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[2-(6-methoxypyridin-3-yl)-1,3-thiazol-4-yl]methanol
propan-2-yl 2-chloro-5-(2,2-dimethyl-4-oxo-3,4-dihydro-2H-pyran-6-amido)benzoate
(3R,4R)-1-[(2-chloro-5-fluorophenyl)methyl]-3-methyl-4-(oxan-4-yl)piperidin-4-ol
N-[(5-ethylpyridin-2-yl)methyl]-7-fluoro-N-methylquinazolin-4-amine
(3S,4R)-1-(3-hydroxy-4-methylbenzoyl)-4-phenylpyrrolidine-3-carboxylic acid
2,6-dimethyl-N-[2-(3-phenylpiperidin-1-yl)ethyl]pyridine-4-carboxamide
{1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}({[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl})amine
N-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-1-(pyrimidin-2-yl)piperidin-3-amine
4-{4-[1-(oxan-4-yl)piperidine-3-carbonyl]piperazin-1-yl}phenol
N-[2-(2,4-dimethoxyphenyl)ethyl]-5-(2,6-dimethylphenoxymethyl)-1,2-oxazole-3-carboxamide
N-{4-[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]phenyl}-2-oxo-1-oxa-3,8-diazaspiro[4.6]undecane-8-carboxamide
5-methyl-N-{[3-methyl-7-(2-oxo-2H-chromene-3-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}thiophene-2-carboxamide
N2,N4-dimethyl-N2-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]pyrimidine-2,4-diamine
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[(2,6-dimethylphenyl)methyl]piperidin-3-ol
3-[({4-chloro-1H-pyrrolo[2,3-b]pyridin-6-yl}amino)methyl]-1λ6-thiolane-1,1-dione
1-(oxan-4-yl)-4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]piperidine
6-(5-ethyl-1,2-oxazole-3-carbonyl)-3-(8-methoxy-2-methylquinolin-5-yl)-1-methyl-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
1-[(2-chloro-4-fluorophenyl)methyl]-N-[2-(4-phenylpiperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-[(3-methyl-1,2-oxazol-5-yl)methyl]-5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
2-(cyclohex-1-en-1-yl)-N-({3-[(3-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazol-5-yl}methyl)acetamide
2-[3-(prop-2-en-1-yl)-4-(propan-2-yloxy)phenyl]-1H-imidazole
2-(5-{[methyl(oxan-4-yl)amino]methyl}furan-2-yl)benzonitrile
N-[1-(1-{[3-(2-hydroxyethoxy)phenyl]methyl}piperidin-4-yl)-2-phenylethyl]-N-methylthiophene-2-carboxamide
2-(dimethyl-1,3-thiazol-4-yl)-N-[(4-methylphenyl)(pyridin-4-yl)methyl]acetamide
4-[(2S,4R)-4-hydroxypyrrolidine-2-carbonyl]-1-(2-phenylphenyl)piperazin-2-one
N6-(2-methoxyethyl)-N5-[(3-methoxyphenyl)methyl]-N5-methyl-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
(2S)-3-(1H-imidazol-4-yl)-2-{[4-methyl-3-(2-oxoimidazolidin-1-yl)phenyl]formamido}propanamide
{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}({[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
3-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)-1-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]propan-1-one
methyl 6-[(3-chlorophenyl)methyl]-2-(piperidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-{ethyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amino}-N-[1-(4-methylphenyl)ethyl]acetamide
2-(2-methoxyphenoxy)-N-({1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperidin-3-yl}methyl)acetamide
3-(3-methyl-1H-pyrazol-1-yl)-N-[3-(2-oxo-1,2-dihydropyridin-1-yl)propyl]propanamide
5-[2-(furan-2-yl)azepane-1-carbonyl]-1H-1,2,3-benzotriazole
ethyl 4-{2-[3-oxo-1-(pyridin-3-ylmethyl)piperazin-2-yl]acetamido}piperidine-1-carboxylate
methyl 3-(furan-2-amido)-1-(3-methylbutyl)-5-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-[2-(2-methyl-1H-indol-3-yl)acetyl]-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-6-(pyridin-4-yl)pyridine-3-carboxamide
N-[(3R,4S)-4-cyclopropyl-1-[(methylcarbamoyl)methyl]pyrrolidin-3-yl]cycloheptanecarboxamide
N,8-dimethyl-3-({methyl[2-(1H-pyrazol-4-yl)ethyl]amino}methyl)-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
(3S,4S)-4-(4-fluorophenyl)-1-(2-hydroxy-4-methoxybenzoyl)piperidin-3-ol
2-{4-[(2-fluoro-5-methoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}-1-phenoxypropan-2-ol
1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-N-methyl-N-(1-methylpiperidin-4-yl)-5-(propan-2-yl)-1H-pyrazole-4-carboxamide
4-ethyl-5-methyl-6-[4-(morpholine-4-carbonyl)piperazin-1-yl]pyrimidin-2-amine
ethyl 1-[2-(3-methoxyphenyl)-1,3-benzoxazole-6-carbonyl]piperidine-3-carboxylate
1-{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}-3-(methoxymethyl)piperidine
3-{[1-benzyl-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]methyl}imidazolidine-2,4-dione
1-(2-{1-[1-(4-methylphenyl)cyclopropanecarbonyl]piperidin-4-yl}ethyl)pyrrolidin-2-one
5,6-dimethyl-3-[4-(1H-pyrazol-5-yl)phenyl]-1,2-dihydropyridin-2-one
3-(5-{1-[2-(pyridin-4-yl)-1H-imidazol-1-yl]ethyl}-1,2,4-oxadiazol-3-yl)pyridine