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3-(azocan-1-yl)-N-[(1-methanesulfonylpiperidin-3-yl)methyl]propanamide
2-[4-({3-methyl-2-oxo-1-oxa-3,7-diazaspiro[4.5]decan-7-yl}methyl)phenyl]acetic acid
1-(diethylamino)-3-{2-methoxy-4-[(3,3,4-trimethylpiperazin-1-yl)methyl]phenoxy}propan-2-ol
N-(4-chloro-3-methylphenyl)-2-{[3-(1H-1,2,4-triazol-1-yl)propyl]amino}acetamide
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-1,3-benzothiazole-2-carboxamide
[(4-methoxy-2,3,6-trimethylphenyl)methyl](2-methoxyethyl)(pyridin-4-ylmethyl)amine
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3,3,3-trifluoropropanamide
N-[(3,5-difluorophenyl)methyl]-1-methyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
5-[5-(2-methylpropyl)-1H-1,2,4-triazol-3-yl]isoquinoline
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-(dicyclopropylmethyl)benzamide
1-[4-(furan-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]-2-phenylethan-1-ol
(4aR,8aS)-1-[(4-fluorophenyl)methyl]-6-[5-(methoxymethyl)furan-2-carbonyl]-decahydro-1,6-naphthyridin-2-one
3-{2-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]-2-oxoethyl}imidazolidine-2,4-dione
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidin-3-ol
4-[2-(3-aminopyrrolidin-1-yl)-2-oxoethyl]-1-(4-chlorophenyl)-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
4-hydroxy-N-(2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-4-yl)-2-(pyridin-2-yl)pyrimidine-5-carboxamide
N-(propan-2-yl)-4-{3-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}pyridine-2-carboxamide
N-{[1-(cyclohex-1-ene-1-carbonyl)piperidin-3-yl]methyl}furan-2-carboxamide
(2S,4S)-1-[(3-acetyl-2,4,6-trimethylphenyl)methyl]-4-amino-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-[7,7-dimethyl-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]cyclobutanecarboxamide
1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-1H,2H,3H,4H,6H,10bH-pyrimido[2,1-a]isoindol-6-one
methyl (2R)-2-[3-(5-cyclohexyl-1,3,4-oxadiazol-2-yl)propanamido]propanoate
1-[2-(dimethylamino)-4-{[2-(4-methoxyphenyl)ethyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
methyl 3-propanamido-5-[(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylformamido)methyl]benzoate
1-{4-[4-(aminomethyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}-2-(2,5-dimethylphenoxy)propan-1-one
1-[2-(dimethylamino)ethyl]-N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-5-oxopyrrolidine-3-carboxamide
2-[2-(2-amino-6-oxo-1,6-dihydropyrimidin-4-yl)acetyl]-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
ethyl 5-{[({4-[3-(diethylamino)-2-hydroxypropoxy]-3-methoxyphenyl}methyl)amino]methyl}furan-2-carboxylate
1-methyl-1'-[2-methyl-2-(morpholin-4-yl)propyl]-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
2-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-1-(pyrrolidin-1-yl)propan-1-one
2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-[1-(2-fluorophenyl)piperidin-4-yl]acetamide
4-{[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-3-methyl-1-propyl-1H-pyrazole
(1-{1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)methanamine
ethyl 3-[({spiro[azepane-4,2'-chromene]-1-yl}carbonyl)amino]propanoate
2-{[3-(2-chlorophenoxy)azetidin-1-yl]methyl}-1H-imidazole
N-[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(4,5,6,7-tetrahydro-2H-indazol-3-yl)propanamide
2-benzyl-4-[(3,4,5-trimethoxyphenyl)methyl]morpholine
5-{[4-(2,2-dimethylpropyl)-3-(2-hydroxyethyl)piperazin-1-yl]methyl}-2-methoxyphenol
2-({4-[6-amino-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-1H-pyrrolo[2,3-b]pyridin-6-yl}amino)acetic acid
(3R,4S)-4-cyclopropyl-1-(5-ethyl-1,2-oxazole-3-carbonyl)pyrrolidin-3-amine
8-chloro-2-ethyl-4-[3-(1H-pyrazol-1-ylmethyl)benzoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-(2-fluorophenyl)-1-(2-methylfuran-3-carbonyl)pyrrolidine
4-(5-ethylfuran-2-yl)-7-hydroxy-6-methyl-1,2,3,4-tetrahydroquinolin-2-one
5-(3-methyl-1,2,4-oxadiazol-5-yl)-N-(oxan-2-ylmethyl)pyridin-2-amine
2-methyl-4-(5-{8-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-2-carbonyl}furan-2-yl)but-3-yn-2-ol
3-(3,4-dimethoxybenzoyl)-1-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}piperidine
1-{2-[1-(2-methoxyphenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]ethyl}-4,6-dimethyl-1,2-dihydropyrimidin-2-one
2-{1-[(2-chloro-4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-hydroxyethyl)-N-methylacetamide
N-benzyl-N-methyl-1-[2-methyl-6-(2-methylpropyl)pyrimidine-4-carbonyl]piperidin-3-amine