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4-[3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propanoyl]-1λ6-thiomorpholine-1,1-dione
N-[2-(2-fluorophenoxy)ethyl]-2-oxo-2-(pyrrolidin-1-yl)acetamide
N-[(3,4-difluorophenyl)methyl]-5-(methoxymethyl)-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-4-(pyrrolidine-1-sulfonyl)piperazine
2-{1-[(3,5-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(3-fluoro-4-methylphenyl)methyl]acetamide
2-amino-1-(3-{5-[(4-hydroxypiperidin-1-yl)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)ethan-1-one
4-(4-cyclobutyl-6-methylpyrimidin-2-yl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
ethyl 3-[(2-methylphenyl)methyl]-1-(pyridine-2-carbonyl)piperidine-3-carboxylate
N-methyl-2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-(pyridin-3-ylmethyl)acetamide
N5-butyl-1-(furan-2-ylmethyl)-N3-methyl-4-oxo-N3-(2-phenylethyl)-1,4-dihydropyridine-3,5-dicarboxamide
8-{[5-(hydroxymethyl)furan-2-yl]methyl}-1-(2-phenylethyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(5-amino-1H-1,2,4-triazol-3-yl)-N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]propanamide
3-(3-fluorophenyl)-4-[3-(propoxymethyl)pyrrolidine-1-carbonyl]-1H-pyrazole
N5-cyclohexyl-1-cyclopropyl-N3-methyl-4-oxo-N3-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide
methyl[(2-methyl-1H-imidazol-4-yl)methyl][4-(morpholin-4-yl)butyl]amine
2-(dimethyl-1,2-oxazol-4-yl)-N-(3-methoxypropyl)-N-(1-methylpiperidin-4-yl)acetamide
(5S,9aS,9bS)-2-[(2-methylphenyl)methyl]-5-(3-methylthiophen-2-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-[2-(4-fluorophenyl)ethyl]piperidine-4-carboxamide
(4aR,7aS)-1-[(5-ethylpyridin-2-yl)methyl]-4-(3-methylbut-2-enoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(4-methyl-1,3-thiazol-5-yl)-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]propanamide
4-{2-[1-(1H-imidazol-4-ylmethyl)piperidin-2-yl]ethyl}morpholine
1-[2-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-2-oxoethyl]-1,2-dihydropyridin-2-one
1-{2-[(3-fluorophenyl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-(1-hydroxy-2-methylpropan-2-yl)piperidine-3-carboxamide
(2E)-3-(4-methoxyphenyl)-N-({4-methyl-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)prop-2-enamide
3-[(4-methoxyphenyl)methyl]-1-(3-methoxypropyl)-8-(oxan-4-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-({8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}methyl)-2-phenylpyrimidine
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-6-methoxy-2,3-dihydro-1H-indene-5-carboxamide
1-{3-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-3-oxopropyl}piperidin-2-one
3-(4-chloro-1H-pyrazol-1-yl)-1-{2-[2-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}propan-1-one
{[2-(azocane-1-carbonyl)-6-chloroimidazo[1,2-a]pyridin-3-yl]methyl}[2-(1,3-thiazol-4-yl)ethyl]amine
4-[(3-fluorophenyl)methyl]-1-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]-1,4-diazepan-5-one
4-(hydroxymethyl)-1-(pyridine-2-carbonyl)azepan-4-ol
2-{3-[3-(5-acetylpyridin-2-yl)phenyl]-1H-pyrazol-1-yl}-1-(piperidin-1-yl)ethan-1-one
1-{4-methyl-2-[4-(morpholine-4-carbonyl)piperazin-1-yl]pyrimidin-5-yl}ethan-1-one
2-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-N-(3-methoxypropyl)-1,3-oxazole-4-carboxamide
2-[(4-chlorophenyl)methyl]-N-[(3R,4R)-3-hydroxypiperidin-4-yl]benzamide
N-[2-(3-methoxyphenyl)ethyl]-5-[3-(trifluoromethyl)phenyl]-1,2,4-triazin-3-amine
3,5-dimethyl-1-(3-{1-[(2S)-oxolan-2-ylmethyl]-1H-imidazol-2-yl}phenyl)-1H-pyrazole
N-[(6-chloropyridin-3-yl)methyl]-N-methyl-3-(1H-pyrazol-1-ylmethyl)benzamide
(2R,6R)-4-[(6-methylpyridin-2-yl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-hydroxy-3-methylbutan-1-one
(4aR,7aS)-1-cyclobutanecarbonyl-4-(1,3-thiazol-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(3R,4S)-1-(3-methoxypropyl)-4-propylpyrrolidin-3-yl]-6-oxo-1,6-dihydropyrimidine-5-carboxamide
4-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-6-(piperidin-1-yl)pyrimidine
(2E)-3-(4-methoxyphenyl)-N-{[4-(2-methylpropyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}prop-2-enamide
N-(3-fluoro-4-methylphenyl)-7-methyl-12-oxo-3,7,11-triazaspiro[5.6]dodecane-3-carboxamide
3-fluoro-N-[(7-{[3-(2-methylphenyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]benzamide
1-[2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)acetyl]-4-[(3-fluorophenyl)methyl]-1,4-diazepan-5-one
3-(oxolan-3-ylmethyl)-1-(4-pentylphenyl)urea
[(2S)-1-[5-(3-fluorophenoxymethyl)-1H-pyrazole-3-carbonyl]pyrrolidin-2-yl]methanol