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N,N-dimethyl-2-{[2-methyl-2-(morpholin-4-yl)propanamido]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
1-{[2-(ethanesulfonyl)-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}-4-(2-methoxyethyl)piperazine
2-methyl-4-phenyl-N-[(3R)-pyrrolidin-3-yl]pyrimidine-5-carboxamide
6-{[3-(furan-2-yl)phenyl]methyl}-N-methyl-N-(1,3-thiazol-4-ylmethyl)-6-azaspiro[2.5]octane-1-carboxamide
3-(5-{3,6-dimethyl-[1,2]oxazolo[5,4-b]pyridine-4-carbonyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl)pyridine
N-[1-(2,5-difluorophenyl)cyclopropyl]-5-[(4-methylpiperazin-1-yl)methyl]furan-2-carboxamide
2-[5-(1-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}pyrrolidin-2-yl)-1,2,4-oxadiazol-3-yl]pyridine
N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
N-(furan-2-ylmethyl)-1-(2-oxo-1,2-dihydroquinoline-4-carbonyl)piperidine-4-carboxamide
5-(5-methylfuran-2-yl)-3-[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]-1,2,4-triazine
5-{[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]methyl}-2-(pyridin-2-yl)pyrimidine
N-(1-methyl-3-phenyl-1H-pyrazol-5-yl)-4-(pyrimidin-2-yloxy)piperidine-1-carboxamide
2-(1-benzothiophen-2-ylmethyl)-4-[4-(piperidine-1-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
2-methyl-2-[4-(morpholin-4-yl)-2-{octahydropyrrolo[1,2-a]piperazin-2-yl}pyrimidin-5-yl]propanoic acid
[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl](methyl)({2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)amine
1-[1'-(3,5-difluorobenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
methyl[3-(5-methylfuran-2-yl)butyl]{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}amine
6-{[9-oxo-8-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-2-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-chloro-N-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-2-propanamidobenzamide
{[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
5-[1-(4-chlorophenyl)cyclobutyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
3-(1H-imidazol-2-yl)-1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]piperidine
9-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-3,9-diazaspiro[5.6]dodecane
3-(1-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl)-4-methyl-1,2,5-oxadiazole
N-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-3-(2-hydroxyphenyl)-N-methyl-1H-pyrazole-5-carboxamide
N-[(4-ethoxyphenyl)methyl]-N-(2-methoxyethyl)-2,8-diazaspiro[4.5]decane-3-carboxamide
1-ethyl-2-oxo-N-[1-(4-propoxyphenyl)ethyl]-1,2-dihydropyridine-4-carboxamide
(3S,4R)-N,N-dimethyl-4-(propan-2-yl)-1-[2-(trifluoromethyl)benzoyl]pyrrolidin-3-amine
2-[3-oxo-9-(9H-purin-6-yl)-2,9-diazaspiro[5.5]undecan-2-yl]acetic acid
1-(4-{2-[benzyl(methyl)amino]-2,3-dihydro-1H-indene-2-carbonyl}-1,4-diazepan-1-yl)ethan-1-one
N-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-2-methyl-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
2-ethyl-5-{[4-(pyridin-3-ylmethyl)piperazin-1-yl]methyl}pyrimidine
2-[4-(2-phenoxyethyl)piperazin-1-yl]-4-(pyridin-4-yl)pyrimidine
N-(furan-2-ylmethyl)-N,7-dimethylimidazo[1,2-a]pyridine-2-carboxamide
2-{methyl[(4-phenoxyphenyl)methyl]amino}-1,3-thiazole-4-carboxamide
(1R,9S)-5-amino-3-(2-methoxypyrimidin-5-yl)-12-methyl-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-triene-4-carbonitrile
ethyl 1-({3-[(1-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}piperidin-4-yl)oxy]phenyl}methyl)piperidine-2-carboxylate
N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]naphthalene-1-carboxamide
methyl 2-[(2,3-dihydro-1H-inden-5-yl)sulfamoyl]-6-[(2-hydroxyphenyl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
[(2S,4R,5R)-4-{[(2H-1,3-benzodioxol-4-ylmethyl)amino]methyl}-5-(4-chlorophenyl)-1-ethyl-2-methylpyrrolidin-2-yl]methanol
1-[2-(2,2-diphenylethyl)morpholin-4-yl]-3-(1,2-oxazolidin-2-yl)propan-1-one
1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
1-[6-(3-chlorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-1,4-diazepan-5-one
(1S,5R)-3-benzyl-6-(4-methyl-1,3-thiazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-[2-(3-acetyl-2,4,6-trimethylphenyl)-1H-imidazol-1-yl]acetamide
2-[3,5-dimethyl-4-(4-phenoxybenzenesulfonamido)-1H-pyrazol-1-yl]acetic acid
3-{[3-(dimethylamino)propyl](methyl)amino}-N-[2-(trifluoromethyl)phenyl]piperidine-1-carboxamide
1-{4-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]phenyl}ethan-1-one
4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(2-fluorobenzoyl)piperidine
N-propyl-5-{1-[2-(pyridin-2-yl)acetyl]pyrrolidin-2-yl}thiophene-2-carboxamide