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(3S,4R)-1-[(cyclohexylcarbamoyl)methyl]-4-(3-fluorophenyl)pyrrolidine-3-carboxylic acid
methyl(1,2-oxazol-3-ylmethyl)[(4-{[1-(2,3,4,9-tetrahydro-1H-carbazole-6-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]amine
3-methyl-1-[1-(6-{[(3-methylpyridin-2-yl)methyl]amino}pyridine-3-carbonyl)piperidin-3-yl]butan-1-one
1-[2-(4-chlorophenyl)morpholin-4-yl]-2-(dimethylamino)ethan-1-one
3-[1-(2H-1,3-benzodioxol-5-ylmethyl)-1H-1,2,4-triazol-5-yl]-1H,2H,5H,6H,7H-cyclopenta[b]pyridin-2-one
(4aR,7aS)-6,6-dioxo-N-[2-(1H-pyrazol-1-yl)phenyl]-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
N-{[(2S,4S)-4-fluoro-1-[(phenylcarbamoyl)carbonyl]pyrrolidin-2-yl]methyl}pyridine-4-carboxamide
N-[1-(2-fluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]quinoxaline-5-carboxamide
4-(benzylamino)-1-[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonan-3-yl]butan-1-one
2-[3-(phenoxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1,8-naphthyridine
2-[3-(3-methyl-1H-1,2,4-triazol-5-yl)piperidine-1-carbonyl]-4-(1H-1,2,3,4-tetrazol-1-yl)phenol
5-(2,6-difluorophenoxymethyl)-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-1,2-oxazole-3-carboxamide
3-{1-[2-(2H-1,2,3-benzotriazol-2-yl)acetyl]piperidin-4-yl}-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
4-methyl-2-{1-[(3-methyl-1,2-oxazol-5-yl)methyl]piperidin-4-yl}-1H-1,3-benzodiazole
4-{[4-(dimethylamino)-5-methylpyrimidin-2-yl]amino}-1-propylpyrrolidin-2-one
5-(4-acetylphenoxymethyl)-N-(2-hydroxyethyl)-N-methyl-1,2-oxazole-3-carboxamide
(1S,5R)-6-(4-chloro-1,5-dimethyl-1H-pyrazole-3-carbonyl)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
5-{[2-(2-oxoimidazolidin-1-yl)ethyl]amino}-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
3-[1-(4-methoxyphenyl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl]piperidine-1-carboxamide
2-phenyl-5,6,7,8-tetrahydroquinazolin-5-amine
2-[(1S,5R)-6-{[5-(2-fluorophenyl)furan-2-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
1-(2-oxo-2-{2-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidin-1-yl}ethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-(2-chlorophenyl)-4-[2-(oxolan-2-ylmethoxy)acetyl]piperazin-2-one
(3aS,6aS)-2-(ethanesulfonyl)-5-[2-(phenylsulfanyl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(2,6-dioxo-1,3-diazinan-1-yl)-N-methyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]acetamide
N-[2-oxo-2-(pyrrolidin-1-yl)ethyl]-3-(1H-pyrazol-1-yl)benzamide
methyl 2-[(4-methylphenyl)sulfamoyl]-6-(2-methylpropanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
(3aS,6aS)-2-[(4-chloro-2-fluorophenyl)methyl]-5-cyclobutanecarbonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(5-methyl-1H-pyrazol-1-yl)ethan-1-one
3-(1-hydroxy-3-methylbutan-2-yl)-5-methyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
1-butyl-3-[(4-methoxyphenyl)methyl]-5-[1-(1H-1,2,4-triazol-1-yl)ethyl]-1H-1,2,4-triazole
methyl (2R,4S)-1-(4-ethenylbenzoyl)-4-hydroxypiperidine-2-carboxylate
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-1-(2-methylpropyl)piperidin-4-amine
4-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]methyl}-1,3-thiazole
N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-4-(pyridin-2-yl)pyrimidin-2-amine
1-[(3R,4S)-4-(dimethylamino)-3-(3-hydroxypropyl)piperidin-1-yl]-3-(3-fluorophenyl)propan-1-one
9-{[2-(methylsulfanyl)phenyl]methyl}-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[2-methyl-3-(pyrrolidine-1-carbonyl)phenyl]-3-[3-(4H-1,2,4-triazol-4-yl)propyl]urea
N,N-diethyl-1-{[8-methyl-2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}pyrrolidin-3-amine
2-(2H-1,3-benzodioxol-5-ylmethyl)-4-[4-(thiophen-2-ylmethyl)piperazin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
3-(3-fluorophenyl)-N-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)-1H-pyrazole-4-carboxamide
N-cyclohexyl-4-methyl-N-(pyridin-3-ylmethyl)pyrimidine-5-carboxamide
2-[methyl({4-methyl-5-[1-(4-methyl-1H-pyrrole-2-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)amino]ethan-1-ol
2-(5-amino-1,3,4-thiadiazol-2-yl)-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}acetamide
1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine-3-carboxamide
N-methyl-4-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyridin-2-amine
1-(adamantan-2-yl)-3-(3,4-dimethoxybenzoyl)piperidine
1-benzyl-3-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
N-(1-{7-[(2-hydroxy-3-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)pyridine-3-carboxamide
N-{[7-chloro-2-(3-methylphenyl)quinolin-3-yl]methyl}-N-(2-methoxyethyl)furan-2-carboxamide