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N'-(2-ethoxyphenyl)-N-[(6-hydroxypyrimidin-4-yl)methyl]propanediamide
6-[2-fluoro-4-(pyrrolidin-1-ylmethyl)phenoxy]pyridine-3-carbonitrile
3-(2-{1-[(4-methoxyphenyl)methyl]-1H-1,2,4-triazol-5-yl}ethyl)-4,5,6,7-tetrahydro-1H-indazole
N-(4-{[4-(3-hydroxypropyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carbonyl)benzamide
N-(4-fluoro-2-methylphenyl)-2-[3-(1,2-oxazinan-2-yl)propanamido]propanamide
3-butyl-4-(1H-imidazol-2-ylmethyl)-1-methylpiperazin-2-one
1-methyl-N-[3-(pyridin-3-yloxy)propyl]-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-(ethanesulfonyl)-N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]piperidine-4-carboxamide
9-(2-hydroxypyridine-3-carbonyl)-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-(3-methoxyphenoxymethyl)-1-{[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine
({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)(oxolan-3-ylmethyl)(pyridin-3-ylmethyl)amine
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-[(1-methyl-1H-imidazol-2-yl)methyl]pyrrolidine-3-carboxylic acid
N,1-dimethyl-N-[1-(1,3-thiazol-2-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-{[7-fluoro-2-(4-methylphenyl)quinolin-3-yl]methyl}-N-(2-methoxyethyl)furan-2-carboxamide
3-{imidazo[1,2-a]pyridin-2-yl}-N-[1-(thiophen-2-ylmethyl)piperidin-4-yl]propanamide
5-{2-[3-cyclopropyl-1-(2-methylpyridin-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1,2-oxazol-3-ol
(1R,5R)-6-[2-(2-ethyl-1H-imidazol-1-yl)acetyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
2-{1-oxa-8-azaspiro[4.5]decan-8-ylmethyl}benzoic acid
ethyl 4-{[(2-methoxyethyl)({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)amino]methyl}-1H-pyrazole-3-carboxylate
2-(azepan-1-yl)-N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}acetamide
N2-{2-methylthieno[3,2-d]pyrimidin-4-yl}-N1-(pyridin-3-yl)ethane-1,2-diamine
9-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(2,3-dihydro-1H-inden-2-yl)-4-(3-fluoropyridin-4-yl)piperazine
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-1-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]ethan-1-one
2-[2-(3-fluorophenyl)-2-oxoethyl]-5-(morpholin-4-yl)-2,3-dihydropyridazin-3-one
1-[cyclohexyl(methyl)amino]-3-(3-{[(2-methoxy-2-methylpropyl)amino]methyl}phenoxy)propan-2-ol
3-{5-[(4-methylpiperidin-1-yl)sulfonyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
4-benzyl-3-methyl-1-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
4-{4-[(4-methoxyphenyl)methyl]piperazin-1-yl}-2-{[4-(trifluoromethyl)phenyl]methyl}-2,3-dihydro-1H-isoindole-1,3-dione
N-(2-chloro-4-fluoro-5-methylphenyl)-4-[(1S,2S)-2-hydroxycyclohexyl]piperazine-1-carboxamide
1-benzyl-8-[(3,5-dimethylphenyl)methyl]-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(4-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}piperidin-1-yl)ethan-1-one
N-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-2-(1-propylpiperidin-4-yl)acetamide
2-(3-chloro-6-oxo-1,6-dihydropyridazin-1-yl)-N-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]acetamide
2-amino-N-[5-(pentan-2-yl)-1,3,4-thiadiazol-2-yl]-6-(propan-2-yl)pyrimidine-4-carboxamide
2-{4-[(2,4-dichlorophenyl)methyl]morpholin-3-yl}acetic acid
N-({5-[(3,5-dimethylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)methanesulfonamide
5-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-1-(2-phenylethyl)-1H-1,2,4-triazole
1-(4-aminoazepan-1-yl)-2-(3-chlorophenoxy)ethan-1-one
N-[(2,3-dimethoxyphenyl)methyl]-5-{1-[2-(4-methoxyphenyl)ethyl]-1H-pyrazol-3-yl}-4-methyl-1,3-thiazol-2-amine
5-{[(6-methylpyridin-3-yl)oxy]methyl}-N-[2-(3-methylthiophen-2-yl)ethyl]-1,2-oxazole-3-carboxamide
(3S,4R)-1-{3-[4-(dimethylamino)phenyl]propanoyl}-4-phenylpyrrolidine-3-carboxylic acid
5-(pyrrolidin-2-yl)-N-(1,3-thiazol-2-yl)thiophene-2-carboxamide
(3S)-1-[2-(3-phenylpropyl)-1,3-benzoxazole-5-carbonyl]pyrrolidin-3-ol
(3S,4R)-4-(4-fluorophenyl)-1-[2-(2-hydroxyphenyl)acetyl]pyrrolidine-3-carboxylic acid
(3S,9aR)-3-benzyl-8-{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-(benzyloxy)-1-[1-(4-fluorophenyl)cyclopropanecarbonyl]azetidine
2-({3-[3-(trifluoromethyl)benzoyl]piperidin-1-yl}methyl)phenol
5-[4-(piperazin-1-yl)phenyl]thiophene-2-sulfonamide
N-({1-[2-(ethylsulfanyl)ethyl]-1,2,5,6-tetrahydropyridin-3-yl}methyl)acetamide