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5-chloro-4,6-dimethyl-3-(3-methylpiperazine-1-carbonyl)-1,2-dihydropyridin-2-one
4-amino-2-(4-{[4-(1H-imidazol-1-yl)phenyl]methyl}piperazin-1-yl)pyrimidine-5-carbonitrile
[(3R,4S)-1-[(2,3-dimethoxyphenyl)methyl]-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}pyrrolidin-3-yl]methanol
1-(1H-indazol-5-yl)-4-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]piperazin-2-one
3-chloro-4-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}-N-(oxan-4-ylmethyl)benzamide
1-{[2-chloro-5-methoxy-4-(propan-2-yloxy)phenyl]methyl}azetidine-3-carboxylic acid
4-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-5-propylpyrimidine
2-{4-[(1-propyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}-4,5,6,7-tetrahydro-1,3-benzothiazole
N-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}-1H-1,2,3-triazole-5-carboxamide
(3S)-1-ethyl-3-methyl-4-(3-{5-[(4-phenylphenyl)methyl]-1,3,4-oxadiazol-2-yl}propanoyl)piperazin-2-one
3-cyclohexyl-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-1H-pyrazole-4-carboxamide
4-phenyl-1-[1-(1H-pyrazol-1-yl)propan-2-yl]-5-{pyrazolo[1,5-a]pyrimidin-3-yl}-1H-imidazole
N-[2-(4-fluorophenyl)ethyl]-6,6-dimethyl-5-oxo-N-(pyridin-3-ylmethyl)thiomorpholine-3-carboxamide
2-{4-[(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)sulfonyl]morpholin-3-yl}acetic acid
2-[4-(1,3-dihydroxypropan-2-yl)piperazin-1-yl]pyridine-3-carbonitrile
1-[1-(2,6-difluoro-3-methoxybenzoyl)piperidin-4-yl]-3-methylbutan-1-ol
3-methyl-4-[5-(oxolan-2-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-1-yl]pyridine
(3aS,6aS)-2-methanesulfonyl-5-[2-oxo-2-(piperidin-1-yl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
8-{6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1H-imidazole-2-carboxamide
1-(3-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}phenyl)ethan-1-one
1-[3-(3-fluorophenoxymethyl)piperidin-1-yl]-3-(pyrrolidin-1-yl)propan-1-one
dimethyl[(4-{1-[3-(1H-pyrazol-1-yl)benzoyl]piperidin-2-yl}phenyl)methyl]amine
N5-cyclopropyl-N6-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
2-{2-[4-(1H-imidazol-1-yl)butoxy]phenyl}-6-methyl-1H-1,3-benzodiazole
N-(2-{imidazo[1,2-a]pyridin-3-yl}ethyl)-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]acetamide
8-[(2S)-2-methoxy-2-phenylacetyl]-2-(3-methylbut-2-en-1-yl)-2,8-diazaspiro[4.5]decan-3-one
2-(1,2-oxazol-5-yl)-4-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}phenol
N-[1-(2,5-difluorophenyl)cyclopropyl]-2,7-dioxo-1,3-diazepane-4-carboxamide
1-ethyl-N-[1-(4-fluorophenyl)-5-oxopyrrolidin-3-yl]-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
N-{[(3S,4S)-1-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]-3-hydroxypiperidin-4-yl]methyl}furan-2-carboxamide
N-(1-{1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-4-phenylbutanamide
N-(2-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]formamido}ethyl)acetamide
1-[4-({4-[5-(4-methoxyphenyl)furan-2-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperazin-1-yl]ethan-1-one
7-[(3-methoxyphenyl)methyl]-2-(4,4,4-trifluorobutyl)-2,7-diazaspiro[4.5]decan-6-one
N-[(3-methylpyridin-4-yl)methyl]-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
2-[2-(benzyloxy)phenyl]-2-(4-hydroxypiperidin-1-yl)acetic acid
N-methyl-N,1-diphenyl-3-(propan-2-yl)-1H-1,2,4-triazole-5-carboxamide
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N-methyl-3-(4-methyl-1,3-thiazol-5-yl)propanamide
{1-[(1-hexylpiperidin-3-yl)methyl]-1H-1,2,3-triazol-4-yl}methanol
3-[(2-ethylpyrimidin-4-yl)methyl]-7,11-dimethyl-3,7,11-triazaspiro[5.6]dodecane
2-[2-chloro-6-methoxy-4-({methyl[(1-methyl-5-oxopyrrolidin-3-yl)methyl]amino}methyl)phenoxy]acetic acid
1-(3,6-dimethyl-1-benzofuran-2-carbonyl)-3-(3-methylphenoxy)azetidine
2-(4-methyl-6-{[2-(pyrazin-2-yl)ethyl]amino}pyrimidin-2-yl)phenol
2-[1-(2-hydroxyethyl)-1H-1,3-benzodiazol-2-yl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
(3S,4R)-1-[2-(morpholin-4-yl)-2-oxoethyl]-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
N,N-dimethyl-4-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperazine-1-carboxamide
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-[2-(ethylsulfanyl)ethyl]acetamide
3-{2-oxo-2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethyl}-1λ6-thiolane-1,1-dione
methyl N-(2-{2-[(3-methoxyphenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}-2-oxoethyl)carbamate