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1-[2-chloro-5-(morpholin-4-yl)phenyl]-3-[2-(2-oxoimidazolidin-1-yl)ethyl]urea
ethyl 4-benzyl-1-{[4-(2-oxoimidazolidin-1-yl)phenyl]methyl}piperidine-4-carboxylate
N-cyclopropyl-1-[3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)propanoyl]piperazine-2-carboxamide
4-amino-2-[4-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)piperazin-1-yl]pyrimidine-5-carbonitrile
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-(1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidin-3-yl)piperazine
{[1,3-dimethyl-5-(morpholin-4-yl)-1H-pyrazol-4-yl]methyl}(methyl)[(3-methyl-1H-indol-2-yl)methyl]amine
2-[2-(1H-imidazol-4-yl)ethyl]-8-[2-(thiophen-3-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-5-methoxybenzamide
1-{[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(pyridin-4-yl)piperazine
9-methoxy-7-(3-methoxyphenyl)-4-[(5-methylthiophen-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
[1-(3-chlorobenzoyl)-3-(2-phenylethyl)piperidin-3-yl]methanol
methyl 1-(2-methylpropyl)-5-[(2-phenylpropyl)amino]-3-(pyridine-3-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
5-[(4-fluoro-3-methoxyphenyl)methyl]-5-{3-oxo-3-[4-(thiophene-2-carbonyl)piperazin-1-yl]propyl}pyrrolidin-2-one
methyl 4-{[(2-{1-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-5-oxopyrrolidin-2-yl}ethyl)amino]methyl}benzoate
4,6-dimethyl-1-{2-[3-(propan-2-yl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1,2-dihydropyrimidin-2-one
3-[3-(2-cyclohexylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-4,6-dimethyl-1,2-dihydropyridin-2-one
4-[(2,2-dimethylpropyl)amino]-1-[(4-fluorophenyl)methyl]pyrrolidin-2-one
methyl 4-[({2-[1-(2-hydroxybutyl)-5-oxopyrrolidin-2-yl]ethyl}amino)methyl]benzoate
2-methoxy-1-{4-[4-(1,2-oxazolidine-2-carbonyl)phenoxy]piperidin-1-yl}ethan-1-one
{1-[1-(piperidine-1-sulfonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methanamine
1-(5-chloro-2-methoxyphenyl)-3-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-3-ethylurea
2-(thiophen-3-ylmethyl)-9-oxa-2-azaspiro[5.5]undecane
7-(5-hydroxypyrazine-2-carbonyl)-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(3S,4S)-1-[(4-methyl-1,3-thiazol-2-yl)methyl]-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
2-fluoro-6-methoxy-N-[2-(1H-pyrazol-4-yl)ethyl]benzamide
4-{4-[(4-methoxy-3-methylphenyl)methyl]piperazin-1-yl}-2-(oxolan-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
methyl[2-(oxan-2-yl)ethyl]({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)amine
(1R,4S)-4-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecane-4-carbonyl}-1,7,7-trimethyl-2-oxabicyclo[2.2.1]heptan-3-one
N-{1-[1-(1H-pyrazol-3-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
[7-(3-methylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methanamine
N-(adamantan-2-ylmethyl)-2-oxo-6-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1,2-dihydropyridine-3-carboxamide
1-[2-(dimethylamino)ethyl]-N-methyl-5-oxo-N-[2-(phenylsulfanyl)ethyl]pyrrolidine-3-carboxamide
3-(1-{1-[(2,6-dimethoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-1-(2-methylphenyl)urea
N-[(2-methoxyphenyl)methyl]-N-(pyridin-3-ylmethyl)-2-(thiophen-2-yl)acetamide
({4-[1-(2H-1,3-benzodioxol-5-yl)-3-cyclopropyl-1H-1,2,4-triazol-5-yl]-1,3-thiazol-2-yl}methyl)dimethylamine
1-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-(2-methoxyphenoxy)piperidine
1-{[2-(1-ethylpiperidin-3-yl)-1H-imidazol-1-yl]methyl}cyclohexan-1-ol
2-{2-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl}pyridine
N,N-dimethyl-2-[N-methyl-2-(2-methyl-4-oxo-1,4-dihydroquinolin-1-yl)acetamido]propanamide
3-[2-(2-fluorophenyl)ethyl]-1-(oxane-4-carbonyl)piperidine
4-ethyl-1-[(4-methoxy-2,5-dimethylphenyl)methyl]-1,4-diazepan-5-one
1-[(5-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]pyrrolidine
N-[1-benzyl-4-(propan-2-yloxy)-1H-indazol-3-yl]-3-(4H-1,2,4-triazol-4-yl)propanamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-{[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}piperazine
2-benzyl-8-cyclopropanecarbonyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-ethyl-7-{4-[(4-fluorophenyl)sulfanyl]piperidine-1-carbonyl}-1-(3-methoxypropyl)-1H-1,3-benzodiazol-5-amine
4-[(4-fluorophenyl)methyl]-1-[2-(methylamino)acetyl]-3-(propan-2-yl)-1,4-diazepan-5-one
2-(3-methoxypropyl)-9-[3-(pyridin-3-yl)propyl]-2,9-diazaspiro[5.5]undecan-3-one
7-(3-chlorophenyl)-4-(5-ethyl-1,2-oxazole-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[1-(cyclohex-1-en-1-yl)ethyl]-1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide