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1-(4-ethoxyphenyl)-3-(oxolan-2-ylmethyl)-3-(pyridin-2-ylmethyl)urea
1-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]butane-1,2-dione
3-methoxy-N-{2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}benzamide
2-methyl-8-(piperidin-4-yl)-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
(3S,4R)-1-{2-[(2-methoxyethyl)(methyl)amino]acetyl}-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
5,5-dimethyl-3-[2-oxo-2-(3-phenylpiperazin-1-yl)ethyl]-1,3-oxazolidine-2,4-dione
5-cyclobutyl-N-(3,4-dihydro-2H-1-benzopyran-3-yl)-1,3,4-oxadiazol-2-amine
4-[3-(pyridin-4-yl)azetidine-1-carbonyl]-1,2-dihydroquinolin-2-one
(1R,3S,5S)-3-(4-methoxyphenyl)-8-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-8-azabicyclo[3.2.1]octane
(4aS,7aR)-1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-(2-methoxyphenyl)-2-methylpiperazine
N-[2-(diethylamino)-2-(furan-2-yl)ethyl]-1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-1-(morpholin-4-yl)ethan-1-one
N-ethyl-2,3,6-trimethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]quinoline-4-carboxamide
N-(3-{[(2-fluorophenyl)methyl]sulfanyl}propyl)-1-methylazepane-2-carboxamide
7-methoxy-3-[2-(4H-1,2,4-triazol-4-yl)pyridine-4-carbonyl]-2,3,4,5-tetrahydro-1H-3-benzazepine
1-{3-oxo-3-[3-(4-phenylbenzoyl)piperidin-1-yl]propyl}pyrrolidin-2-one
N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-2-methyloxolane-2-carboxamide
5-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]furan-2-carboxamide
1-{[5-chloro-1-methyl-3-(5-methyl-1,2-oxazol-3-yl)-1H-pyrazol-4-yl]methyl}-4-(1,2,4-oxadiazol-3-yl)piperidine
{3-benzyl-1-[(trimethyl-1H-pyrazol-4-yl)sulfonyl]piperidin-3-yl}methanol
{[3-(3-chlorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(2,3-dihydro-1-benzofuran-2-ylmethyl)methylamine
1-(5-{[butyl(methyl)amino]methyl}-2-methoxyphenoxy)-3-(4-methyl-1,4-diazepan-1-yl)propan-2-ol
N-({3-methyl-7-[2-(7-methyl-2-oxo-2H-chromen-4-yl)acetyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)thiophene-3-carboxamide
2-({2-[(2-methylprop-2-en-1-yl)oxy]phenyl}formamido)-N-(1,3-thiazol-2-yl)acetamide
4-ethyl-3-[1-(6-methoxypyrimidin-4-yl)piperidin-3-yl]-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
(3S,5R)-5-(cyclopropylcarbamoyl)-1-(2-phenylbenzoyl)piperidine-3-carboxylic acid
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[cyclopropyl(phenyl)methyl]-3-propyl-1H-pyrazole-5-carboxamide
N-{[3-(2-methylphenyl)phenyl]methyl}-1-(pyrimidin-2-yl)piperidin-3-amine
5-{1-[2-(methylsulfanyl)acetyl]pyrrolidin-2-yl}-N-[3-(1H-pyrazol-1-yl)propyl]thiophene-2-carboxamide
1-{2-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]propyl}-1H-imidazole
(1S,5R)-3-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[cyclohexyl(methyl)amino]-3-(3-{[methyl(quinolin-4-ylmethyl)amino]methyl}phenoxy)propan-2-ol
3-(1H-imidazol-1-ylmethyl)-1-{2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}piperidine
3-[2-(4-methylpiperazin-1-yl)ethyl]-3H,4H-thieno[3,2-d]pyrimidin-4-one
(1R,5R)-3-[3-(2-ethoxyethoxy)benzoyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonane
2-amino-6-tert-butyl-4-(2,3,4-trimethoxyphenyl)pyridine-3-carbonitrile
methyl 4-(5-methyl-4-{[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]methyl}-1,3-oxazol-2-yl)benzoate
4-({3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)-1-azatricyclo[7.3.1.05,13]trideca-3,5,7,9(13)-tetraen-2-one
N,N-dimethyl-2-[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]aniline
2,4-dimethyl-N-(4-{4-[(oxolan-3-yl)amino]piperidin-1-yl}phenyl)benzamide
N-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)-2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetamide
2-benzyl-5-(2-ethoxybenzoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine
1-{3-[(4-methoxyphenyl)amino]piperidin-1-yl}-2-(thiophen-3-yl)ethan-1-one
2-(1,4-dithiepan-6-yl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
diethyl({3-[3-(1H-pyrazol-1-yl)azetidine-1-carbonyl]pyrazolo[1,5-a]pyrimidin-6-yl}methyl)amine
N-(2-hydroxyethyl)-5-[2-(1H-imidazol-2-yl)benzoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
ethyl 3-(2-methoxyethyl)-1-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]piperidine-3-carboxylate
8-{[3-(4-chlorophenoxy)phenyl]methyl}-1-(2-methoxyethyl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione