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1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
5-fluoro-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-4-(pyrrolidin-1-yl)pyrimidin-2-amine
ethyl 5-[({5-cyclopropyl-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-1H-pyrazol-4-yl}formamido)methyl]furan-2-carboxylate
1-[(5-ethylfuran-2-yl)methyl]-N-[2-(pyridin-3-yloxy)phenyl]piperidine-3-carboxamide
5-(3-fluorophenoxymethyl)-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-1H-pyrazole-3-carboxamide
1-(3-methoxyphenoxy)-3-[4-phenyl-5-(pyridin-3-yl)-1H-imidazol-1-yl]propan-2-ol
3-(2-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}-2-oxoethyl)-4-(propan-2-yl)piperazin-2-one
(1S,5R)-6-(cyclopropylmethyl)-3-[6-(trifluoromethyl)pyridin-2-yl]-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(naphthalen-2-yl)ethan-1-one
(3S,4S)-1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-cyclopropylpyrrolidine-3-carboxylic acid
3-{[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]amino}-N-(1,3-thiazol-2-yl)propanamide
[1-(1H-imidazol-1-yl)propan-2-yl]({[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl})amine
1-[2-({1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)ethyl]imidazolidin-2-one
1-[2-(dimethylamino)ethyl]-N-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)-5-oxopyrrolidine-3-carboxamide
1-tert-butyl-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
N-cyclopropyl-3-(3-fluorophenyl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1H-pyrazole-4-carboxamide
ethyl 1-(prop-2-en-1-yl)-5-(pyridine-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
methyl 1-[(3S,5S)-1-[(4-chlorophenyl)methyl]-5-[4-(4-fluorophenyl)piperazine-1-carbonyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
7-methoxy-3-{octahydropyrrolo[1,2-a]piperazin-2-ylmethyl}-1,2-dihydroquinolin-2-one
1-{2-amino-6-[(propan-2-yl)amino]pyrimidin-4-yl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N4-[(1-benzyl-1H-imidazol-2-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
9-[2-(benzyloxy)ethyl]-1,4,9-triazaspiro[5.5]undecan-5-one
2-(2-hydroxypropanoyl)-N-(thiophen-2-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
1-(1-benzothiophen-2-ylmethyl)-4-[2-(morpholine-4-carbonyl)-1-benzofuran-5-yl]piperidin-4-ol
[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)methylamine
7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decane
4-(5-cyclopropyl-1,2-oxazole-3-carbonyl)-1-[(4-methoxyphenyl)methyl]-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
4-[(2-butyl-1H-imidazol-4-yl)methyl]-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
1-{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}-3-propoxypiperidine
(3aR,6aR)-2-methyl-N-[2-(4-sulfamoylphenyl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
4-chloro-3-{1-[1-(1,3-dimethyl-1H-pyrazol-4-yl)ethyl]-1H-imidazol-2-yl}-1-methyl-1H-indazole
3-(1,1-dioxo-1λ6-thiolan-3-yl)-3-(2-hydroxyethyl)-1-(6-methoxy-2H-1,3-benzodioxol-5-yl)urea
N-[(3S,4S)-4-methoxy-1-(propan-2-yl)pyrrolidin-3-yl]-1H-pyrazole-4-carboxamide
N-[2-methyl-1-(7-{[4-(2-methylpropyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)propyl]furan-3-carboxamide
3-[(pyridin-3-ylmethyl)sulfamoyl]-N-(pyrrolidin-3-yl)benzamide
4-[3-cyclopropyl-5-(1,2-oxazol-5-yl)-1H-1,2,4-triazol-1-yl]-2-methylpyridine
4-(furan-3-ylmethyl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-{[(2S,4S)-1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-4-fluoropyrrolidin-2-yl]methyl}cyclohexanecarboxamide
2-{1-[(4-ethoxyphenyl)methyl]-4-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]piperazin-2-yl}ethan-1-ol
1-[(4aR,8aR)-4a-hydroxy-7-[(2Z)-5-methyl-2-phenylhex-2-en-1-yl]-decahydro-2,7-naphthyridin-2-yl]ethan-1-one
[1-(3-chloro-4-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}benzoyl)piperidin-3-yl]methanol
{[5-(cyclohex-3-en-1-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}(methyl)(pyridin-3-ylmethyl)amine
N2-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)pyrrolidine-1,2-dicarboxamide
2-({1-[(4-fluorophenyl)methyl]-1H-1,2,4-triazol-5-yl}methyl)-1,4-dimethylpiperazine
methyl 4-({3-[4-methyl-5-(prop-2-en-1-ylsulfanyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)benzoate
5-[(isoquinolin-5-yloxy)methyl]-N-[(6-methylpyridin-2-yl)methyl]-1,2-oxazole-3-carboxamide
1-(furan-2-ylmethyl)-N-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}piperidine-3-carboxamide
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-methyl-N-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}propanamide
methyl 6-(2,2-dimethylpropanoyl)-2-{[2-(2-fluorophenyl)ethyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-butyl-4-{[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine