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N-{2-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}methanesulfonamide
N-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}pyrazin-2-amine
(2S,4S)-N-ethyl-4-(3-methoxypropanamido)-1-(2-methylpyrimidine-5-carbonyl)pyrrolidine-2-carboxamide
8-(2-fluoro-4-methylbenzoyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(4-{4-[(2H-1,3-benzodioxol-5-ylmethyl)amino]piperidin-1-yl}benzoyl)piperidin-3-ol
2-cyclohexyl-N-[(2S)-1-hydroxy-4-(methylsulfanyl)butan-2-yl]-1,3-benzoxazole-6-carboxamide
{[5-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-3-yl]methyl}({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
(1R,5S)-6-[3-(1,4-diazepane-1-sulfonyl)benzoyl]-6-azabicyclo[3.2.1]octane
N-methyl-N-[(3-methyl-1H-indol-2-yl)methyl]-2-(pyridin-3-yloxy)acetamide
1-[2-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-4-(3-methylphenyl)piperazine
N-{2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]pyridin-3-yl}-2-methylpropanamide
3-{1-[4-(4-fluorophenyl)butanoyl]piperidin-3-yl}-N-(4-methoxy-2-methylphenyl)propanamide
ethyl 1-{[1-(2-methoxyethyl)-2-oxo-1H,2H,6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}piperidine-3-carboxylate
{3-ethyl-1-[1-(morpholin-4-yl)cyclohexanecarbonyl]piperidin-3-yl}methanol
1-(cyclopropylmethyl)-3-hydroxy-3-{[methyl(quinolin-4-ylmethyl)amino]methyl}piperidin-2-one
9-ethyl-1-methyl-4-(quinoxalin-2-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
N-{[7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclopent-1-ene-1-carboxamide
(2S)-1-{5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-1H-pyrazole-3-carbonyl}-4-methyl-2-(propan-2-yl)piperazine
1,3-dimethyl-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
7-[ethoxy(phenyl)methyl]-4-{imidazo[1,2-a]pyridine-2-carbonyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-(5-phenyl-1,2-oxazole-3-carbonyl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
1-cyclohexyl-4-[4-(dimethylamino)phenyl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
methyl (2S,4R)-4-(5-chloro-3-phenyl-1H-indole-2-amido)-1-[(3-fluorophenyl)methyl]pyrrolidine-2-carboxylate
4-methyl-2-[1-(5-methylpyrazine-2-carbonyl)piperidin-3-yl]-1H-1,3-benzodiazole
9-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-2-[(1r,4r)-4-hydroxycyclohexyl]-2,9-diazaspiro[5.5]undecan-3-one
[(3R,4R)-1-(6-chloro-1,3-benzothiazol-2-yl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
5,8-dichloro-3-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-3,4-dihydroquinazolin-4-one
(3R,4R)-1-{[5-(2-fluorophenyl)furan-2-yl]methyl}-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
methyl (2S,4S)-1-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}-4-propanamidopyrrolidine-2-carboxylate
4-methoxy-N-(2-methoxyethyl)-2-[(1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)oxy]benzamide
(2S,4R,5R)-8-amino-10-(4-methanesulfonylphenyl)-5-methyl-2-(propan-2-yl)-7-azatricyclo[4.4.0.02,4]deca-1(6),7,9-triene-9-carbonitrile
3-({1-[2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carbonyl]pyrrolidin-3-yl}methyl)benzamide
4-[1-(3-cyclopropylpropanoyl)piperidin-3-yl]benzoic acid
1-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)-4-(pyridin-2-yl)piperazine
(4aS,8aR)-6-(1H-1,3-benzodiazole-5-carbonyl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
1'-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]-3H-spiro[2-benzofuran-1,4'-piperidine]-3-one
N,N-dimethyl-2-[(1S,5R)-6-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
(1R,5R)-6-(2-cyanobenzoyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
2-[4-(5-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]pyridine-3-carbonitrile
3-[2-(4-methoxy-4-phenylpiperidin-1-yl)-2-oxoethyl]-1,3-diazinane-2,4-dione
(3aS,6aR)-3-[2-(piperidin-1-yl)ethyl]-5-[5-(trifluoromethyl)pyridin-2-yl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-(phenylsulfanyl)-1-[1-(pyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]ethan-1-one
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-8-fluoroquinoline-2-carboxamide
2-(4-methoxy-1H-indol-1-yl)-N-[1-(thiophen-2-ylmethyl)-1H-pyrazol-5-yl]acetamide
1-methyl-N-{3-[5-methyl-4-({[2-(methylsulfanyl)phenyl]formamido}methyl)-1,3-oxazol-2-yl]phenyl}piperidine-3-carboxamide
[(2-cyclohexylpyrimidin-5-yl)methyl](methyl)[1-(pyridin-3-yl)ethyl]amine
1'-(4-methanesulfonylbenzoyl)-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
2-cyclopropyl-1-[(2R,3R,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
4-{1-[2-(cyclohex-1-en-1-yl)ethyl]-1H-imidazol-2-yl}benzamide