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N,N-dimethyl-2-[(1S,5R)-7-oxo-3-(3-propyl-1H-pyrazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
4-({[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]amino}methyl)-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
1-{3-[3-({[2-(2-chlorophenyl)ethyl]amino}methyl)phenoxy]-2-hydroxypropyl}piperidin-4-ol
5-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-6-methyl-4-(thiophen-2-yl)-1,2,3,4-tetrahydropyrimidin-2-one
1-[(3ar,6ar)-octahydropyrrolo[3,4-c]pyrrole-3a-carbonyl]-4-(piperidin-1-yl)piperidine-4-carboxamide
(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-6-[2-(methylsulfanyl)pyridine-3-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
1-methyl-4-[(1-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)methyl]piperazine
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-4-(pyridin-3-yl)pyrimidin-2-amine
2-{4-[(1-ethyl-1H-indol-5-yl)methyl]-2-oxopiperazin-1-yl}benzonitrile
6-[4-(hydroxymethyl)phenyl]-N,N-dimethylpyridine-2-carboxamide
2-methyl-4-{4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidine
(2R,3R)-3-amino-1'-[4-(trifluoromethyl)pyridin-2-yl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-(2-cyano-3-methylphenyl)-3-{[methyl(oxolan-2-ylmethyl)amino]methyl}benzamide
1-[(2-chloro-4-fluorophenyl)methyl]-N-[2-(3-methoxyphenyl)ethyl]-1H-1,2,3-triazole-4-carboxamide
3-(4,5-dimethyl-1H-1,3-benzodiazol-6-yl)-1-[2-(pyrrolidine-1-sulfonyl)ethyl]urea
5-(1,2-oxazinane-2-carbonyl)-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidin-2-one
N-[(3S,4R)-1-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-propylpyrrolidin-3-yl]methanesulfonamide
3-[3-(1H-pyrazol-1-yl)phenyl]pyridin-4-amine
3-ethyl-5-methyl-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-1,2-oxazole-4-carboxamide
3-[(4aS,8aR)-decahydroisoquinoline-2-carbonyl]-1-cyclohexyl-5-(pyrrolidine-1-carbonyl)-1,4-dihydropyridin-4-one
5-(1-cyclohexyl-4-hydroxypiperidin-4-yl)-N-methyl-N-(quinolin-6-ylmethyl)-1-benzofuran-2-carboxamide
N-({2-[(2-oxopyrrolidin-1-yl)methyl]phenyl}methyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-[2-(1H-indol-1-yl)ethyl]-N-methylquinoxaline-5-carboxamide
N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}-2-(thiophen-3-yl)acetamide
2-(4-{5-[3-(3-methylbutanoyl)piperidine-1-carbonyl]pyridin-2-yl}phenyl)acetic acid
4-(3-methoxyphenyl)-2-{5-methyl-4-[4-(propan-2-yl)piperazine-1-carbonyl]-1H-pyrazol-1-yl}pyrimidine
N-(3-{2-[2-(propan-2-yl)pyrimidin-4-yl]-1H-imidazol-1-yl}phenyl)acetamide
N-(2-hydroxyethyl)-2-(2-oxopiperidin-1-yl)-N-(1,3-thiazol-2-ylmethyl)acetamide
2-(3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidine-1-carbonyl)benzonitrile
(3R,4R)-1-[(2,3-dichloro-4-methylphenyl)methyl]-4-(hydroxymethyl)piperidin-3-ol
N-[(3R,5S)-5-(diethylcarbamoyl)-1-(3-methylbutyl)pyrrolidin-3-yl]-2-hydroxypyridine-3-carboxamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[1-(prop-2-ene-1-sulfonyl)piperidin-3-yl]piperazine
2-(2,4-difluorophenyl)-5-(oxolane-3-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
2-[(isoquinolin-5-yloxy)methyl]-N-methyl-N-(1-methylpiperidin-4-yl)-1,3-oxazole-4-carboxamide
N-[(3,4-dimethoxyphenyl)methyl]-3-(4-fluorophenyl)-N-(pyridin-4-ylmethyl)benzamide
3-cyclohexyl-N-(1-cyclopropanecarbonylazepan-3-yl)-1H-pyrazole-4-carboxamide
1-{3-[3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl]phenyl}pyrrolidin-2-one
3-({5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}amino)propan-1-ol
(4-{[1-(5-ethylthiophene-3-carbonyl)pyrrolidin-3-yl]methyl}phenyl)methanol
2-(dimethylamino)-7-[2-(1H-pyrazol-1-yl)benzoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(3S,9aR)-3-[(2S)-butan-2-yl]-8-(4-chlorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4,4,4-trifluoro-N-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]butanamide
(1S,4S)-2-(2-chlorophenyl)-5-{[3-(trifluoromethyl)phenyl]methyl}-2,5-diazabicyclo[2.2.1]heptan-3-one
(3aR,6aR)-2-cyclopentyl-5-[4-(hydroxymethyl)benzoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N4-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)pyrimidine-2,4-diamine
N-(1-{1-[(2E)-3-(2-fluorophenyl)prop-2-enoyl]piperidin-4-yl}-2-phenylethyl)-N,1-dimethyl-1H-pyrazole-3-carboxamide
1-[1-(2-phenylethyl)piperidin-4-yl]-N-(piperidin-4-ylmethyl)piperidine-3-carboxamide
N-methyl-2-(2-oxo-1,3-oxazolidin-3-yl)-N-[(1-phenylpyrrolidin-3-yl)methyl]acetamide
[4-(5-chloro-2-methoxypyridin-4-yl)-3-(hydroxymethyl)phenyl]methanol
2-chloro-N-{1-[1-(2,2-dimethylpropyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide