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5-[1-(but-2-ynoyl)piperidin-4-yl]-5-(pyridin-3-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
1-(4-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}piperidin-1-yl)ethan-1-one
N-methyl-N-(2-methylpropyl)-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-methyl-4-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)piperazine
3-(2-methoxyethyl)-1-[4-(1H-pyrazol-1-yl)phenyl]-3-[(trimethyl-1H-pyrazol-4-yl)methyl]urea
N-[(2S)-1-hydroxy-3-methylbutan-2-yl]-5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
3-{[(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}pyridin-2-amine
5-[2-(3-methoxyphenyl)pyrrolidine-1-carbonyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole
2-(2H-1,3-benzodioxol-5-yloxy)-N-methyl-N-(thiophen-3-ylmethyl)propanamide
1-{3-[3-(4-benzylpiperazin-1-yl)-3-oxopropyl]piperidin-1-yl}-3-(1,2-oxazolidin-2-yl)propan-1-one
3-ethyl-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)-1H-pyrazole-5-carboxamide
6-[(4aR,8aR)-4a-hydroxy-7-(2-methoxyacetyl)-decahydro-2,7-naphthyridin-2-yl]-3-chloropyridine-2-carboxylic acid
6-cyano-N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}pyridine-3-carboxamide
N-(4-acetylphenyl)-4-(1-methyl-1H-imidazol-2-yl)piperidine-1-carboxamide
N-methyl-N-(2-phenylethyl)-5-({[4-(1H-pyrazol-1-yl)butan-2-yl]amino}methyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
8-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
7-({cyclopropyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
2-[(E)-2-phenylethenyl]-5-(pyrrolidin-1-ylmethyl)pyridine
2-{2,5-dioxo-3-phenyl-1-[3-(pyridin-3-yloxy)propyl]pyrrolidin-3-yl}-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]acetamide
1-amino-N-[3-(2-chlorophenoxy)propyl]-N-methylcyclopropane-1-carboxamide
N,N-dimethyl-3-[({1H-pyrrolo[2,3-b]pyridin-6-yl}amino)methyl]benzamide
(2R,3R)-3-amino-1'-(quinoxalin-2-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-{2-[2-(pyridin-3-yl)-1,3-thiazol-4-yl]ethyl}morpholine-2-carboxamide
1-[4-chloro-3-(furan-2-amido)phenyl]-5-oxopyrrolidine-3-carboxylic acid
N-phenyl-2-{[2-(propan-2-yloxy)ethyl]amino}butanamide
3-(4-methanesulfonylphenyl)-5-methyl-2-(4H-1,2,4-triazol-4-yl)pyridine
5-(2-ethoxypyridin-3-yl)-N-ethylthiophene-2-carboxamide
1-(1-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}piperidin-3-yl)pyrrolidin-2-one
N-(quinolin-8-ylmethyl)-3,4-dihydro-2H-1-benzopyran-3-amine
N-{[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}-2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
N-[(2-{4-[5-(methoxymethyl)thiophene-2-amido]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]-2,6-dimethylpyrimidine-4-carboxamide
methyl 4-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidine-1-carboxylate
N-(2-hydroxyethyl)-N-methyl-1-(1-{[4-(propan-2-yl)phenyl]methyl}piperidin-3-yl)-1H-1,2,3-triazole-4-carboxamide
1-(furan-3-carbonyl)-N-[2-(3-methoxyphenyl)phenyl]piperidine-4-carboxamide
N-[2-(dimethylamino)-2-(2-methylphenyl)ethyl]-3-(4-fluorophenyl)-1H-pyrazole-5-carboxamide
2-benzyl-8-(2,4-dimethylpyrimidine-5-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
1-[2-({[2-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]amino}methyl)phenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl](methyl)[(5-methylfuran-2-yl)methyl]amine
1-butyl-5-[2-(1H-1,2,4-triazol-1-yl)phenyl]-1H-1,2,4-triazole
3-methoxy-5-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyridine
3-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]-1-propyl-1H-pyrazole-4-carboxamide
4-[(1R,5S)-3,8-diazabicyclo[3.2.1]octane-8-carbonyl]-6-ethyl-2-methylquinoline
N-ethyl-3-(4-fluorophenyl)-N-[2-(1H-pyrazol-1-yl)ethyl]-1H-pyrazole-5-carboxamide
N-[3-(3-chlorophenyl)phenyl]-1-(2-methoxyacetyl)piperidine-4-carboxamide
3-cyclopentaneamido-N-methyl-N-[(3-methylpyridin-2-yl)methyl]benzamide
2-cyclopropyl-N-[4-(methylsulfanyl)phenyl]-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
N-[2-(azepan-1-yl)ethyl]-2-(dimethylamino)-2-(3-fluorophenyl)acetamide
N-(3-phenylprop-2-yn-1-yl)-N-propylbut-3-enamide
({6-[4-(3-chlorophenyl)piperazin-1-yl]-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl}methyl)[1-(thiophen-2-yl)ethyl]amine