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4-(3-phenyl-1,2,4-oxadiazol-5-yl)-2-(trifluoromethyl)morpholine
N-({4-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)cyclohexanecarboxamide
2-[2-(4-methylpentyl)morpholin-4-yl]pyridine-3-carboxamide
N-[(1S,2R)-2-aminocyclobutyl]-5-methoxy-1H-indole-2-carboxamide
3-hydroxy-1-[(3-methoxyphenyl)methyl]-3-{[(3-methylpentan-3-yl)amino]methyl}piperidin-2-one
3-methyl-5-(2-methyl-2,3-dihydro-1-benzofuran-5-yl)-1H-1,2,4-triazole
5-(phenoxymethyl)-N-[3-(1H-pyrazol-1-yl)propyl]-1,2-oxazole-3-carboxamide
6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]-N-(pyridin-4-ylmethyl)piperidine-3-carboxamide
1-(4-{[(1S,5R)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}thiophen-2-yl)ethan-1-one
(3S,4S)-1-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)-4-(pyrrolidin-1-yl)pyrrolidin-3-ol
5-(1-{[4-(dimethylamino)phenyl]methyl}piperidin-4-yl)-5-methylimidazolidine-2,4-dione
8-(3-phenylbutyl)-5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine
2-(2-{4-[(dimethylamino)methyl]phenyl}piperidine-1-carbonyl)-N,N-dimethylaniline
6-[2-(2-methyl-1H-indol-3-yl)acetyl]-N-[3-(pyridin-4-yl)propyl]-6-azaspiro[2.5]octane-1-carboxamide
1-{3-[2-(2-methylphenyl)ethyl]piperidin-1-yl}-2-(1H-pyrazol-1-yl)ethan-1-one
7-(cyclobutylmethyl)-2-(3-phenoxypropanoyl)-2,7-diazaspiro[4.5]decan-6-one
N-(2-hydroxy-2-phenylethyl)-N-methyl-3-(5-{[3-(trifluoromethyl)phenyl]methyl}-1,3,4-oxadiazol-2-yl)propanamide
N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,6-dimethoxypyridine-3-carboxamide
3-(4-methoxy-4-phenylpiperidine-1-carbonyl)-N,N-dimethylpiperidine-1-carboxamide
5-{3-chloro-6-methylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
(4aS,7aR)-1-(furan-2-carbonyl)-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(pyridin-2-ylmethyl)-8-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-2,8-diazaspiro[5.5]undecan-3-one
N-[(2,4-dihydroxyphenyl)methyl]-5-(2-fluorophenoxymethyl)-1H-pyrazole-3-carboxamide
(4aS,7aR)-1-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-methyl-8-[(2-phenyl-1,3-thiazol-4-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
5-chloro-3-methyl-N-{[4-(oxolan-2-ylmethoxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)-1H-indole-2-carboxamide
1-[4-(dimethylamino)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-(1H-imidazol-1-yl)propan-1-one
N-[(3R,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-methoxybenzamide
1-{[3-(cyclopentyloxy)phenyl]methyl}-N-[2-(dimethylamino)ethyl]-N-methylpiperidin-3-amine
(2S)-N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-5-oxopyrrolidine-2-carboxamide
8-[(2S,3R)-2-amino-3-hydroxybutanoyl]-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-[4-(4-methyl-1H-pyrazol-1-yl)phenyl]phenol
2-[1,3-dimethyl-4-(2-methylpyrrolidin-1-yl)-1H-pyrazolo[3,4-d]pyrimidin-6-yl]pyridine
N,N-dimethyl-2-[1-(3-methylpentanoyl)-3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-4'-yl]acetamide
3-methoxy-2-({[2-(4-methoxyphenyl)ethyl][(1-methylpiperidin-4-yl)methyl]amino}methyl)phenol
2-{4-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-1,4-diazepan-1-yl}-4,6,7-trimethylquinazoline
N-[(1,2-dimethyl-1H-1,3-benzodiazol-5-yl)methyl]-1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
N-methyl-2-[1-methyl-2,5-dioxo-3-(4-phenylphenyl)pyrrolidin-3-yl]-N-[2-(1H-pyrazol-4-yl)ethyl]acetamide
2-{4-[(2,6-difluorophenyl)methyl]-1-(2,2-dimethylpropyl)piperazin-2-yl}ethan-1-ol
4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]-1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]piperidine
ethyl 1-[(4-methoxyphenyl)methyl]-5-(5-methyl-1H-pyrazole-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-[(3R,4R)-3-hydroxy-1-[(1-methyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]piperidin-4-yl]pyridine-4-carboxamide
8-{[3-hydroxy-1-(2-methoxyethyl)-2-oxopiperidin-3-yl]methyl}-2-methyl-1,3,8-triazaspiro[4.5]dec-1-en-4-one
1-[(4-fluoro-3-methoxyphenyl)methyl]-4-(2-methylpropyl)-1,4-diazepan-5-one
N-[1-(2-{8-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-2-oxoethyl)-1H-pyrazol-4-yl]-3-(2-methoxyphenyl)propanamide
(1S,5R)-6-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
8-[(4-methoxyphenyl)methyl]-1-(2-phenylethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(7-methoxy-4-methylquinolin-2-yl)butan-2-ol
N-[(3S,5S)-5-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1-(naphthalen-2-ylmethyl)pyrrolidin-3-yl]-1-propylpiperidin-4-amine
1-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-(pyridin-4-yl)ethan-1-one