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(3S,9aR)-3-propyl-8-(2,4,5-trifluorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-({2-[2-(morpholin-4-ylmethyl)phenyl]phenyl}methyl)propanamide
2-(ethylamino)-N-[(2-methyl-1,3-thiazol-4-yl)methyl]pyrimidine-5-carboxamide
N-(5-{[1-(pyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}thiophen-2-yl)acetamide
N-[(2-chlorophenyl)methyl]-1-(diphenylmethyl)-N-methyl-1H-1,2,3-triazole-4-carboxamide
{[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[2-(4,6-dimethylpyrimidin-2-yl)ethyl]amine
3-(5-methylfuran-2-yl)-N-[3-(4-methylpiperazin-1-yl)butyl]benzamide
8-(furan-3-ylmethyl)-3-[(4-methoxyphenyl)methyl]-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{3-[9-methoxy-7-(3-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]phenyl}pyrrolidin-2-one
4-(4-chlorophenoxy)-N-(2-ethoxyethyl)piperidine-4-carboxamide
3-{5-[2-(3,4-dimethoxyphenyl)ethyl]-1,2,4-oxadiazol-3-yl}pyridazine
2-(dimethylamino)-2-(2-methylphenyl)-N-[(4-phenyloxan-4-yl)methyl]acetamide
N-(2-{[2-(morpholin-4-yl)pyrimidin-5-yl]formamido}ethyl)pyridine-3-carboxamide
(1-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-1,3-benzodiazol-2-yl)methanol
2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]-1-[4-(6-methylpyridin-2-yl)piperazin-1-yl]ethan-1-one
1-(cyclohexylmethyl)-4-[3-(2-hydroxyethoxy)phenyl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl){[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amine
3-[3-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]-6-methylpyridazine
1-[2-(4-methoxyphenyl)ethyl]-6-oxo-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]piperidine-3-carboxamide
N-[(1,2-dimethyl-1H-1,3-benzodiazol-5-yl)methyl]-2,3-dimethylquinoxaline-6-carboxamide
7-(cyclohexylmethyl)-2-cyclopropanecarbonyl-2,7-diazaspiro[4.5]decan-6-one
3-(1,2-dihydroacenaphthylene-5-carbonyl)-1-[(trimethyl-1H-pyrazol-4-yl)sulfonyl]piperidine
2-amino-N-[(4,6-dimethylpyrimidin-2-yl)methyl]-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
4-methyl-2-{2-[2-(2,5,7-trimethyl-1H-indol-3-yl)acetamido]ethyl}-1,3-thiazole-5-carboxylic acid
2-{1-[(4-ethoxyphenyl)methyl]-4-[(1-ethyl-1H-imidazol-2-yl)methyl]piperazin-2-yl}ethan-1-ol
5-[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl]-3,4-dihydropyrimidin-4-one
{4-fluoro-3-[(E)-2-phenylethenyl]phenyl}methanamine
N-[2-(oxolan-2-ylmethoxy)phenyl]-4-(pyridin-2-yl)piperazine-1-carboxamide
4-(3-methoxyphenyl)-6-methylpyrimidin-2-amine
3-(tert-butylsulfamoyl)-5-{[(4-fluorophenyl)methyl]amino}-N-[(1-methylpiperidin-3-yl)methyl]benzamide
1-(2-methylpropyl)-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
2-(6-chloro-2H-1,3-benzodioxol-5-yl)-4-{[2-(4-fluorophenyl)pyrrolidin-1-yl]methyl}-5-methyl-1,3-oxazole
1-methyl-N-(2-methylpropyl)-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[(4-hydroxyphenyl)methyl]-2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-1H-1,3-benzodiazole-5-carboxamide
N-[1-(thian-4-yl)piperidin-4-yl]-1,2-oxazole-3-carboxamide
3-[(3R,4S)-4-(dimethylamino)-1-(4-methoxyquinoline-2-carbonyl)piperidin-3-yl]propan-1-ol
2-[3-(4-methoxyphenoxymethyl)piperidine-1-carbonyl]benzonitrile
1-(3-methylpyridin-2-yl)-4-[4-(propan-2-yl)-1,3-thiazole-2-carbonyl]piperazine
2-(4-{[4-(prop-2-en-1-yl)piperazin-1-yl]methyl}phenyl)-6-(pyridin-3-yl)-3,4-dihydropyrimidin-4-one
(3R)-1-[6-methyl-2-(pyridin-3-yl)pyrimidin-4-yl]pyrrolidin-3-ol
(4aR,8aS)-1-{6-chloroimidazo[1,2-a]pyridine-2-carbonyl}-6-(4-fluorobenzoyl)-decahydro-1,6-naphthyridine
1-{2-[methyl({[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl})amino]ethyl}cyclopentan-1-ol
1-[2-(4-methoxyphenyl)ethyl]-8-[(4-methoxyphenyl)methyl]-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[(2R)-2-aminopropanoyl]-N-[4-(2-fluorophenoxy)phenyl]piperidine-4-carboxamide
3-[(2,5-difluorophenyl)methyl]-6,7-dimethoxy-3,4-dihydroquinazolin-4-one
(2S)-1-(2-{tricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}acetyl)pyrrolidine-2-carboxamide
N-cyclobutyl-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamide
5-ethyl-6-methyl-N4-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)pyrimidine-2,4-diamine
2-({3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-yl}carbonyl)benzonitrile
1-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(4-methyl-1,2,5-oxadiazol-3-yl)piperazine