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9-methoxy-3-{[4-(2-methylphenyl)phenyl]methyl}-10-(pyrrolidine-1-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
3-[2-(ethoxymethyl)pyrrolidine-1-carbonyl]-8-fluoro-1,4-dihydroquinolin-4-one
2-[(7-methyl-1H-indol-3-yl)methyl]-2,8-diazaspiro[4.5]decane
N-(3-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)-2-(1H-1,2,3,4-tetrazol-1-yl)acetamide
2-{1-[(4-methanesulfonylphenyl)methyl]pyrrolidin-2-yl}-4-methyl-1H-1,3-benzodiazole
4-{[2-(5-ethylfuran-2-yl)-1H-imidazol-1-yl]methyl}-1-(propan-2-yl)pyrrolidin-2-one
3-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidine-1-carbonyl]piperidine-1-carboxamide
5-[2-(aminomethyl)-2,3-dihydro-1-benzofuran-7-yl]-N-(2-fluorophenyl)furan-2-carboxamide
9-(5-fluoro-2-methylbenzoyl)-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
(1-{[methyl({6-[(propan-2-yl)amino]pyrimidin-4-yl})amino]methyl}cyclobutyl)methanol
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1-phenylcyclohexane-1-carboxamide
3-[3-(2-methyl-1H-imidazol-1-yl)propyl]-1,3-diazinane-2,4-dione
{3-[(3-chlorophenyl)methyl]-1-(1,3-thiazol-2-yl)piperidin-3-yl}methanol
(3R)-1-(5,6-dimethylpyrazin-2-yl)-3,4,4-trimethylpyrrolidin-3-ol
1-[(2-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-ylmethyl}phenyl)methyl]-1H-pyrazole
N-cyclopentyl-4-oxo-4-{4-[2-oxo-2-(pyrrolidin-1-yl)ethyl]piperazin-1-yl}butanamide
1-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrol-1-yl]-2-(4-methyl-1,2,5-oxadiazol-3-yl)ethan-1-one
3-(pentan-2-yl)-8-(4,4,4-trifluorobutanoyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(2,1,3-benzothiadiazole-4-sulfonyl)-N-methyl-N-[2-(pyridin-2-yl)ethyl]piperidin-3-amine
(2S,4R)-4-amino-1-[2-(2-fluorophenyl)benzoyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-2-oxo-1,2-dihydroquinoline-4-carboxamide
ethyl 2-(3-{2-[(4-methoxy-2-methylphenyl)carbamoyl]ethyl}piperidin-1-yl)pyridine-3-carboxylate
1-[(3S)-3-(dimethylamino)azepan-1-yl]-2-(pyridin-4-yl)ethan-1-one
N-(1-{1-[(5-acetylthiophen-3-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
3-(azepane-1-carbonyl)-N,1-dimethyl-N-(thiophen-3-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-cyclopropyl-1-[1-(pyrimidin-2-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
2-{2-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepan-1-yl]-2-oxoethyl}-6-methyl-2,3-dihydropyridazin-3-one
1-[4-hydroxy-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidin-1-yl]-2-(1H-indazol-1-yl)ethan-1-one
1-methyl-4-({1-[(3-methylphenyl)methyl]-5-(oxan-2-yl)-1H-1,2,4-triazol-3-yl}methyl)piperidine
3-(2,5-dioxoimidazolidin-4-yl)-N-[1-(2-fluorophenyl)piperidin-4-yl]propanamide
N-[2-(5-chloro-2-methyl-1H-indol-3-yl)ethyl]-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carboxamide
N-(1-{5H,6H,7H,8H-imidazo[1,5-a]pyrazine-7-carbonyl}cyclohexyl)-3,4-dimethylaniline
(3S,7S)-5-(2-methyl-1,3-thiazole-4-carbonyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
6-ethyl-N4-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-5-methylpyrimidine-2,4-diamine
N-{2-[(4-chlorophenyl)sulfanyl]ethyl}-N-(2-hydroxyethyl)-1-methyl-1H-imidazole-2-carboxamide
methyl(thiophen-2-ylmethyl)[(2,3,4-trimethoxyphenyl)methyl]amine
2-[2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-methylacetamido]-N,N-dimethylpropanamide
5-methyl-2-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
2-({3-[5-(benzylsulfanyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)phenol
3-{2-[2-(3-methylbut-2-en-1-yl)-3-oxo-2,8-diazaspiro[4.5]decan-8-yl]-2-oxoethyl}-2,3-dihydro-1λ6-thiophene-1,1-dione
2-(4-{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)-N-(propan-2-yl)acetamide
1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-N-(1,4-dioxan-2-ylmethyl)-5-(methoxymethyl)-1H-pyrazole-4-carboxamide
1-(6-{methyl[(5-methyl-1H-pyrazol-3-yl)methyl]amino}pyridin-3-yl)ethan-1-one
{[2-(azocane-1-carbonyl)-6-chloroimidazo[1,2-a]pyridin-3-yl]methyl}[1-(pyrazin-2-yl)propan-2-yl]amine
(1S,2R)-N1-[(1-hydroxycyclohexyl)methyl]-N2-(prop-2-en-1-yl)cyclohexane-1,2-dicarboxamide
2-[4-(3-cyclohexyl-1H-pyrazole-4-carbonyl)morpholin-3-yl]-N-pentylacetamide
1-[1-(2,2-dimethylpropyl)piperidin-4-yl]-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
N,N-dimethyl-4-({[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}methyl)-1,3-thiazol-2-amine
5-[(1R,3S,5S)-3-(4-fluoro-3-methylphenyl)-8-azabicyclo[3.2.1]octane-8-carbonyl]-1H-imidazole-4-carboxylic acid
3-({[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)propane-1,2-diol