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3-fluoro-4-[3-(piperidin-1-ylmethyl)piperidin-1-yl]pyridine
1-{3-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}-2-propoxyethan-1-one
N-[3-(4-fluorophenyl)phenyl]-1-[2-(1H-pyrazol-4-yl)ethyl]piperidine-3-carboxamide
3-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-carbonyl}-5-phenyl-1,2-oxazole
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)-2-(2-oxopiperidin-1-yl)acetamide
N-[2-(7-{[5-(4-chlorophenyl)furan-2-yl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]oxolane-2-carboxamide
1-(1H-imidazol-2-ylmethyl)-4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
N-[(4-phenyloxan-4-yl)methyl]-2-(pyrrolidin-1-yl)-5,6,7,8-tetrahydroquinazoline-4-carboxamide
5-(1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1H-1,2,3-triazol-4-yl)-N,N-dimethylpyrimidin-2-amine
N-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}-N-(pyridin-3-ylmethyl)cyclopropanamine
1,9-dimethyl-4-(pyridine-3-sulfonyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
2-phenoxy-N-(4-{4-[(thiophen-3-ylmethyl)amino]piperidin-1-yl}phenyl)acetamide
4-(2H-1,3-benzodioxol-5-ylmethyl)-1-[(2-methyl-1,3-thiazol-4-yl)methyl]-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
9-[(5-fluoro-3-methyl-1H-indol-2-yl)methyl]-6-oxa-9-azaspiro[4.5]decane
6-cyclopropyl-N-{[1-(2-phenylethyl)piperidin-3-yl]methyl}pyrimidin-4-amine
4-(piperidin-1-yl)-N-[2-(pyrazin-2-yl)ethyl]butanamide
1-[3-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-1-yl]-3-(pyridin-3-yl)propan-1-one
N-(5-methyl-1,2-oxazol-3-yl)-2-oxo-2-[(2R,6S)-6-phenyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]acetamide
1-{2-[(2,3-dimethoxyphenyl)formamido]ethyl}-N-phenyl-1H-1,2,3-triazole-4-carboxamide
methyl 4-{[(2-{5-oxo-1-[(4-phenyloxan-4-yl)methyl]pyrrolidin-2-yl}ethyl)amino]methyl}benzoate
1-[2-({6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)ethyl]pyrrolidin-2-one
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-2-methyl-1,3-benzothiazole-6-carboxamide
N-{[7-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-1,3-thiazole-5-carboxamide
1-(4-{2-[(3-methoxyphenyl)methyl]morpholin-4-yl}piperidin-1-yl)ethan-1-one
2-(1-{[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}piperidin-4-yl)-1H-1,3-benzodiazole
5-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-4-methyl-1,2,3-thiadiazole
[(3R,4R)-1-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
1-{1'-[2-(2-methyl-1H-imidazol-1-yl)acetyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
methyl 2-(cyclopentylsulfamoyl)-6-[(4-methoxy-2,3-dimethylphenyl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
ethyl 4-{[4-(pyridine-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperazine-1-carboxylate
(2-{4-[(4-methylphenyl)sulfanyl]piperidin-1-yl}-1,3-thiazol-4-yl)methanol
4-[(1-butanoylpiperidin-4-yl)amino]-1-propylpyrrolidin-2-one
[(2S)-1-({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)pyrrolidin-2-yl]methanol
[1-(2,4-dimethoxyphenyl)ethyl](methyl){[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amine
1-methyl-8-(2-methylpyrimidin-4-yl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-ethyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)pyridine-3-carboxamide
2-{1-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]pyrrolidin-2-yl}pyridine
N-[(3R,4S)-1-(oxan-4-yl)-4-propylpyrrolidin-3-yl]-3-(pyrazin-2-yl)propanamide
N-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-pyrrolo[2,3-b]pyridin-6-amine
6-{3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}pyrazine-2-carboxamide
7-(cyclopropylmethyl)-2-[2-(methylamino)pyridine-4-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
(3aS,6aS)-2-[(3-methyl-1H-1,2,4-triazol-5-yl)methyl]-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-(3-hydroxy-3-methylbutyl)-N-{[5-(thiophen-2-yl)-1,2,4-oxadiazol-3-yl]methyl}benzamide
N-cyclobutyl-2-(3-methoxyphenoxymethyl)-1,3-oxazole-4-carboxamide
2-{[4-(2-chlorophenyl)-5-(1,5-dimethyl-1H-pyrazol-3-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
3-(1-cyclopentyl-4-methyl-1H-pyrazol-5-yl)-1-cyclopropyl-1-(1H-indol-5-ylmethyl)urea
4-[(2-methyl-4-phenylpiperazin-1-yl)methyl]benzonitrile
4-chloro-N-[(3-fluorophenyl)methyl]-N-(1-methoxypropan-2-yl)-1H-pyrrole-2-carboxamide
5-(2-{[(2-fluorophenyl)methyl]amino}ethyl)-1-{[4-(trifluoromethoxy)phenyl]methyl}pyrrolidin-2-one
methyl({[4-methyl-5-(piperidin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl})[1-(1,3-thiazol-2-yl)ethyl]amine