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N-[7-oxo-5-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl]cyclobutanecarboxamide
N4-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-ethyl-N4,5-dimethylpyrimidine-2,4-diamine
N-[4-methoxy-2-(2-methylpropanamido)phenyl]-6-methyl-2-oxo-1,2-dihydropyridine-4-carboxamide
N-[2-(3-methoxyphenyl)-1-{1-[2-(phenylsulfanyl)acetyl]piperidin-4-yl}ethyl]-N,3-dimethylbutanamide
[(3R,4R)-1-(isoquinoline-5-carbonyl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
N-[3-(cyclohexylsulfanyl)propyl]-1-methyl-6-oxo-1,6-dihydropyridazine-3-carboxamide
ethyl 4-[(3-fluorophenyl)methyl]-1-(oxan-4-yl)piperidine-4-carboxylate
3-[(3-chlorophenyl)methyl]-1-(3-fluoropyridin-2-yl)piperidine-3-carboxylic acid
1-[2-({2-[(2-methylprop-2-en-1-yl)oxy]phenyl}formamido)ethyl]piperidine-3-carboxamide
N-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-(1H-1,3-benzodiazol-2-yl)propanamide
2-{[2-(1-{thieno[3,2-d]pyrimidin-4-yl}piperidin-4-yl)-1H-imidazol-1-yl]methyl}pyridine
methyl 3-({imidazo[1,2-a]pyridin-2-ylformamido}methyl)-5-[2-(thiophen-3-yl)acetamido]benzoate
2-[4-(2-amino-6-methylpyridin-3-yl)-1H-pyrazol-1-yl]-N-[1-(propan-2-yl)-1H-1,2,3-triazol-4-yl]acetamide
5-methanesulfonamido-N-methyl-1-(2-phenylethyl)-N-(thiophen-3-ylmethyl)-1H-1,3-benzodiazole-7-carboxamide
1-ethyl-3-methyl-8-{[4-(pyrimidin-2-yloxy)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[3-(2-methoxyphenoxy)azetidin-1-yl]-2-[methyl(phenyl)amino]ethan-1-one
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-oxo-1-oxaspiro[4.4]nonane-4-carboxamide
[(2S,4R)-4-(dimethylamino)-1-{[3-(trifluoromethyl)phenyl]methyl}pyrrolidin-2-yl]methanol
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)naphthalene-1-carboxamide
(2S)-N-[2-(2-chloro-6-methylphenoxy)ethyl]-1-(piperidin-4-yl)pyrrolidine-2-carboxamide
1-tert-butyl-N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
1-(4-methoxybenzoyl)-4-(2,4,5-trimethylbenzoyl)piperazine
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-(2-hydroxyphenyl)acetamide
2,2-dimethylpropyl 9-oxo-8-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecane-2-carboxylate
1-(4-cyclohexylpiperazin-1-yl)-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}ethan-1-one
5-[2-(1-phenylethyl)-1H-imidazol-1-yl]pyridine-3-carboxylic acid
N-[2-hydroxy-3-(3-methoxyphenoxy)propyl]-2-(pyrrolidin-1-yl)-5,6,7,8-tetrahydroquinazoline-4-carboxamide
1-[4-({3-[1-(pyrimidin-2-yl)piperidin-4-yl]pyrrolidin-1-yl}methyl)thiophen-2-yl]ethan-1-one
4-{1-[2-(2,4-dimethoxyphenyl)acetyl]piperidin-3-yl}benzoic acid
N-({7-[(2E)-3-(4-methoxyphenyl)prop-2-enoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)thiophene-2-sulfonamide
(3aR,6aR)-2-(1H-indol-7-ylmethyl)-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[2-(2,4-dichlorophenyl)ethyl]-5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carboxamide
3-(1-ethyl-1H-imidazol-2-yl)-1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]piperidine
3-benzyl-4-(4-chloro-1,5-dimethyl-1H-pyrazole-3-carbonyl)piperazin-2-one
N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)-3-(2-oxopyrrolidin-1-yl)propanamide
1-(2,1,3-benzothiadiazol-4-yl)-3-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]urea
1-methyl-4-{1-[3-(2-methylphenyl)phenyl]piperidin-4-yl}-1,4-diazepane
(4-{[1-(2,1,3-benzoxadiazol-4-ylmethyl)pyrrolidin-3-yl]methyl}phenyl)methanol
1-[(3-fluorophenyl)methyl]-4-(1-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carbonyl)piperazine
1-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-3-(5-methyl-2,1,3-benzothiadiazol-4-yl)urea
1-ethyl-N-(furan-3-ylmethyl)-N-methyl-5-(piperidin-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-[5-(2-chloro-4-methoxyphenoxymethyl)-1,2-oxazole-3-carbonyl]azepane
2-(3-{[4-(4-ethyl-1-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}phenoxy)acetamide
ethyl 1-(3-ethyl-1-methyl-1H-pyrazole-5-carbonyl)-3-[(2-fluorophenyl)methyl]piperidine-3-carboxylate
2-(methoxymethyl)-1-({2-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)piperidine
N,N-dimethyl-1-(1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}piperidine-4-carbonyl)pyrrolidin-3-amine
ethyl[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)amine
5-methyl-5-(4-methylpent-3-en-1-yl)-1-[2-(1H-pyrazol-4-yl)ethyl]piperidin-2-one
N-(1-methoxybutan-2-yl)-3-{[(3-methylthiophen-2-yl)methyl]amino}benzamide
5-[3-(3-methylphenoxy)azetidine-1-carbonyl]-N-phenylpyrimidin-2-amine