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5-{1-[(2E)-4-methylpent-2-enoyl]piperidin-4-yl}-5-(pyridin-3-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
6-[2-(hydroxymethyl)phenyl]pyridine-3-carboxamide
1'-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-[1-(propan-2-yl)piperidine-4-carbonyl]-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
(1S,6R)-9-{[1,2,4]triazolo[4,3-a]pyridine-7-carbonyl}-3,9-diazabicyclo[4.2.1]nonane
N-({1-[(4-methylpiperazin-1-yl)methyl]cyclopropyl}methyl)-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
4-(2-hydroxy-5-methoxyphenyl)-1-methyl-3-phenyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-[1-(4-methylphenyl)ethyl]-2-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]acetamide
5-(2-methoxyphenoxymethyl)-N-(pentan-2-yl)-1H-pyrazole-3-carboxamide
8-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-1-(2-phenylethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-(cyclopropylmethyl)-1-(5-methoxy-4-oxo-1,4-dihydropyridine-2-carbonyl)-3-(propan-2-yl)-1,4-diazepan-5-one
5-{2-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carbonyl}-2-(pyridin-2-yl)pyrimidin-4-ol
3-propyl-5-{[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}imidazolidine-2,4-dione
N-benzyl-4-hydroxy-2-methyl-N-[(4-methyl-1,3-thiazol-5-yl)methyl]pyrimidine-5-carboxamide
8-(6-methylpyrimidin-4-yl)-3-{3-[4-(propan-2-yl)piperazin-1-yl]propyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(1-benzyl-3-oxopiperazin-2-yl)-N-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]acetamide
N-(2,4-dimethoxyphenyl)-3-[1-(oxolane-2-carbonyl)piperidin-4-yl]propanamide
1-(4-methoxyphenyl)-4-[4-(morpholin-4-ylmethyl)piperidin-1-yl]butane-1,4-dione
4-[(1S,5R)-6-(cyclobutylmethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]benzene-1-sulfonamide
5-{1-[(2-fluorophenyl)methyl]-1H-pyrazol-3-yl}-N-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-methyl-1,3-thiazol-2-amine
N-(adamantan-2-ylmethyl)-3-(6-oxo-1,6-dihydropyridazin-3-yl)propanamide
N-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)-3-phenyl-1H-pyrazole-4-carboxamide
3-methoxy-N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}propanamide
3-[4-({[(dimethyl-1,2-oxazol-4-yl)methyl](methyl)amino}methyl)-1H-pyrazol-1-yl]propanoic acid
N-[(2-phenoxypyridin-3-yl)methyl]-4-sulfamoylbenzamide
2-{1-[3-(dimethyl-1,3-thiazol-2-yl)propyl]-1H-imidazol-2-yl}benzoic acid
[(3R,4R)-4-(azepan-1-ylmethyl)-1-(3-ethyl-1H-pyrazole-4-carbonyl)pyrrolidin-3-yl]methanol
4-[(2R,3S,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]butanoic acid
5-(2,6-difluorophenoxymethyl)-N-(2-hydroxy-3-methoxypropyl)-1,2-oxazole-3-carboxamide
(5S,9aS,9bS)-5-(6-chloro-2H-1,3-benzodioxol-5-yl)-2-cyclopentyl-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-[3-(pyridine-2-carbonyl)piperidin-1-yl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethan-1-one
2-{1-[(4-ethoxyphenyl)methyl]-4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperazin-2-yl}ethan-1-ol
(1R,5R)-3-(2,6,8-trimethylquinoline-4-carbonyl)-3,9-diazabicyclo[3.3.2]decan-10-one
1-{3-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidine-1-carbonyl}cyclopropan-1-amine
N4-{[5-(4-methoxyphenyl)-1,2-oxazol-3-yl]methyl}-5,6-dimethylpyrimidine-2,4-diamine
methyl 4-({5-[(isoquinolin-5-yloxy)methyl]-1,2-oxazol-3-yl}formamido)butanoate
3-[(3R,4S)-4-(morpholin-4-yl)-1-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]piperidin-3-yl]propan-1-ol
1-[2-(3-methyl-3-phenylpiperidin-1-yl)-2-oxoethyl]-1,2-dihydropyridin-2-one
N-[(1-{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}piperidin-3-yl)methyl]acetamide
methyl 2-[(oxolan-2-ylmethyl)sulfamoyl]-6-{[4-(propan-2-yl)phenyl]methyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-(1-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)-N-[(2-fluorophenyl)methyl]propanamide
3-ethyl-N-[3-(3-oxopiperazin-1-yl)propyl]-1H-indole-2-carboxamide
methyl 3-[(5-ethylfuran-2-yl)methyl]-7-oxo-9-(3-phenylpropoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-({5-methyl-2-[2-(3-phenoxypropanamido)phenyl]-1,3-oxazol-4-yl}methyl)-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
2-methoxy-N-(1-{7-[(4-methoxy-2,5-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)acetamide
1-{3-[(3,4-difluorophenyl)amino]piperidin-1-yl}-3-(5-methyl-1H-pyrazol-1-yl)propan-1-one
N-(1H-1,3-benzodiazol-2-ylmethyl)-2-(thiomorpholin-4-yl)-6-(thiophen-3-yl)pyridine-3-carboxamide
1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-8-(pyridin-2-yl)-1,8-diazaspiro[4.5]decane
(2S,4S,5R)-4-[ethyl(methyl)carbamoyl]-1,2-dimethyl-5-phenylpyrrolidine-2-carboxylic acid
2-(5-chloro-1H-1,3-benzodiazol-2-yl)-1-[(3S,4S)-3,4-dihydroxy-4-methylpiperidin-1-yl]ethan-1-one