hydroxymethyl)-1-[(5-methylfuran-2-yl)methyl]pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
N-(4-ethoxy-2-fluorophenyl)-3-(morpholin-4-ylmethyl)piperidine-1-carboxamide
2-{2,5-dioxo-3-phenyl-1-[3-(pyridin-3-yloxy)propyl]pyrrolidin-3-yl}-N-ethyl-N-(oxolan-2-ylmethyl)acetamide
1-[2-(dimethylamino)ethyl]-4-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidine-1-carbonyl}pyrrolidin-2-one
N-[(3S,4R)-1-[2-(4-fluorophenoxy)ethyl]-4-propylpyrrolidin-3-yl]acetamide
3-(2-methyl-1,3-benzothiazol-5-yl)-1-(oxolan-2-ylmethyl)-1-(pyridin-4-ylmethyl)urea
N-cyclopropyl-1-{1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]piperidin-4-yl}piperidine-3-carboxamide
N-[2-(2-methoxyphenyl)ethyl]-3-[(3S,4R)-1-(propan-2-yl)-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]propanamide
2-(3-{[4-(dimethylamino)azepan-1-yl]methyl}phenoxy)ethan-1-ol
2-methyl-4-phenyl-9-(pyrazin-2-yl)-2,9-diazaspiro[5.5]undecane
3-[8-(5-methoxyfuran-2-carbonyl)-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl]propanoic acid