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N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
1-(2-methoxyphenyl)-5-[(3-methyl-1,2-oxazol-5-yl)methyl]-3-(2-methylpropyl)-1H-1,2,4-triazole
5-benzyl-3-{[2-(3-fluorophenyl)-1H-imidazol-1-yl]methyl}-1,2,4-oxadiazole
1-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-6-(thiophene-3-carbonyl)-6-azaspiro[2.5]octane
[3-propyl-1-(3-propyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]methanol
3-[(3R,4S)-4-(dimethylamino)-1-{[5-(2-fluorophenyl)furan-2-yl]methyl}piperidin-3-yl]propan-1-ol
(2R)-N1-(2-methylquinolin-8-yl)pyrrolidine-1,2-dicarboxamide
1-[(1S,5R)-6-(3-methylbenzenesulfonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
4-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2-(2-phenylethyl)morpholine
{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}({1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl})amine
6-fluoro-4-[4-(2-methoxyacetyl)-1,4-diazepane-1-carbonyl]-1,2,3,4-tetrahydroquinolin-2-one
(3S,9aR)-3-(cyclohexylmethyl)-8-(4-methylbenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
[(3R,4R)-1-(3,4-dimethoxybenzoyl)-4-{[ethyl(methyl)amino]methyl}pyrrolidin-3-yl]methanol
3-{1-[2-(2H-indazol-2-yl)acetyl]piperidin-3-yl}-N-(4-methoxy-2-methylphenyl)propanamide
4-[(4-ethoxyphenyl)methyl]-3-{2-[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin-1-yl]-2-oxoethyl}piperazin-2-one
(1R,5S,6S)-6-{[4-(thiophen-2-ylmethyl)piperazin-1-yl]methyl}-3-azabicyclo[3.1.0]hexane
9-(cyclopropylmethyl)-1-methyl-4-{[2-(methylamino)-1,3-thiazol-4-yl]methyl}-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
2-{4-[(2,6-difluorophenyl)methyl]-1-[(2-ethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-3-azaspiro[5.5]undecan-9-amine
3-({1-[2-(morpholin-4-yl)acetyl]pyrrolidin-3-yl}methyl)benzoic acid
1-[2-methoxy-4-({[2-(2-methylphenyl)ethyl]amino}methyl)phenoxy]-3-(morpholin-4-yl)propan-2-ol
{1-[2-(cyclopentylamino)ethyl]piperidin-2-yl}methanol
2-{3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}-N,N-diethylacetamide
(4aS,7aR)-1-(3-hydroxypropanoyl)-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-[2-(1,3-benzothiazol-2-yl)pyrrolidine-1-carbonyl]-2-(2-methoxyethyl)-1,3-benzoxazole
N-{[1-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)piperidin-4-yl]methyl}acetamide
N-[(3R,4R)-3-hydroxy-1-(quinoxalin-2-yl)piperidin-4-yl]pyridine-2-carboxamide
(3aS,6aS)-2-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[4-(morpholine-4-carbonyl)phenyl]-N-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}piperidin-4-amine
6-[4-(3-methylphenoxy)piperidin-1-yl]-9H-purin-2-amine
1-[(2R)-2-(methoxymethyl)pyrrolidin-1-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
methyl 5-(2-phenoxypropanoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
2-(pyridin-3-yl)-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)acetamide
4-amino-1-[(2-chlorophenyl)methyl]pyrrolidin-2-one
2-[3-(2-chlorophenyl)-1-cyclopentyl-2,5-dioxopyrrolidin-3-yl]-N-[(4-fluorophenyl)methyl]-N-methylacetamide
[(2,3-difluoro-6-methoxyphenyl)methyl](methyl)[(1-methylpyrrolidin-3-yl)methyl]amine
(3S,4S)-1-[1-(carbamoylmethyl)piperidine-4-carbonyl]-4-propylpyrrolidine-3-carboxylic acid
4-chloro-5-{[3-(methanesulfonylmethyl)piperidin-1-yl]methyl}-N,N-dimethyl-1,3-thiazol-2-amine
1-{[3-(pyridin-2-ylmethoxy)phenyl]methyl}-4-(pyridin-4-yl)piperazine
3-[5-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
N-[(4-acetamidophenyl)methyl]-2-[(3-hydroxyadamantan-1-yl)amino]acetamide
N-{2-[3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-oxoethyl}-2-methylpropanamide
1-[(4-phenyloxan-4-yl)methyl]-5-[2-({[3-(trifluoromethyl)phenyl]methyl}amino)ethyl]pyrrolidin-2-one
(3R,9aR)-3-[(benzylsulfanyl)methyl]-8-(2,5-difluorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-[4-hydroxy-4-(2-methylquinolin-6-yl)piperidin-1-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
3-(8-methoxy-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]propanamide
1-[4-({[(2S)-1-ethylpyrrolidin-2-yl]methyl}amino)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
3-(2,3-dihydro-1H-inden-2-yl)-1-(2-methoxyethyl)-8-[(4-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}pyridine-3-carboxamide