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3-benzyl-5-(cyclopentylmethyl)-1H-1,2,4-triazole
5-{[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]methyl}-N,N-dimethylpyrimidin-2-amine
N-[(4-hydroxy-3-methoxyphenyl)methyl]-8-methyl-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
7-fluoro-N,3-dimethyl-N-[1-(1,3-thiazol-2-yl)ethyl]-1-benzofuran-2-carboxamide
7-{[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]methyl}-2-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one
7-(cyclopropylmethyl)-2-{2-[4-(dimethylamino)phenyl]acetyl}-2,7-diazaspiro[4.5]decan-6-one
2-(1-cyclopentyl-4-methylpiperazin-2-yl)ethan-1-ol
1-(1,3-benzothiazol-2-yl)-N-(thiophen-3-ylmethyl)piperidin-4-amine
(3R,4R)-1-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-4-(morpholin-4-yl)piperidin-3-ol
1-[7-(1-benzothiophen-3-yl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-cyclopentylethan-1-one
[1-(3-ethyl-1,2-oxazol-5-yl)ethyl]({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl})amine
1-[(2-methylphenyl)methyl]-5-[2-(trimethyl-1H-pyrazol-4-yl)ethyl]-1H-1,2,4-triazole
4-[6-(propan-2-yl)-2-(trifluoromethyl)pyrimidin-4-yl]benzamide
2-[(4aR,7aS)-4-[(3-methylphenyl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
1-[3-(2-chlorophenyl)pyrrolidin-1-yl]-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propan-1-one
methyl (2S,4R)-1-[(2,3-dimethoxyphenyl)methyl]-4-(naphthalene-1-amido)pyrrolidine-2-carboxylate
6-[2-(3-methoxyphenyl)azetidine-1-carbonyl]-2-methyl-1,3-benzoxazole
N-(3-methoxypropyl)-N-{[2-(3-methylphenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}furan-2-carboxamide
2-propyl-4-[2-(trifluoromethyl)pyrrolidine-1-carbonyl]-1,3-thiazole
4-(3-chloro-4-hydroxybenzoyl)-5-methyl-1-(4-methylphenyl)piperazin-2-one
{[4-(pyrrolidine-1-carbonyl)phenyl]methyl}[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]amine
1'-[(1,5-dimethyl-1H-indol-2-yl)methyl]-5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[(2R,3R)-1'-[2-(5-acetylthiophen-3-yl)acetyl]-2-(prop-2-en-1-yloxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methoxyacetamide
3-[(5,8-dimethoxy-4-methylquinolin-2-yl)amino]-1λ6-thiolane-1,1-dione
N-{[4-(4-fluorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}pent-4-enamide
2-[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-5-methylphenol
2-[(3-methoxyphenyl)methyl]-4-(prop-2-ene-1-sulfonyl)morpholine
2-(2,4-dioxoimidazolidin-1-yl)-N-[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]acetamide
3-(5-cyclohexyl-1,3,4-oxadiazol-2-yl)-N-methyl-N-[4-(morpholin-4-yl)butyl]propanamide
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-1-(pyridin-2-yl)piperidine-3-carboxamide
5-[1-(3-phenylbutyl)piperidin-4-yl]-5-(3-phenylpropyl)imidazolidine-2,4-dione
4-benzyl-3-{2-[4-(2-methoxyethoxy)piperidin-1-yl]-2-oxoethyl}piperazin-2-one
5-(2,6-difluoro-3-methylbenzoyl)-2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
(1R,7S)-3-[(3-methoxyphenyl)methyl]-6-[4-(prop-2-en-1-yl)piperazine-1-carbonyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
2-[4-(furan-2-ylmethyl)-1-(propan-2-yl)piperazin-2-yl]ethan-1-ol
1-(4-phenyl-1,4-diazepan-1-yl)-3-[5-(thiophen-3-yl)-1,3,4-oxadiazol-2-yl]propan-1-one
3-({[(4-fluorophenyl)methyl]amino}methyl)-3-hydroxy-1-(2-phenylethyl)piperidin-2-one
N4-(6-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)-6-methylpyrimidine-2,4-diamine
N-{[5-fluoro-7-(4-fluoro-3-methylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
2-(1-methyl-1H-pyrrol-3-yl)-1-[1-(pyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]ethan-1-one
3-benzyl-5-[3-(3-fluorophenyl)-1H-pyrazol-4-yl]-1H-1,2,4-triazole
3-[1-(1H-indazol-6-yl)-1H-imidazol-2-yl]benzonitrile
[1-(4-aminopyrimidin-2-yl)-3-(cyclopropylmethyl)piperidin-3-yl]methanol
(1-{[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}piperidin-4-yl)methanol
2-(2-methoxyethyl)-8-{[5-(4-methylphenyl)furan-2-yl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
3-(piperidine-1-carbonyl)-1-propyl-N-(pyridin-4-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(3S,4R)-1-(2,6-difluoro-4-methoxybenzoyl)-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
2-ethoxy-N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]pyridine-3-carboxamide
N-[(2,6-difluorophenyl)methyl]-1-methyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-amino-6-(2-methylphenyl)-4-(piperidin-4-yl)pyridine-3-carbonitrile