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(3S,4R)-4-(2-methoxyphenyl)-1-[(2-methyl-1,3-thiazol-4-yl)methyl]pyrrolidine-3-carboxylic acid
2-(6-methoxynaphthalen-2-yl)-4-{[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}morpholine
1-[(5-methylfuran-2-yl)methyl]-4-(2-methylpyridin-4-yl)-1,4-diazepane
7-{6-[(piperidin-4-yl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-3,4-dihydro-2H-1-benzopyran-4-one
2-(2,5-dioxoimidazolidin-1-yl)-N-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]acetamide
3-[4-(4-tert-butyl-1H-1,2,3-triazol-1-yl)piperidine-1-carbonyl]-2,6-dimethoxypyridine
2-{4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-fluoropyridine
8-(2-methyl-6-oxo-1,6-dihydropyrimidine-5-carbonyl)-2-(3-methylbut-2-en-1-yl)-2,8-diazaspiro[4.5]decan-3-one
2-[5-(2-cyclopropyl-4-methylpyrimidin-5-yl)-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-1-yl]acetic acid
5-(4-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}phenyl)-2-methyl-2H-1,2,3,4-tetrazole
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
2-(3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}pyrrolidin-1-yl)-4-methyl-6-(2-methylpropyl)pyrimidine
N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
1-(2-methoxyphenyl)-4-[1-(prop-2-ene-1-sulfonyl)piperidin-3-yl]piperazine
1-[4-(1-hydroxy-3-phenylpropyl)piperidin-1-yl]-2-{imidazo[1,2-a]pyridin-3-yl}ethan-1-one
(1S,5S)-3-[(4-methoxy-2,3-dimethylphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
2-(4-methyl-1,4-diazepan-1-yl)-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}acetamide
N-benzyl-2-{[(1H-imidazol-2-ylmethyl)amino]methyl}-N-methyl-2,3-dihydro-1H-inden-2-amine
2-[(4-methoxyphenyl)methyl]-N-[2-(6-methylpyridin-2-yl)ethyl]-1,3-benzoxazole-6-carboxamide
N,N-dimethyl-2-{[2-(methylamino)-2-phenylacetamido]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
1-(4-methoxyphenyl)-2,2-dimethyl-4-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperazine
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-1-{4-[hydroxy(1-methyl-1H-imidazol-2-yl)methyl]piperidin-1-yl}ethan-1-one
3-(2-{5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}ethyl)-2,3-dihydro-1,3-benzoxazol-2-one
N-{[3-(oxolan-3-yloxy)phenyl]methyl}-2-(piperidin-1-yl)-N-(pyridin-4-ylmethyl)acetamide
1-{[1-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)piperidin-3-yl]methyl}-3-ethylurea
N,N-dimethyl-3-{[2-(2,4,7-trimethyl-1H-indol-3-yl)acetamido]methyl}benzamide
4-methyl-N-{3-[3-(1,2-oxazolidin-2-yl)propanamido]phenyl}benzamide
1-(4-{[3-(6-methoxynaphthalene-2-carbonyl)piperidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
7-fluoro-2-(1-methyl-1H-pyrazol-4-yl)-N-(propan-2-yl)-N-(pyridin-3-ylmethyl)quinoline-4-carboxamide
2-amino-6-(2H-1,3-benzodioxol-5-yl)-4-(1,3-dimethyl-1H-pyrazol-4-yl)-5-methylpyridine-3-carbonitrile
1-[(dimethyl-1,3-thiazol-2-yl)methyl]-4-phenyl-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
6-ethyl-1,5-dimethyl-3-{6-oxo-1H,2H,3H,4H,6H,10bH-pyrimido[2,1-a]isoindole-1-carbonyl}-1,2-dihydropyridin-2-one
1-[2-({4-ethyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)-4-methylphenyl]-1H-pyrazole
(3aR,5R,6S,7aS)-2-(3-chlorobenzoyl)-octahydro-1H-isoindole-5,6-diol
8-(9H-fluoren-2-ylmethyl)-1-methoxy-1,8-diazaspiro[4.5]decan-2-one
1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-3-(morpholin-4-yl)propan-1-one
(3aS,6aS)-2-(2-hydroxyethyl)-5-{[4-(5-methylfuran-2-yl)phenyl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
6-(2-aminoethyl)-N,2-dimethyl-N-(1-methylpyrrolidin-3-yl)pyrimidin-4-amine
3-cyclopropyl-5-[(2-phenyl-1H-imidazol-1-yl)methyl]-1,2,4-oxadiazole
1,2-dimethyl-3-{4-[(3-methylpyridin-2-yl)methyl]piperazine-1-carbonyl}-1H-indol-5-ol
4-{4-[4-(azepan-1-ylmethyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}butan-2-ol
1-{1-[(2-chloro-6-fluoro-3-methoxyphenyl)methyl]piperidin-4-yl}piperidin-4-ol
2-(methylamino)-N-[1-(pyrazin-2-yl)piperidin-3-yl]-1,3-thiazole-4-carboxamide
N-(2-methoxyethyl)-N-(pyridin-2-ylmethyl)quinoxaline-6-carboxamide
1-{7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
[(5-tert-butyl-1H-pyrazol-3-yl)methyl](ethyl){[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}amine
N-[2-(dimethylamino)ethyl]-N-methyl-1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carboxamide
2-(2,6-dimethoxypyridin-3-yl)-2-[4-(hydroxymethyl)piperidin-1-yl]acetic acid
1-methyl-1-[2-(pyridin-2-yl)ethyl]-3-(2,4,6-trimethylpyridin-3-yl)urea
4-[(3-methylpyridin-2-yl)methyl]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol