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5-(4-cyclohexylpiperazin-1-yl)-1-(4-methylpentyl)azepan-2-one
1-methyl-4-[4-methyl-2-(propan-2-yl)pyrimidine-5-carbonyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
N,N-dimethyl-3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-sulfonamide
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-1-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecan-4-yl]ethan-1-one
2-({1-[1-(2-phenylethyl)piperidin-4-yl]piperidin-3-yl}formamido)acetamide
N-{4-[9-methoxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-4-oxobutan-2-yl}acetamide
N-(2-methoxyethyl)-N-[(4-methylphenyl)methyl]-2-(4-oxo-3,4-dihydrophthalazin-1-yl)propanamide
6-[3-(2-methoxyphenyl)propanoyl]-N-(2-methyl-1,3-benzothiazol-5-yl)-6-azaspiro[2.5]octane-1-carboxamide
N-{[2-(azepan-1-yl)-6-methylquinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)acetamide
({5-[1-(2,6-dimethylpyrimidine-4-carbonyl)piperidin-3-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
7-(cyclopropylmethyl)-2-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
1-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]-2-phenyl-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
N-cyclopropyl-5-(1H-imidazol-4-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
5-[4-(4-methoxybenzoyl)piperazine-1-carbonyl]-1-(2-phenylethyl)piperidin-2-one
2-{1-[5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]piperidin-3-yl}propan-2-ol
5-{3-[4-(methylsulfanyl)benzoyl]piperidine-1-carbonyl}-1H-1,3-benzodiazole
1-[1'-(1,2-oxazole-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
1-(3-chlorophenyl)-5-methyl-4-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}piperazin-2-one
8-[(3,4-dimethylphenyl)methyl]-2-(3-hydroxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
(3aS,6aS)-2-(6-carbamoylpyrazin-2-yl)-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-cyclopentyl-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-6-oxopiperidine-3-carboxamide
2-methoxy-2-methyl-1-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)propan-1-one
1-(4-methoxybutyl)-4-(5-propyl-1,2-oxazole-3-carbonyl)piperazine
4-cyano-N-[3,5-difluoro-4-(trifluoromethyl)phenyl]piperidine-1-carboxamide
(3aR,6aR)-N-{[2-(2-methoxyphenyl)-1,3-thiazol-5-yl]methyl}-2-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
N-{[5-methyl-7-(2-methylquinolin-6-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}furan-2-carboxamide
5-[(3-fluorophenyl)methyl]-3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
6-[(1R,2S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]tridecan-11-yl]pyridine-2-carbonitrile
2-[1-(5-propyl-1,2-oxazole-3-carbonyl)piperidine-3-carbonyl]pyridine
N-ethyl-5-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]-N-[(1-methyl-1H-imidazol-2-yl)methyl]pyridin-2-amine
4-{[4-(3-chlorophenyl)-1H-1,2,3-triazol-1-yl]methyl}-1-(1H-imidazole-2-carbonyl)piperidine
(2S)-2-({2,7-dimethyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)-3-phenylpropanamide
3-{2-[4-(4,6-dimethylpyrimidin-2-yl)piperazin-1-yl]-2-oxoethyl}-2,3-dihydro-1H-isoindol-1-one
8-(furan-2-ylmethyl)-3-[(4-methoxyphenyl)methyl]-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
methyl 3-(2-chlorobenzenesulfonamido)-5-{[(3-fluorophenyl)formamido]methyl}benzoate
3-cyclopentaneamido-N-(furan-2-ylmethyl)-N-(prop-2-en-1-yl)benzamide
1-(1,3-thiazole-5-carbonyl)-4-(1H-1,2,3-triazol-4-ylmethyl)-1,4-diazepan-6-ol
N-{3-[(3-methyl-3-phenylpiperidin-1-yl)sulfonyl]phenyl}acetamide
1-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-4-(4-fluorophenyl)butan-1-one
6-[(3-methoxyphenyl)methoxy]-1-(2-phenylethyl)-4-[3-(pyridin-2-yl)propanoyl]-1,4-diazepan-2-one
1-{1-[(2-cyanophenyl)methyl]piperidin-4-yl}-N-cyclopropylpiperidine-3-carboxamide
3-amino-N-ethyl-N-[(3-methoxyphenyl)methyl]-1H-1,2,4-triazole-5-carboxamide
1-cyclohexyl-5-[4-(1H-pyrazol-1-yl)phenyl]-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazole
N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
4-(piperidin-1-yl)-1-[4-(1H-1,2,4-triazole-3-carbonyl)piperazin-1-yl]butan-1-one
(6-methylhept-5-en-2-yl)[3-(oxolan-3-yl)propyl]amine
N-[2-(4-chlorophenyl)-2-(pyrrolidin-1-yl)ethyl]-5,6,7,8-tetrahydroquinoline-3-carboxamide
3,5-dimethyl-4-{1-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]pyrrolidin-2-yl}-1,2-oxazole
1-[4-hydroxy-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidin-1-yl]-3-(1-methyl-1H-pyrazol-5-yl)propan-1-one
7-({[2-methoxy-1-(pyridin-2-yl)ethyl](methyl)amino}methyl)-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one