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2-{1-benzyl-4-[(6-fluoroquinolin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
1-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]-4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}piperidin-4-ol
5-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
3-{[(2-methoxy-2-methylpropyl)carbamoyl]methyl}-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
5-{1-[(6-methyl-4-oxo-4H-chromen-3-yl)methyl]pyrrolidin-2-yl}thiophene-2-carboxamide
1,5-dimethyl-N-[(2-phenoxypyridin-3-yl)methyl]-1H-pyrazole-3-carboxamide
4,6-dimethyl-N-{[3-(pyrrolidin-1-ylmethyl)phenyl]methyl}pyrimidin-2-amine
2-(1H-indol-3-yl)-N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]acetamide
7-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(thiophen-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-(1-acetylazepan-3-yl)-2-[(2-methoxyethyl)amino]-1-methyl-1H-1,3-benzodiazole-5-carboxamide
N-[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]-3-(3-hydroxy-3-methylbutyl)benzamide
2-amino-3-ethyl-N-[2-(propylsulfanyl)ethyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
N-[2-(dimethylamino)ethyl]-N-methyl-1-{3-methyl-3H-[1,2,3]triazolo[4,5-b]pyridine-6-carbonyl}piperidin-3-amine
(4aR,7aS)-1-methyl-4-[2-(1H-pyrazol-1-yl)benzoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-4-(4-methylphenoxy)piperidine-4-carboxamide
N-[(2,4-dimethoxyphenyl)methyl]-2-(pyrrolidin-3-yl)acetamide
1-[(4aS,8aR)-4a-(hydroxymethyl)-decahydro-1,6-naphthyridin-6-yl]-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethan-1-one
4-(1H-1,3-benzodiazol-1-yl)-1-(cyclopropanesulfonyl)piperidine-4-carboxylic acid
1-[3-methoxy-5-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-3-methyl-3-[1-(1,2-oxazol-3-yl)ethyl]urea
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-acetamidopropanamide
(2E)-N-(2H-1,3-benzodioxol-5-ylmethyl)-3-(3-fluorophenyl)-N-{[2-(4-hydroxypiperidin-1-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}prop-2-enamide
2-chloro-4-fluoro-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]benzamide
7-(5-chloropyridin-2-yl)-4-[(2R)-pyrrolidine-2-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-(propan-2-yl)-5-[4-(pyrimidin-2-yl)piperazine-1-carbonyl]-1,3-benzoxazole
N-(5-carbamoyl-2-methylphenyl)-6-hydroxy-1,4-oxazepane-4-carboxamide
3-methyl-6-(5-{1-[2-(propan-2-yl)-1H-imidazol-1-yl]ethyl}-1,2,4-oxadiazol-3-yl)pyridazine
9-methoxy-4-(naphthalen-2-ylmethyl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-(3-methoxypropyl)-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]acetamide
1-(4-{[3-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
7-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-1,2-dihydroisoquinolin-1-one
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-5-(3-hydroxy-3-methylbut-1-yn-1-yl)furan-2-carboxamide
methyl (2S)-2-phenyl-2-({5-[3-(trifluoromethyl)phenoxymethyl]-1,2-oxazol-3-yl}formamido)acetate
2-{[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]amino}-N-(1,3-thiazol-2-yl)propanamide
N-[4-(2-fluorophenoxy)phenyl]-1-(3-hydroxy-2,2-dimethylpropyl)piperidine-4-carboxamide
3-(azetidine-1-carbonyl)-1-[1-(2-phenylethyl)piperidin-4-yl]piperidine
7-fluoro-2-{2-methylimidazo[1,2-a]pyridine-6-carbonyl}-1,2,3,4-tetrahydroisoquinoline
N-[3-(3-chlorophenyl)phenyl]-1-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperidine-4-carboxamide
7-(cyclopropylmethyl)-N-(2-methoxy-2-methylpropyl)-6-(4-methoxyphenyl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2-(2-{4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-1-yl}-2-oxoethyl)-2,3-dihydro-1,2-benzothiazol-3-one
N-{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N-methyloxolan-3-amine
(4-{[(2S,5R)-5-{[(furan-3-ylmethyl)(methyl)amino]methyl}oxolan-2-yl]methyl}phenyl)methanol
naphthalen-1-yl (7S,9aR)-7-(cyclohexylmethyl)-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
1-[2-({[3-(methylsulfanyl)propyl]amino}methyl)phenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidin-2-one
3-{4-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrole-5-carbonyl]phenyl}-1H-pyrazole
9-[(5-propylfuran-2-yl)methyl]-2-[(1r,4r)-4-hydroxycyclohexyl]-2,9-diazaspiro[5.5]undecan-3-one
1-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-5-(2-{[(3-methoxyphenyl)methyl]amino}ethyl)pyrrolidin-2-one
({4-cyclopropyl-5-[1-(3-fluoropyridin-4-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
N-cyclohexyl-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)butanamide
2-[(3-methoxyphenyl)methyl]-4-{[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}morpholine