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4-(4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-3-fluoropyridine
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)-5-(2-methylpropyl)-1,2-oxazole-3-carboxamide
3-ethyl-8-[1-(2-fluorophenyl)cyclopropanecarbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
9-[(2S)-2-(dimethylamino)-3-phenylpropanoyl]-2-ethyl-2,9-diazaspiro[5.5]undecan-3-one
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]oxane-4-carboxamide
4-(4-chlorophenyl)-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]butanamide
5-[2-fluoro-6-(propan-2-yloxy)phenyl]thiophene-2-carboxamide
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}-4-(1H-pyrazol-1-yl)butanamide
2-[2-({6-ethyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)ethyl]-1,2,3,4-tetrahydrophthalazine-1,4-dione
[(3R,4S)-1-[(4-fluoro-3-methoxyphenyl)methyl]-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
3-{5-[methoxy(phenyl)methyl]-1,3,4-oxadiazol-2-yl}-1-[4-(3-methylphenoxy)piperidin-1-yl]propan-1-one
N-[(5-benzyl-1,2,4-oxadiazol-3-yl)methyl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
N-[(3-ethoxy-4-methoxyphenyl)methyl]-N-methyl-N'-(4-methylphenyl)propanediamide
4-{1-[1-(cyclohex-1-ene-1-carbonyl)piperidin-4-yl]piperidine-4-carbonyl}morpholine
1,3-dimethyl-N-{[1-(morpholin-4-yl)cycloheptyl]methyl}-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
4-(propan-2-yl)-N-[4-(pyrrolidin-1-yl)butyl]pyrimidin-2-amine
N-ethyl-2,2-dimethyl-N-(pyridin-4-ylmethyl)oxan-4-amine
(3aR,5S,6S,7aS)-2-[1-(3-chloro-4-methylphenyl)piperidin-4-yl]-octahydro-1H-isoindole-5,6-diol
N-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
7-acetamido-2-(2-methoxyphenyl)-N,1-dimethyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
(1S,9aR)-1-{[4-(1,3-benzoxazol-2-yl)piperazin-1-yl]methyl}-octahydro-1H-quinolizine
methyl({[1-(3-methylbutyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl})(oxan-2-ylmethyl)amine
N,1,3-trimethyl-N-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N-ethyl-5-methyl-6-(4-methylpiperazine-1-carbonyl)thieno[2,3-d]pyrimidin-4-amine
1-[4-(2-hydroxyphenyl)piperazin-1-yl]-2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
5-({ethyl[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]amino}methyl)-N-(propan-2-yl)pyrimidin-2-amine
2-[3-(1H-indol-3-yl)-5-{[4-(propan-2-yl)morpholin-2-yl]methyl}-1H-1,2,4-triazol-1-yl]ethan-1-ol
N,N,7,8-tetramethyl-2-[2-(propan-2-yl)pyrimidin-5-yl]quinoline-4-carboxamide
N-[1-(butan-2-yl)-1H-pyrazol-5-yl]-2-(3-methylphenyl)acetamide
5-[3-(methoxymethyl)piperidine-1-carbonyl]-N-methyl-N-[2-(oxan-4-yl)ethyl]pyridin-2-amine
6-{6-amino-1H-pyrrolo[2,3-b]pyridin-4-yl}-4-methyl-1,2-dihydroquinolin-2-one
(2S,4R)-4-amino-N,N-diethyl-1-(1H-indole-5-carbonyl)pyrrolidine-2-carboxamide
(3S)-4-{4-[(1-cyclopentylpiperidin-4-yl)oxy]-3-methoxybenzoyl}-1,3-dimethylpiperazin-2-one
propyl (4aR,7aS)-4-[(1-ethyl-1H-imidazol-2-yl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxylate
1-(5-cyclobutyl-1,3,4-oxadiazol-2-yl)-4-(3-methyl-1H-1,2,4-triazol-5-yl)piperidine
N-(3-{[(2-hydroxy-3-phenylpropyl)carbamoyl]methoxy}phenyl)propanamide
N-cyclohexyl-9-(2-methoxyethyl)-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecane-4-carboxamide
2-(3-fluorophenoxymethyl)-N-[(1R)-1-(4-methoxyphenyl)ethyl]-1,3-oxazole-4-carboxamide
ethyl 4-{[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]amino}piperidine-1-carboxylate
2-{3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidin-4-amine
2-[(dimethylamino)methyl]-4-{1-[2-(pyridin-3-yl)ethyl]-1H-imidazol-2-yl}phenol
(3S,4S)-4-(propan-2-yl)-1-{2-[(propan-2-yl)amino]pyrimidine-5-carbonyl}pyrrolidine-3-carboxylic acid
2-[1-(2,3-dihydro-1-benzofuran-5-ylmethyl)piperidin-3-yl]-6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline
1-[2-(propan-2-ylsulfanyl)acetyl]-N-(pyridin-3-ylmethyl)piperazine-2-carboxamide
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-3-oxo-2,3-dihydro-1H-indene-1-carboxamide
N-methyl-2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)sulfanyl]-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
[7-(2,4-dimethoxypyrimidin-5-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methanamine
{[1-benzyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine
{[1-butyl-2-(cyclohexanesulfonyl)-1H-imidazol-5-yl]methyl}(1,4-dioxan-2-ylmethyl)methylamine
(3R,4R)-4-cyclopropyl-1-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-3-methylpiperidin-4-ol