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3-(3-methylbutyl)-8-[2-(3-oxopiperazin-1-yl)acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-[4-(2-methoxyphenyl)-3,3-dimethylpiperazine-1-carbonyl]-5-methylpyrazine
2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(propan-2-yloxy)ethyl]acetamide
N-{2-[4-(pyridin-3-ylmethyl)morpholin-2-yl]ethyl}thiophene-3-carboxamide
2-methyl-6-{[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]methyl}pyridine
2-[1-(3-methylbutyl)-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl]-N-(thiophen-2-ylmethyl)acetamide
1-(4-fluorophenyl)-4-[1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-3-yl]piperazine
3-propyl-1-(5-propyl-1,3,4-thiadiazol-2-yl)piperidine-3-carboxylic acid
8-[(4-chloro-2-methylphenyl)carbamoyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-[(3R,4S)-1-(2-ethylbutanoyl)-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
5-[(3-methoxyphenyl)methyl]-1-(2-phenylethyl)-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[cyclohexyl(methyl)amino]-3-[3-({methyl[(5-methylfuran-2-yl)methyl]amino}methyl)phenoxy]propan-2-ol
6-methyl-3-[(1S,5R)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,2-dihydropyridin-2-one
4-[2-(methylsulfanyl)propyl]-1-[2-(thiophen-2-yl)ethyl]-1H-1,2,3-triazole
6-oxo-N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)-1,6-dihydropyridine-3-carboxamide
5-cyclopropyl-3-methyl-N-[2-(3-phenylpyrrolidin-1-yl)ethyl]-1H-pyrazole-4-carboxamide
3-(3-hydroxy-1,2-oxazol-5-yl)-1-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}propan-1-one
N-{2-[4-(4-ethyl-2,5-dioxoimidazolidin-4-yl)piperidin-1-yl]-2-oxoethyl}methanesulfonamide
N-[(2,6-difluoro-4-methoxyphenyl)methyl]-N-methylthian-4-amine
4-(2,6-dimethylpyridin-3-yl)-2-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}pyrimidine
2-(oxolan-2-ylmethyl)-9-(pyrimidin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-{5-cyclobutanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-methoxybutan-1-one
(3R,4R)-4-(hydroxymethyl)-1-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-ol
3-{1-[(2-hydroxyphenyl)methyl]piperidin-4-yl}-N-{[3-(trifluoromethyl)phenyl]methyl}propanamide
2-amino-4-{3-[(dimethylamino)methyl]-4-hydroxyphenyl}-5H,6H,7H-pyrrolo[2,3-h]quinoline-3-carbonitrile
ethyl 4-[2-(dimethylamino)-2-(2-methylphenyl)acetyl]piperazine-1-carboxylate
5-[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-1-(2-methylphenyl)-3-phenyl-1H-1,2,4-triazole
5-[(2-fluoro-5-methoxyphenyl)methyl]-5-(3-oxo-3-{1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl}propyl)pyrrolidin-2-one
5-methyl-3-phenyl-N-{[5-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-3-yl]methyl}-1,2-oxazole-4-carboxamide
N-[(2-chloro-6-fluorophenyl)methyl]-N-cyclopropyloxane-2-carboxamide
[(1-{[1-(3-chloropyridine-4-carbonyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl](methyl)amine
N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-3-(1H-1,2,4-triazol-1-yl)propanamide
(1R,5R)-N,N-dimethyl-6-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
6-(3-{3-[benzyl(methyl)amino]piperidin-1-yl}-3-oxopropyl)-2,3,4,5-tetrahydropyridazin-3-one
2-[2-(2-ethylphenoxy)ethyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
3-[(3-hydroxypropyl)[(5-methylthiophen-2-yl)methyl]amino]propane-1,2-diol
N-cyclohexyl-3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carboxamide
4-phenyl-1-{3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}butane-1,2-dione
2-[1-(5-chloropyridin-2-yl)-1H-pyrrol-2-yl]-1H-1,3-benzodiazole-5-carbonitrile
methyl 8-[(5-methylfuran-2-yl)methyl]-2-oxo-1-(prop-2-en-1-yloxy)-1,8-diazaspiro[4.5]decane-4-carboxylate
(4aS,8aS)-2-cyclohexyl-7-(4-methylpyridine-3-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
4-{4-[2-(2-chlorophenyl)-2-hydroxyacetyl]piperazin-1-yl}-2-(pyridin-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
N-(2-hydroxyethyl)-5-[(2-methoxyphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
1-[(3-benzyl-1H-1,2,4-triazol-5-yl)methyl]-1H-1,2,3,4-tetrazole
4-[4-(6-hydroxypyrimidin-4-yl)piperidine-1-carbonyl]-1-oxaspiro[4.4]nonan-2-one
2-methoxy-4-[3-(1H-pyrazol-3-yl)phenyl]phenol
3-{imidazo[1,2-a]pyridin-2-yl}-5-[3-(1H-pyrazol-1-ylmethyl)phenyl]-1,2,4-oxadiazole
2-methylpropyl 2-(1-methyl-1H-1,3-benzodiazol-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxylate
3-(4-methoxyphenyl)-5-{3-methyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl}-1H-pyrazole
3-[2-(4-hydroxypiperidin-1-yl)-2-oxoethyl]-4-(naphthalen-1-ylmethyl)piperazin-2-one