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1-ethyl-N-methyl-N-[1-(pyridin-2-yl)propyl]-1H-pyrazole-5-carboxamide
4-(4-fluorophenyl)-N-(3-methyl-1,2,4-thiadiazol-5-yl)-1,4-diazepane-1-carboxamide
N-[(3,4-dimethoxyphenyl)methyl]-N-methyl-3-(3-methylpiperidin-1-yl)propanamide
2-[4-(1H-imidazol-1-ylmethyl)piperidin-1-yl]-2-[4-(2-methylpropanamido)phenyl]acetic acid
[2-(furan-2-yl)ethyl]({[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl})amine
{[2-(2,3-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(furan-2-ylmethyl)(prop-2-yn-1-yl)amine
5-chloro-6-{4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidin-1-yl}pyridine-3-carboxylic acid
N-(1-{1-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]piperidin-4-yl}-2-phenylethyl)-N-methylthiophene-2-carboxamide
4-(4-{[2-(oxolan-3-yl)ethyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl)benzamide
N-({1-[2-(quinazolin-4-yloxy)acetyl]piperidin-3-yl}methyl)thiophene-2-sulfonamide
2,6-diamino-4-(3-cyclohexyl-1H-pyrazol-4-yl)-5,6,7,8-tetrahydroquinoline-3-carbonitrile
5-methoxy-4-oxo-N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]-1,4-dihydropyridine-2-carboxamide
N-(1-{7-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-3-methoxypropanamide
{9-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-(oxan-4-yl)-3,9-diazaspiro[5.5]undecan-1-yl}methanol
1-cyclopentyl-N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]piperidine-3-carboxamide
2-phenoxy-N-({7-[(2,4,6-trimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)acetamide
3-[(1E)-3-{3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-3-oxoprop-1-en-1-yl]-4H-chromen-4-one
2-{2-[2-(3-hydroxyphenyl)-1H-imidazol-1-yl]phenyl}-N,N-dimethylacetamide
N-[(3,4-dimethoxyphenyl)methyl]-N,5-dimethyl-2-(2-methylpropanamido)benzamide
[(1-methylpiperidin-4-yl)methyl](2-phenylethyl)(pyridin-3-ylmethyl)amine
N-(1-{7-[(3-fluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-phenoxyacetamide
3-({2-[1-(dimethyl-1,3-oxazole-5-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
3-(2-methyl-1H-indol-1-yl)-N-(oxan-4-ylmethyl)propanamide
N-methyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}-2-(pyrrolidin-3-yl)benzamide
4-(2-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}phenyl)morpholine
methyl[(3-methylquinoxalin-2-yl)methyl][1-(pyrazin-2-yl)propan-2-yl]amine
4-{[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-2-butyl-1H-imidazole
1-(1-{[3-(cyclopropylmethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-3-yl)-3-phenylpropan-1-one
{1-[1-(9H-fluoren-2-ylmethyl)piperidin-3-yl]piperidin-4-yl}methanol
N-ethyl-3-{imidazo[1,2-a]pyridin-2-yl}-N-[(2E)-3-phenylprop-2-en-1-yl]propanamide
7-methoxy-N-{2-[(4-methylpyridin-2-yl)amino]ethyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-{4-[3-(3-chlorophenyl)pyrrolidine-1-carbonyl]-1H-1,2,3-triazol-1-yl}-N,N-diethylacetamide
N-({1-[(5-methylthiophen-2-yl)methyl]piperidin-3-yl}methyl)-3-(trifluoromethyl)benzamide
1-[9-(cyclopropylmethyl)-1-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-3-yl]-3-(1-methyl-1H-pyrazol-5-yl)propan-1-one
N-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}acetamide
2-[3-(3-methoxypropyl)piperidin-1-yl]quinoline
2-(4-hydroxyphenyl)-7-(2-methoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
(4aS,7aR)-1-(6-oxo-1,6-dihydropyridine-3-carbonyl)-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(1,3-benzothiazole-6-carbonyl)-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one
N-[4-(1H-pyrazol-1-yl)phenyl]-1-(4,4,4-trifluorobutyl)pyrrolidine-2-carboxamide
3-({1-[6-methyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-4-yl}amino)-2,3-dihydro-1λ6-thiophene-1,1-dione
2-ethyl-4-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridine
2-[2-fluoro-5-(trifluoromethyl)phenyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-(4-{[4-(dimethylamino)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)-1-phenoxypropan-2-ol
3-[(dimethylamino)methyl]-1-[(5-ethylpyridin-2-yl)methyl]pyrrolidin-3-ol
1-[5-(methoxymethyl)-1,3,4-oxadiazole-2-carbonyl]-4-(6-methylpyridin-2-yl)piperazine
8-(4-aminobutanoyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
4-{4-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperazin-1-yl}quinazoline
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-6-methoxy-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
(4aS,7aR)-N-butyl-4-[(2-methylphenyl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide