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(2S,4R)-1-[(3-fluorophenyl)methyl]-N,N-dimethyl-4-[(1-methyl-1H-imidazol-2-yl)sulfanyl]pyrrolidine-2-carboxamide
1-[1-(2-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-2-{[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}ethan-1-one
1-acetyl-N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}piperidine-4-carboxamide
1-[(3-methoxyphenyl)methyl]-5-{6-methyl-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}piperidin-2-one
4-{8-methoxy-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-3-methyl-1-propyl-1H-pyrazole
1-{1-[(2-hydroxy-3-methylphenyl)methyl]piperidin-4-yl}pyrrolidin-2-one
(3S,5S)-1-benzyl-5-[(4-fluorophenyl)carbamoyl]piperidine-3-carboxylic acid
1-methyl-3-{[4-(pyridin-4-yl)piperidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
dimethyl(2-{[(3-methyl-1H-pyrazol-5-yl)methyl][(3-methylthiophen-2-yl)methyl]amino}ethyl)amine
4-ethoxy-2-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]pyrimidine
1-{3,3-dimethyl-2-methylidenebicyclo[2.2.1]heptane-1-carbonyl}-3-(1H-imidazol-1-ylmethyl)piperidine
3-(N-methyl-1-{1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidin-3-yl}formamido)propanamide
1-(4-aminopyrimidin-2-yl)-4-(2-phenylethyl)piperidine-4-carboxylic acid
1-{[1-(2-chlorophenyl)-1H-pyrazol-4-yl]methyl}-4-methylpiperidine-4-carbonitrile
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)-2-(1H-pyrazol-1-yl)benzamide
1-(cyclopentylmethyl)-4-{[3-(3-fluorophenyl)oxolan-3-yl]methyl}piperazine
2-(dimethylamino)-2-(3-methylphenyl)-N-[3-(pyridin-4-yl)propyl]acetamide
9-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(butan-2-yl)-2-hydroxy-4-methoxy-N-(pyridin-3-ylmethyl)benzamide
4-(3,3-difluoropiperidine-1-carbonyl)-6-ethyl-2-(1-methyl-1H-pyrazol-4-yl)quinoline
1'-[1-(propan-2-yl)piperidine-4-carbonyl]-3,4-dihydrospiro[1-benzopyran-2,3'-pyrrolidine]-4-one
methyl 5-[(2-methylbutyl)amino]-3-(oxolane-2-amido)-1-(2-phenylethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-(1-methoxypropan-2-yl)-5-[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
(2S,4S)-4-amino-1-{2-[2-(3-methoxyphenyl)ethyl]benzoyl}pyrrolidine-2-carboxylic acid
2-(1-cyclopropanecarbonylpiperidin-4-yl)-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-methanesulfonyl-4-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]piperazine
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-2-(phenylsulfanyl)acetamide
8-[2-(3,4-dimethyl-6-oxo-1,6-dihydropyridazin-1-yl)acetyl]-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
3-{1-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}propanoic acid
3-benzyl-4-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]piperazin-2-one
2-(1-cyclopentyl-3-oxopiperazin-2-yl)-N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-N-methylacetamide
N-{[2-(4-acetylpiperazin-1-yl)pyridin-3-yl]methyl}-2,2,3,3-tetramethylcyclopropane-1-carboxamide
2-[3-(3-fluorophenyl)-2,5-dioxo-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]-N-methyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]acetamide
5-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3-ethyl-1-(propan-2-yl)-1H-1,2,4-triazole
N-{4-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidin-1-yl]-4-oxobutyl}acetamide
1-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-3-(3-methoxy-1,5-dimethyl-1H-pyrazol-4-yl)urea
3-(4-chloro-2-methylbenzoyl)-1-(1H-imidazol-2-ylmethyl)piperidine
1-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]piperidine-2-carboxamide
N-(2-{7-[(4-methoxy-2,5-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-2-carboxamide
(2,1,3-benzoxadiazol-5-ylmethyl)(methyl)[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]amine
2-methyl-2-[4-(morpholin-4-yl)-2-[(oxan-2-ylmethyl)amino]pyrimidin-5-yl]propanoic acid
5-[8-(2-methoxyethyl)-9-oxo-2,8-diazaspiro[5.5]undecane-2-carbonyl]pyridine-2-carbonitrile
N-(1-{7-[(2,4-difluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)oxolane-3-carboxamide
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]acetamide
N-[3-(furan-2-amido)-4-methoxyphenyl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
1-[1-(cyclopropanesulfonyl)azepan-3-yl]-3-(2,4-difluorophenyl)urea
N-(3-acetylphenyl)-3-(5-fluoro-2-methoxybenzoyl)piperidine-1-carboxamide
(3aR,6aS)-N-[2-(benzyloxy)phenyl]-octahydropyrrolo[3,4-c]pyrrole-2-carboxamide
2-(3-chloro-4-hydroxyphenyl)-1-[(1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
(3R,4R)-N-(3,4-dichlorophenyl)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidine-1-carboxamide