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5-methyl-N-(3-{5-methyl-4-[(2-phenoxyacetamido)methyl]-1,3-oxazol-2-yl}phenyl)thiophene-2-carboxamide
1-ethyl-N,5-dimethyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1H-pyrazole-3-carboxamide
N-[1-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
4-{4-[3-(2-chlorophenyl)propanoyl]-2-oxopiperazin-1-yl}benzonitrile
ethyl 2-[6-oxo-4-(pyrrolidin-1-yl)-1,6-dihydropyridazin-1-yl]pentanoate
1-{3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}-2-(1H-imidazol-1-yl)ethan-1-one
diethyl({[3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)pyrazolo[1,5-a]pyrimidin-6-yl]methyl})amine
N-{[5-methyl-7-(2-methylquinolin-6-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}oxane-4-carboxamide
8-chloro-4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-2-methylquinoline
N-[(1S,2R,4R)-bicyclo[2.2.1]heptan-2-yl]-5-(2-fluorophenoxymethyl)-1H-pyrazole-3-carboxamide
N-{1-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
1-[3-(1H-imidazol-2-yl)benzoyl]-2-methyl-4-(2-methylphenyl)piperazine
1-[5-(4-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]-3-methoxypiperidine
3-{2-ethyl-3-oxo-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-N,N-dimethylpropanamide
N-(2-oxopiperidin-3-yl)-3-(trimethyl-1H-pyrazol-4-yl)propanamide
N-(2-{7-[(3,4-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-4-methoxybenzamide
N-methyl-5-[3-(1H-pyrazol-1-ylmethyl)benzoyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-3-carboxamide
3-oxo-2-(3-phenylpropyl)-N-propyl-2,8-diazaspiro[4.5]decane-8-carboxamide
3-(2-chlorophenoxy)-1-(2-fluoro-4-methylbenzoyl)azetidine
(4aR,8aR)-4a-hydroxy-7-(4-methoxypyrimidin-2-yl)-N,N-dimethyl-decahydro-2,7-naphthyridine-2-sulfonamide
N-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-3-(piperidin-3-yl)benzamide
2-[(thiophen-2-ylmethyl)[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]amino]ethan-1-ol
ethyl 2-(1-{3-[2-(2H-1,3-benzodioxol-5-ylmethyl)-5-oxopyrrolidin-2-yl]propanoyl}piperidin-2-yl)acetate
N-({5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl}methyl)pyridine-4-carboxamide
1-[5-(methoxymethyl)furan-2-carbonyl]-3-[2-(3-methoxyphenyl)ethyl]piperidine
2-(4-fluorophenyl)-N-(2-methoxyethyl)-N-methylimidazo[1,2-a]pyridine-6-carboxamide
1-[(3,4-dimethylphenyl)methyl]-4-(2-methyl-1,3-thiazole-5-carbonyl)piperazin-2-one
(1S,5R)-N-butyl-7-oxo-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
7-(1,3-benzothiazol-2-yl)-4-[(2-ethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-{[3-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]methyl}benzonitrile
2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methylacetamide
1-[4-({4-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperazin-1-yl]ethan-1-one
3-[(3R,4S)-1-[2-(2,3-dihydro-1H-isoindol-2-yl)acetyl]-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
ethyl 1-(4-methyl-1,3-oxazole-5-carbonyl)-3-(3-phenylpropyl)piperidine-3-carboxylate
3-[(1-acetylpiperidin-4-yl)oxy]-4-methoxy-N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]benzamide
methyl (2S,4R)-4-(2,3-dimethyl-1H-indole-7-amido)-1-[(2-fluorophenyl)methyl]pyrrolidine-2-carboxylate
1-cyclopentyl-N-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)-6-oxopiperidine-3-carboxamide
3-{[1-(ethanesulfonyl)piperidin-4-yl]oxy}-N-(pyridin-2-ylmethyl)benzamide
2-[(3R,4S)-3-(3-hydroxypropanamido)-4-propylpyrrolidin-1-yl]-N-methylpyridine-3-carboxamide
methyl 2-({1-[2-(3-fluorophenyl)ethyl]-6-oxopiperidin-3-yl}formamido)acetate
3-{imidazo[1,2-a]pyridin-2-yl}-1-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]propan-1-one
4-({4-phenyl-5-[(1,3-thiazol-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)piperidine
3-(3,4-dimethoxyphenyl)-N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}propanamide
N-ethyl-4-[(1-methoxybutan-2-yl)amino]-5-methyl-N-(2-methylprop-2-en-1-yl)thieno[2,3-d]pyrimidine-6-carboxamide
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-2-methyl-1,3-thiazole-4-carboxamide
methyl 2-[(4-{1-[4-(dimethylamino)butanoyl]piperidin-4-yl}-5-(3-methoxyphenyl)pyrimidin-2-yl)sulfanyl]acetate
ethyl 2-{1-[2-(methylsulfanyl)pyrimidine-5-carbonyl]piperidin-2-yl}acetate
6-methyl-2-[1-(pyrazine-2-carbonyl)pyrrolidin-2-yl]-1H-1,3-benzodiazole
N-{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-1H-indazole-3-carboxamide
6-methyl-2-({4-[6-(propan-2-yl)pyridin-2-yl]piperazin-1-yl}methyl)pyridin-3-ol