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5-chloro-N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}thiophene-2-carboxamide
2-[4-(4-ethylpiperazine-1-carbonyl)-5-methyl-1H-pyrazol-1-yl]-4-(thiophen-2-yl)pyrimidine
N-ethyl-N-methyl-2-[5-oxo-4-phenyl-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]acetamide
2-(3-methoxypropyl)-9-{[1,2,4]triazolo[1,5-a]pyrimidin-2-ylmethyl}-2,9-diazaspiro[5.5]undecan-3-one
3-[(3S,4S)-4-methoxy-1-(propan-2-yl)pyrrolidin-3-yl]-1-(2-methyl-1-benzofuran-5-yl)urea
N-(2,2-difluoroethyl)-4-methoxy-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzamide
3-({4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}methyl)-5-methoxy-1H-indazole
(2S,4S)-N-(2-methoxyethyl)-1-(1-propylpiperidin-4-yl)-4-({[4-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
2-(2-methyl-1,3-thiazol-4-yl)-5-[4-(pyridin-2-yl)piperazine-1-carbonyl]pyrimidin-4-ol
5-{4-[(4-hydroxy-6-methylquinolin-2-yl)methyl]piperazin-1-yl}-2-methyl-2,3-dihydropyridazin-3-one
3-{[(butan-2-yl)(pyridin-3-ylmethyl)amino]methyl}benzonitrile
[(3R,4R)-1-(2-methoxy-5-methylbenzoyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
N-[(2R,3R)-2-(benzyloxy)-1'-[(2E)-3-(thiophen-2-yl)prop-2-enoyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
1-(3-fluorobenzoyl)-4-[4-(2-phenylethyl)-1H-pyrazol-5-yl]piperidine
{1-[(1-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl)methyl]-1H-1,2,3-triazol-4-yl}methanol
N-[4-(1H-1,3-benzodiazol-2-yl)phenyl]-1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)piperidine-4-carboxamide
N-methyl-5-(morpholin-4-ylmethyl)-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)furan-3-carboxamide
ethyl 4-{1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]piperidin-3-yl}piperazine-1-carboxylate
methyl 3-(furan-3-amido)-5-{[(3-hydroxy-4-methoxyphenyl)methyl]amino}-1-(2-methylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-(naphthalen-1-ylmethyl)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-[1-(piperidin-1-yl)cyclohexanecarbonyl]-3-(1H-pyrazol-5-yl)piperidine
1-(1-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}-4-phenylpiperidin-4-yl)ethan-1-one
[(3-chloro-4-methoxyphenyl)methyl][2-(1H-imidazol-1-yl)ethyl]methylamine
2-(4-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-1-(thiophen-2-ylmethyl)piperazin-2-yl)ethan-1-ol
2-methyl-5-(1H-pyrazol-1-yl)-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}benzene-1-sulfonamide
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-(pyridin-2-ylmethyl)piperidine-4-carboxamide
N-[3-(benzyloxy)phenyl]-3-acetamidopyrrolidine-1-carboxamide
1-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]-2-(pyridin-4-yl)ethan-1-one
2-cyclopentyl-9-[(3,5-dimethoxyphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
(2S)-1-[9-methoxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
2-[4-({2-[(4-chlorophenyl)methoxy]phenyl}methyl)morpholin-2-yl]ethan-1-amine
5-({2-[2-(2-ethoxyphenyl)-1H-imidazol-1-yl]ethyl}sulfanyl)-1-methyl-1H-1,2,3,4-tetrazole
(5S,9aS,9bS)-5-(1,5-dimethyl-1H-pyrazol-4-yl)-2-phenyl-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
5-butyl-1'-(5-methoxyfuran-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[2-(azepan-1-yl)ethyl]-6-methyl-2-oxo-N-(propan-2-yl)-1,2-dihydropyridine-4-carboxamide
1-{1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}-4-[3-(trifluoromethyl)phenyl]piperazine
1-(2-{1-[2-(1H-imidazol-5-yl)ethyl]-3-phenyl-1H-1,2,4-triazol-5-yl}ethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
methyl 3-(2-chlorobenzamido)-6-(piperidin-1-ylmethyl)thieno[2,3-b]pyridine-2-carboxylate
methyl (2S,4R)-4-(6-chloro-2-oxo-2H-chromene-3-amido)-1-methylpyrrolidine-2-carboxylate
1-(4-methoxyphenyl)-6,6-dimethyl-4-(2-methylpyridine-3-carbonyl)piperazin-2-one
N-[(3S,4R)-1-[(1-ethyl-1H-indol-4-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
1-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]-2-[methyl(pyridin-2-ylmethyl)amino]ethan-1-one
(1S,6R)-3-{[3-(2,6-dichlorophenyl)-5-methyl-1,2-oxazol-4-yl]methyl}-3,9-diazabicyclo[4.2.1]nonan-4-one
3-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)-N-[2-(1,3-thiazol-4-yl)ethyl]propanamide
4-[({3-azaspiro[5.5]undecan-9-yl}(methyl)amino)methyl]-1-cyclopentylpyrrolidin-2-one
5-[({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)carbamoyl]-2,1,3-benzoxadiazol-1-ium-1-olate
N-[1-(furan-2-ylmethyl)-1H-pyrazol-5-yl]-2-[4-(quinolin-8-yl)-1H-pyrazol-1-yl]acetamide
(3R,4R)-4-ethyl-1-[4-(3-fluorophenyl)benzoyl]piperidine-3,4-diol
2-[(1-ethyl-2-oxo-1,2-dihydropyridin-4-yl)formamido]hexanamide
N-cyclohexyl-3-(4-methylpiperazine-1-carbonyl)-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-amine