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N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
2-cyclopropyl-4-hydroxy-N-{1-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}pyrimidine-5-carboxamide
7-{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-(2-methoxyphenyl)-1-{2-[(4-methoxyphenyl)formamido]ethyl}-1H-1,2,3-triazole-4-carboxamide
N-(3-benzylphenyl)-3-(4-methylpiperazin-1-yl)pyrrolidine-1-carboxamide
2-(dimethylamino)-2-(2-fluorophenyl)-N-[1-(morpholin-4-ylmethyl)cyclopentyl]acetamide
N-[(2R,3R)-1'-(2,2-dimethylpropyl)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
1-benzyl-N3-cyclopropyl-N5-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
4-[(2-methylphenyl)methyl]-1-[(2,3,6-trifluorophenyl)methyl]-1,4-diazepan-5-one
methyl 2-{5-methyl-2-[(2-methylpropanamido)methyl]-2,3-dihydro-1-benzofuran-7-yl}benzoate
ethyl 4-(4-{4-[(2,3-dihydro-1H-inden-2-yl)amino]piperidin-1-yl}benzoyl)piperazine-1-carboxylate
4-benzyl-3-ethyl-1-(1-methyl-1H-pyrrole-2-carbonyl)-1,4-diazepan-5-one
1-[3-(3-methoxyphenyl)-1H-pyrazole-5-carbonyl]-4-(1H-pyrrole-2-carbonyl)piperazine
1-(3-chloro-4-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}benzoyl)piperazine
7-(cyclobutylmethyl)-2-[(4-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decane
(2,3-dihydro-1-benzofuran-2-ylmethyl)({[2-(ethylsulfanyl)pyrimidin-5-yl]methyl})methylamine
5-methanesulfonyl-1'-(2-methyl-1H-pyrrole-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-[(2-fluorophenyl)methyl]-N-methyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
4-({1-[5-(hydroxymethyl)furan-2-carbonyl]pyrrolidin-3-yl}methyl)benzoic acid
[3-(prop-2-en-1-yl)-1-(pyridine-4-carbonyl)piperidin-3-yl]methanol
N-[1-(4-fluorophenyl)-4-(propan-2-yloxy)-1H-indazol-3-yl]-2-(1H-1,2,4-triazol-1-yl)acetamide
N-[4-({8-methyl-2,8-diazaspiro[4.5]decan-2-yl}sulfonyl)phenyl]acetamide
methyl 1-({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidine-4-carboxylate
1-[6-(3-fluorophenyl)pyridine-3-carbonyl]-4-phenylazepane
1-(furan-2-carbonyl)-N-{2-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-3-amine
(5-{[3-(hydroxymethyl)-3-[(3-methoxyphenyl)methyl]piperidin-1-yl]methyl}furan-2-yl)methanol
(cyclohexylmethyl)({[1-(2-methoxyethyl)piperidin-4-yl]methyl})(pyridin-4-ylmethyl)amine
1-(2H-1,3-benzodioxol-5-ylmethyl)-6-methyl-3-[4-(2-methylphenyl)piperazine-1-carbonyl]-2-propyl-1,4-dihydropyridin-4-one
3-({5-[4-(2-phenylethyl)piperidine-1-carbonyl]pyridin-2-yl}amino)butan-1-ol
1-[(4-{[3-(furan-2-yl)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)methyl]-4-(pyridin-3-yl)piperidin-4-ol
5-(2-chlorophenyl)-N-(1H-imidazol-2-ylmethyl)-2-methylfuran-3-carboxamide
2-(2-chlorophenyl)-N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylacetamide
8-[4-(2-methyl-1H-imidazol-1-yl)butanoyl]-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
ethyl 3-[(4-fluorophenyl)methyl]-1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidine-3-carboxylate
N-methyl-N-(1,2-oxazol-5-ylmethyl)-5-[3-(trifluoromethyl)phenoxymethyl]-1H-pyrazole-3-carboxamide
2-(dimethylamino)-2-(4-fluorophenyl)-1-[4-(1H-pyrazol-1-ylmethyl)piperidin-1-yl]ethan-1-one
2-{7-hydroxy-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}-N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}acetamide
6-(3-fluorophenyl)-N-methyl-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
2-[5-(methoxymethyl)-4-[4-(piperidin-1-yl)piperidine-1-carbonyl]-1H-pyrazol-1-yl]-4-(thiophen-2-yl)pyrimidine
4-[(3,5-dimethoxyphenyl)methyl]-1,4-oxazepan-5-one
N-[2-methyl-2-(morpholin-4-yl)propyl]-5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carboxamide
4-ethyl-5-methyl-6-{4-[2-(pyrrolidin-1-yl)ethyl]piperazin-1-yl}pyrimidin-2-amine
methyl 3-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)propanoate
N-ethyl-1-[2-(4-methoxyphenyl)ethyl]-N-(2-methylprop-2-en-1-yl)-6-oxopiperidine-3-carboxamide
ethyl 4-[(4-chlorophenyl)methyl]-1-{spiro[2.4]heptane-1-carbonyl}piperidine-4-carboxylate
N-[2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-2H-1,3-benzodioxole-5-carboxamide
4-[(dimethylamino)methyl]-1-[2-(phenylamino)pyrimidine-5-carbonyl]azepan-4-ol
N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)cyclopropanecarboxamide
N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-6-fluoro-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide